ChemInform Abstract: Stereocontrolled Synthesis of Pseudo C2-Symmetric 1,3-Diamino-2- propanol Core Units of HIV Protease Inhibitors.

A. DONDONI; D. PERRONE

doi:10.1002/chin.199718113

ChemInform Abstract: Stereocontrolled Synthesis of Pseudo C2-Symmetric 1,3-Diamino-2- propanol Core Units of HIV Protease Inhibitors.

ChemInform ◽

10.1002/chin.199718113 ◽

2010 ◽

Vol 28 (18) ◽

pp. no-no

Author(s):

A. DONDONI ◽

D. PERRONE

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis

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ChemInform Abstract: Transition-State Mimetics for HIV Protease Inhibitors: Stereocontrolled Synthesis of Hydroxyethylene and Hydroxyethylamine Isosteres by Ester-Derived Titanium Enolate syn and anti-Aldol Reactions.

ChemInform ◽

10.1002/chin.199905090 ◽

2010 ◽

Vol 30 (5) ◽

pp. no-no

Author(s):

A. K. GHOSH ◽

S. FIDANZE

Keyword(s):

Transition State ◽

Protease Inhibitors ◽

Hiv Protease ◽

Aldol Reactions ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis ◽

Hydroxyethylamine Isosteres

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Stereocontrolled synthesis of C2-symmetric and pseudo-C2-symmetric diamino alcohols and diols for use in HIV protease inhibitors

The Journal of Organic Chemistry ◽

10.1021/jo00047a023 ◽

1992 ◽

Vol 57 (21) ◽

pp. 5692-5700 ◽

Cited By ~ 53

Author(s):

Dale J. Kempf ◽

Thomas J. Sowin ◽

Elizabeth M. Doherty ◽

Steven M. Hannick ◽

LynnMarie Codavoci ◽

...

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis

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Stereocontrolled synthesis of pseudo C2-symmetric 1,3-diamino-2-propanol core units of HIV protease inhibitors

Tetrahedron Letters ◽

10.1016/s0040-4039(96)02355-6 ◽

1997 ◽

Vol 38 (3) ◽

pp. 499-502 ◽

Cited By ~ 8

Author(s):

Alessandro Dondoni ◽

Daniela Perrone

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis

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ChemInform Abstract: CrCl2 Mediated Addition of Allylic Halides or Phosphates to N- Protected α-Amino Aldehydes. Stereocontrolled Synthesis of a New Core for C2 Symmetric HIV-Protease Inhibitors.

ChemInform ◽

10.1002/chin.199638054 ◽

2010 ◽

Vol 27 (38) ◽

pp. no-no

Author(s):

P. CIAPETTI ◽

M. FALORNI ◽

M. TADDEI

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Amino Aldehydes ◽

Stereocontrolled Synthesis ◽

Allylic Halides

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ChemInform Abstract: Stereocontrolled Synthesis of C2-Symmetric and Pseudo-C2-Symmetric Diamino Alcohols and Diols for Use in HIV Protease Inhibitors.

ChemInform ◽

10.1002/chin.199307101 ◽

2010 ◽

Vol 24 (7) ◽

pp. no-no

Author(s):

D. J. KEMPF ◽

T. J. SOWIN ◽

E. M. DOHERTY ◽

S. M. HANNICK ◽

L. CODAVOCI ◽

...

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis

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Transition-State Mimetics for HIV Protease Inhibitors: Stereocontrolled Synthesis of Hydroxyethylene and Hydroxyethylamine Isosteres by Ester-Derived Titanium Enolate Syn and Anti-Aldol Reactions

The Journal of Organic Chemistry ◽

10.1021/jo980159i ◽

1998 ◽

Vol 63 (18) ◽

pp. 6146-6152 ◽

Cited By ~ 44

Author(s):

Arun K. Ghosh ◽

Steve Fidanze

Keyword(s):

Transition State ◽

Protease Inhibitors ◽

Hiv Protease ◽

Aldol Reactions ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis ◽

Hydroxyethylamine Isosteres

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Concise and Stereocontrolled Synthesis of Pseudo-C2-symmetric Diamino Alcohols and Triamines for Use in HIV Protease Inhibitors

The Journal of Organic Chemistry ◽

10.1021/jo026616j ◽

2003 ◽

Vol 68 (4) ◽

pp. 1418-1425 ◽

Cited By ~ 19

Author(s):

Luca Bernardi ◽

Bianca F. Bonini ◽

Gabriella Dessole ◽

Mariafrancesca Fochi ◽

Mauro Comes-Franchini ◽

...

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Stereocontrolled Synthesis

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CrCl2 Mediated addition of allylic halides or phosphates to N-protected α-amino aldehydes. Stereocontrolled synthesis of a new core for C2 symmetric HIV-protease inhibitors

Tetrahedron ◽

10.1016/0040-4020(96)00258-x ◽

1996 ◽

Vol 52 (21) ◽

pp. 7379-7390 ◽

Cited By ~ 18

Author(s):

Paola Ciapetti ◽

Massimo Falorni ◽

Maurizio Taddei

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Amino Aldehydes ◽

Stereocontrolled Synthesis ◽

Allylic Halides

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Determining and Overcoming Resistance to HIV Protease Inhibitors

Current Drug Targets - Infectious Disorders ◽

10.2174/1568005043340984 ◽

2004 ◽

Vol 4 (2) ◽

pp. 137-152 ◽

Cited By ~ 17

Author(s):

Jana Prejdova ◽

Milan Soucek ◽

Jan Konvalinka

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors

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A QSAR Study of HIV Protease Inhibitors Using Theoretical Descriptors

Current Computer - Aided Drug Design ◽

10.2174/1573409911006040269 ◽

2010 ◽

Vol 6 (4) ◽

pp. 269-282 ◽

Cited By ~ 4

Author(s):

Subhash C. Basak ◽

Denise Mills ◽

Rajni Garg ◽

Barun Bhhatarai

Keyword(s):

Protease Inhibitors ◽

Hiv Protease ◽

Hiv Protease Inhibitors ◽

Qsar Study

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