ChemInform Abstract: Transformations of Amino Acids. Part 2. Reaction of 3-Thiazolines with Carboxylic Acid Chlorides.

ChemInform ◽  
1987 ◽  
Vol 18 (44) ◽  
Author(s):  
W. SCHWARZE ◽  
K. DRAUZ ◽  
J. MARTENS
Keyword(s):  
Amino Acids ◽  
Carboxylic Acid ◽  
Acid Chlorides

Synthesis and Antibacterial Potency of 4-Methyl-2,7-dioxo-1,2,3,4,7,10- hexahydropyrido[2,3-ƒ]quinoxaline-8-carboxylic acid, Selected [a]-Fused Heterocyles and Acyclic Precursors

2007 ◽  
Vol 62 (11) ◽  
pp. 1453-1458 ◽  
Author(s):  
Yusuf M. Al-Hiari ◽  
Ali M. Qaisia ◽  
Mohammad Y.Abu Shuheil ◽  
Mustafa M. El-Abadelah ◽  
Wolfgang Voelter
Keyword(s):  
Amino Acids ◽  
Carboxylic Acid ◽  
Antibacterial Activities ◽  
Sodium Dithionite ◽  
E Coli ◽  
Pipecolinic Acid

The reaction of 7-chloro-1-cyclopropyl-6-fluoro-8-nitro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid (7) with each of sarcosine and (±)-pipecolinic acid afforded the corresponding N-(4- oxoquinolin-7-yl)-α-amino acids 8 and 9. Reductive lactamization of the latter with sodium dithionite gave hexahydropyrido[2,3- f ]quinoxaline (10) and octahydrodipyrido[1,2-a : 2,3- f ]quinoxaline (11) derivatives, respectively. Compounds 8 - 11 and their homologs 1 - 6, accessible from (S)-proline, (2S, 4R)-4-hydroxyproline and (S)-tetrahydroisoquinoline-3-carboxylic acid exhibit good to excellent antibacterial activities against E. coli and S. aureus.

scholarly journals Synthesis and Characterization of the Germathioacid Chloride Coordinated by an N-Heterocyclic Carbene §

Inorganics ◽  
2018 ◽  
Vol 6 (3) ◽  
pp. 76 ◽  
Author(s):  
Yasunobu Egawa ◽  
Chihiro Fukumoto ◽  
Koichiro Mikami ◽  
Nobuhiro Takeda ◽  
Masafumi Unno
Keyword(s):  
Carboxylic Acid ◽  
Density Functional ◽  
Dft Calculation ◽  
Acid Chlorides ◽  
Carboxylic Acid Chloride ◽  
Functional Theory ◽  
Nitrogen Ligands ◽  
Bond Property ◽  
Nitrogen Bonds

Carboxylic acid chlorides are useful substrates in organic chemistry. Many germanium analogues of carboxylic acid chloride have been synthesized so far. Nevertheless, all of the reported germathioacid chlorides use bidentate nitrogen ligands and contain germanium-nitrogen bonds. Our group synthesized germathioacid chloride, Ge(S)Cl{C6H3-2,6-Tip2}(Im-i-Pr2Me2), using N-heterocyclic carbene (Im-i-Pr2Me2). As a result of density functional theory (DFT) calculation, it was found that electrons are localized on sulfur, and the germanium-sulfur bond is a single bond with a slight double bond property.

Enzymatic resolution of (±)-5-phenyl-4,5-dihydroisoxazole-3-carboxylic acid ethyl ester and its transformations into polyfunctionalised amino acids and dipeptides

2009 ◽  
Vol 20 (16) ◽  
pp. 1940-1947 ◽  
Author(s):  
Giuseppe Cremonesi ◽  
Piero Dalla Croce ◽  
Alessandra Forni ◽  
Maddalena Gallanti ◽  
Raffaella Gandolfi ◽  
...  
Keyword(s):  
Amino Acids ◽  
Carboxylic Acid ◽  
Ethyl Ester ◽  
Acid Ethyl Ester ◽  
Enzymatic Resolution

Acylation of 4,6-diamino-2-mercaptopyrimidine and its salts with carboxylic acid chlorides

1980 ◽  
Vol 29 (10) ◽  
pp. 1662-1665 ◽  
Author(s):  
G. I. Podzigun ◽  
N. G. Pashkurov ◽  
V. S. Reznik ◽  
B. E. Ivanov
Keyword(s):  
Carboxylic Acid ◽  
Acid Chlorides

A synthetic route to highly substituted ketones. Acylations of .alpha. anions of carboxylic acid salts with acid chlorides

1977 ◽  
Vol 42 (7) ◽  
pp. 1189-1194 ◽  
Author(s):  
A. Paul Krapcho ◽  
David S. Kashdan ◽  
E. G. E. Jahngen ◽  
A. J. Lovey
Keyword(s):  
Carboxylic Acid ◽  
Acid Chlorides ◽  
Synthetic Route ◽  
Acid Salts

ChemInform Abstract: Trialkylamine-Mediated Intramolecular Acylation of Alkenes with Carboxylic Acid Chlorides

ChemInform ◽  
2010 ◽  
Vol 41 (39) ◽  
pp. no-no
Author(s):  
Jun-ichi Matsuo ◽  
Takaya Hoshikawa ◽  
Shun Sasaki ◽  
Hiroyuki Ishibashi
Keyword(s):  
Carboxylic Acid ◽  
Acid Chlorides

ChemInform Abstract: REACTION OF TETRAALKYL METHYLENEDIPHOSPHONITES WITH CARBOXYLIC ACID CHLORIDES

1979 ◽  
Vol 10 (35) ◽  
Author(s):  
Z. S. NOVIKOVA ◽  
A. A. PRISHCHENKO ◽  
I. F. LUTSENKO
Keyword(s):  
Carboxylic Acid ◽  
Acid Chlorides
Sign in / Sign up

Export Citation Format

Share Document