ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 49. Synthesis of Substituted Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides with Increased Affinities for Isozyme I.

C. T. SUPURAN; A. SCOZZAFAVA; B. C. JURCA; M. A. ILIES

doi:10.1002/chin.199829111

ChemInform Abstract: Carbonic Anhydrase Inhibitors. Part 49. Synthesis of Substituted Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides with Increased Affinities for Isozyme I.

ChemInform ◽

10.1002/chin.199829111 ◽

2010 ◽

Vol 29 (29) ◽

pp. no-no

Author(s):

C. T. SUPURAN ◽

A. SCOZZAFAVA ◽

B. C. JURCA ◽

M. A. ILIES

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of ◽

Aromatic Heterocyclic

Download Full-text

QSAR Studies on Carbonic Anhydrase Inhibitors: A Case of Ureido and Thioureido Derivatives of Aromatic/Heterocyclic Sulfonamides

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00123-2 ◽

2002 ◽

Vol 10 (9) ◽

pp. 2993-2999 ◽

Cited By ~ 19

Author(s):

Vijay K. Agrawal ◽

Ruchi Sharma ◽

Padmakar V. Khadikar

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Qsar Studies ◽

Derivatives Of ◽

Aromatic Heterocyclic

Download Full-text

Carbonic anhydrase inhibitors - Part 49: Synthesis of substituted ureido and thioureido derivatives of aromatic/heterocyclic sulfonamides with increased affinities for isozyme I

European Journal of Medicinal Chemistry ◽

10.1016/s0223-5234(98)80033-0 ◽

1998 ◽

Vol 33 (2) ◽

pp. 83-93 ◽

Cited By ~ 113

Author(s):

Claudiu T. Supuran ◽

Andrea Scozzafava ◽

Bogdan C. Jurca ◽

Marc A. Ilies

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of ◽

Aromatic Heterocyclic

Download Full-text

Carbonic Anhydrase Inhibitors: Perfluoroalkyl/Aryl-Substituted Derivatives of Aromatic/Heterocyclic Sulfonamides as Topical Intraocular Pressure-Lowering Agents with Prolonged Duration of Action

Journal of Medicinal Chemistry ◽

10.1021/jm000296j ◽

2000 ◽

Vol 43 (23) ◽

pp. 4542-4551 ◽

Cited By ~ 90

Author(s):

Andrea Scozzafava ◽

Luca Menabuoni ◽

Francesco Mincione ◽

Fabrizio Briganti ◽

Giovanna Mincione ◽

...

Keyword(s):

Intraocular Pressure ◽

Carbonic Anhydrase ◽

Duration Of Action ◽

Carbonic Anhydrase Inhibitors ◽

Prolonged Duration ◽

Pressure Lowering ◽

Derivatives Of ◽

Aromatic Heterocyclic ◽

Aryl Substituted Derivatives

Download Full-text

Carbonic anhydrase inhibitors – part 70. Synthesis and ocular pharmacology of a new class of water-soluble, topically effective intraocular pressure lowering agents derived from nicotinic acid and aromatic/heterocyclic sulfonamides

European Journal of Medicinal Chemistry ◽

10.1016/s0223-5234(99)00212-3 ◽

1999 ◽

Vol 34 (10) ◽

pp. 799-808 ◽

Cited By ~ 9

Author(s):

C Supuran

Keyword(s):

Intraocular Pressure ◽

Carbonic Anhydrase ◽

Nicotinic Acid ◽

Water Soluble ◽

Carbonic Anhydrase Inhibitors ◽

New Class ◽

Pressure Lowering ◽

Aromatic Heterocyclic ◽

Ocular Pharmacology

Download Full-text

Bioorganometallic derivatives of 4-hydrazino-benzenesulphonamide as carbonic anhydrase inhibitors: synthesis, characterisation and biological evaluation

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2020.1724995 ◽

2020 ◽

Vol 35 (1) ◽

pp. 622-628 ◽

Cited By ~ 2

Author(s):

Jeremie Brichet ◽

Rodrigo Arancibia ◽

Emanuela Berrino ◽

Claudiu T. Supuran

Keyword(s):

Carbonic Anhydrase ◽

Biological Evaluation ◽

Carbonic Anhydrase Inhibitors ◽

Derivatives Of

Download Full-text

Carbonic anhydrase inhibitors: Copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.11.025 ◽

2008 ◽

Vol 18 (2) ◽

pp. 836-841 ◽

Cited By ~ 26

Author(s):

Marouan Rami ◽

Jean-Yves Winum ◽

Alessio Innocenti ◽

Jean-Louis Montero ◽

Andrea Scozzafava ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Aromatic Heterocyclic

Download Full-text

Carbonic anhydrase inhibitors. Part 36. Inhibition of isozymes I and II with Schiff bases derived from chalkones and aromatic/heterocyclic sulfonamides

European Journal of Medicinal Chemistry ◽

10.1016/0223-5234(96)85164-6 ◽

1996 ◽

Vol 31 (6) ◽

pp. 439-447 ◽

Cited By ~ 54

Author(s):

CT Supuran ◽

A Popescu ◽

M Ilisiu ◽

A Costandache ◽

MD Banciu

Keyword(s):

Carbonic Anhydrase ◽

Schiff Bases ◽

Carbonic Anhydrase Inhibitors ◽

Aromatic Heterocyclic

Download Full-text

A quantitative structure–activity relationship study on some aromatic/heterocyclic sulfonamides and their charged derivatives acting as carbonic anhydrase inhibitors

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360500067439 ◽

2005 ◽

Vol 20 (3) ◽

pp. 251-259 ◽

Cited By ~ 5

Author(s):

S. P. Gupta ◽

S. Kumaran

Keyword(s):

Carbonic Anhydrase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Carbonic Anhydrase Inhibitors ◽

Structure Activity ◽

Relationship Study ◽

Aromatic Heterocyclic

Download Full-text

QSAR study on carbonic anhydrase inhibitors: aromatic/heterocyclic sulfonamides containing 8-quinoline-sulfonyl moieties, with topical activity as antiglaucoma agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2004.03.002 ◽

2004 ◽

Vol 39 (7) ◽

pp. 593-600 ◽

Cited By ~ 28

Author(s):

Vijay K Agrawal ◽

Shahnaz Bano ◽

Claudiu T Supuran ◽

Padmakar V Khadikar

Keyword(s):

Carbonic Anhydrase ◽

Qsar Study ◽

Carbonic Anhydrase Inhibitors ◽

Antiglaucoma Agents ◽

Aromatic Heterocyclic

Download Full-text

Carbonic anhydrase inhibitors. Aromatic/heterocyclic sulfonamides incorporating phenacetyl, pyridylacetyl and thienylacetyl tails act as potent inhibitors of human mitochondrial isoforms VA and VB

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.06.006 ◽

2009 ◽

Vol 17 (14) ◽

pp. 4894-4899 ◽

Cited By ~ 31

Author(s):

Özlen Güzel ◽

Alessio Innocenti ◽

Andrea Scozzafava ◽

Aydın Salman ◽

Claudiu T. Supuran

Keyword(s):

Carbonic Anhydrase ◽

Carbonic Anhydrase Inhibitors ◽

Aromatic Heterocyclic

Download Full-text