ChemInform Abstract: Facile Synthesis of β-Phenylethylamine Derivatives Related to Baclofen via Aziridine Ring Opening.

ChemInform ◽  
1990 ◽  
Vol 21 (37) ◽  
Author(s):  
R. D. ALLAN ◽  
H. W. TRAN
Keyword(s):  
Ring Opening ◽  
Facile Synthesis ◽  
Aziridine Ring

Chiral aziridine ring opening: facile synthesis of (R)-mexiletine and (R)-phenoxybenzamine hydrochloride

2015 ◽  
Vol 56 (38) ◽  
pp. 5269-5271 ◽  
Author(s):  
N. Viswanadh ◽  
R. Velayudham ◽  
S. Jambu ◽  
M. Sasikumar ◽  
M. Muthukrishnan
Keyword(s):  
Ring Opening ◽  
Facile Synthesis ◽  
Aziridine Ring

Chemistry of Tetrathiomolybdate:  Aziridine Ring Opening Reactions and Facile Synthesis of Interesting Sulfur Heterocycles

2005 ◽  
Vol 127 (37) ◽  
pp. 12760-12761 ◽  
Author(s):  
Devarajulu Sureshkumar ◽  
Srinivasa Murthy Koutha ◽  
Srinivasan Chandrasekaran
Keyword(s):  
Ring Opening ◽  
Facile Synthesis ◽  
Aziridine Ring ◽  
Ring Opening Reactions ◽  
Sulfur Heterocycles

Facile Synthesis of β-Phenylethylamine Derivatives Related to Baclofen via Aziridine Ring Opening

1990 ◽  
Vol 43 (6) ◽  
pp. 1123 ◽  
Author(s):  
RD Allan ◽  
HW Tran
Keyword(s):  
Ring Opening ◽  
Receptor Agonist ◽  
Gabab Receptor ◽  
Facile Synthesis ◽  
Aziridine Ring ◽  
Simple Route ◽  
Nucleophilic Ring Opening

Nucleophilic ring opening of the protonated salt of 2-(4-chlorophenyl ) aziridine with substituted thiols provides a very simple route to β- phenylethylamine derivatives which are analogues of the GABAB receptor agonist baclofen and its antagonists phaclofen and saclofen.

scholarly journals Intramolecular N–Me and N–H aminoetherification for the synthesis of N-unprotected 3-amino-O-heterocycles

2021 ◽  
Author(s):  
Mahesh P. Paudyal ◽  
Mingliang Wang ◽  
Juha H. Siitonen ◽  
Yimin Hu ◽  
Muhammed Yousufuddin ◽  
...  
Keyword(s):  
Ring Opening ◽  
Domino Reaction ◽  
Aziridine Ring

A mild Rh-catalyzed method for synthesis of cyclic unprotected N–Me and N–H 2,3-aminoethers using an olefin aziridination–aziridine ring-opening domino reaction has been developed.

Stereoselective Syntheses of 4-Oxa Diaminopimelic Acid and Its Protected Derivatives via Aziridine Ring Opening

2007 ◽  
Vol 9 (21) ◽  
pp. 4211-4214 ◽  
Author(s):  
Hongqiang Liu ◽  
Vijaya R. Pattabiraman ◽  
John C. Vederas
Keyword(s):  
Ring Opening ◽  
Diaminopimelic Acid ◽  
Aziridine Ring ◽  
Stereoselective Syntheses

ChemInform Abstract: Divergent Reactions of Indoles with Aminobenzaldehydes: Indole Ring-Opening vs. Annulation and Facile Synthesis of Neocryptolepine.

ChemInform ◽  
2012 ◽  
Vol 43 (9) ◽  
pp. no-no
Author(s):  
Matthew K. Vecchione ◽  
Aaron X. Sun ◽  
Daniel Seidel ◽  
et al. et al.
Keyword(s):  
Ring Opening ◽  
Indole Ring ◽  
Facile Synthesis

Tandem Ring Opening/Cyclization of Vinylcyclopropanes: A Facile Synthesis of Chiral Bicyclic Amidines

2011 ◽  
Vol 123 (26) ◽  
pp. 6000-6003 ◽  
Author(s):  
Venkataraman Ganesh ◽  
Devarajulu Sureshkumar ◽  
Srinivasan Chandrasekaran
Keyword(s):  
Ring Opening ◽  
Facile Synthesis

Neutral lutetium complex/polyamine mediated immortal ring-opening polymerization of rac-lactide: facile synthesis of well-defined hydroxyl-end and amide-core stereoregular star polylactide

2015 ◽  
Vol 6 (44) ◽  
pp. 7711-7716 ◽  
Author(s):  
Wei Zhao ◽  
Bo Liu ◽  
Xinli Liu ◽  
Xue Wang ◽  
Yang Wang ◽  
...  
Keyword(s):  
Ring Opening ◽  
Ring Opening Polymerization ◽  
Facile Synthesis

A facile way to obtain well-defined hydroxyl-end and amide-core stereoregular star polylactide.

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