Design and Synthesis of Fluorinated and/or Hydroxylated 2‐Arylidene‐1‐indanone Derivatives as an Inhibitor of LPS‐stimulated ROS Production in RAW 264.7 Macrophages with Structure–Activity Relationship Study

Pramila Katila; Aastha Shrestha; Aarajana Shrestha; Ritina Shrestha; Pil‐Hoon Park; Eung‐Seok Lee

doi:10.1002/bkcs.11618

Design and Synthesis of Fluorinated and/or Hydroxylated 2‐Arylidene‐1‐indanone Derivatives as an Inhibitor of LPS‐stimulated ROS Production in RAW 264.7 Macrophages with Structure–Activity Relationship Study

Bulletin of the Korean Chemical Society ◽

10.1002/bkcs.11618 ◽

2018 ◽

Vol 39 (12) ◽

pp. 1432-1441 ◽

Cited By ~ 2

Author(s):

Pramila Katila ◽

Aastha Shrestha ◽

Aarajana Shrestha ◽

Ritina Shrestha ◽

Pil‐Hoon Park ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Raw 264.7 ◽

Ros Production ◽

Raw 264.7 Macrophages ◽

Design And Synthesis ◽

Structure Activity ◽

Relationship Study

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Design, synthesis, and structure-activity relationship study of halogen containing 2-benzylidene-1-indanone derivatives for inhibition of LPS-stimulated ROS production in RAW 264.7 macrophages

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2017.03.049 ◽

2017 ◽

Vol 133 ◽

pp. 121-138 ◽

Cited By ~ 10

Author(s):

Aarajana Shrestha ◽

Hye Jin Oh ◽

Mi Jin Kim ◽

Nirmala Tilija Pun ◽

Til Bahadur Thapa Magar ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Raw 264.7 ◽

Ros Production ◽

Design Synthesis ◽

Raw 264.7 Macrophages ◽

Structure Activity ◽

Relationship Study

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Hydroxyl‐ and Halogen‐containing Chalcones for the Inhibition of LPS‐stimulated ROS Production in RAW 264.7 Macrophages: Design, Synthesis and Structure–Activity Relationship Study

Bulletin of the Korean Chemical Society ◽

10.1002/bkcs.11813 ◽

2019 ◽

Vol 40 (7) ◽

pp. 729-734

Author(s):

Aarajana Shrestha ◽

Aastha Shrestha ◽

Pil‐Hoon Park ◽

Eung‐Seok Lee

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Raw 264.7 ◽

Ros Production ◽

Design Synthesis ◽

Raw 264.7 Macrophages ◽

Structure Activity ◽

Relationship Study

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Inhibition of LPS-stimulated ROS production by fluorinated and hydroxylated chalcones in RAW 264.7 macrophages with structure-activity relationship study

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2017.01.061 ◽

2017 ◽

Vol 27 (5) ◽

pp. 1205-1209 ◽

Cited By ~ 12

Author(s):

Ganesh Bist ◽

Nirmala Tilija Pun ◽

Til Bahadur Thapa Magar ◽

Aarajana Shrestha ◽

Hye Jin Oh ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Raw 264.7 ◽

Ros Production ◽

Raw 264.7 Macrophages ◽

Structure Activity ◽

Relationship Study

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Thieny/Furanyl-hydroxyphenylpropenones as Inhibitors of LPS-induced ROS and NO Production in RAW 264.7 Macrophages, and Their Structure-Activity Relationship Study

Bulletin of the Korean Chemical Society ◽

10.5012/bkcs.2014.35.8.2481 ◽

2014 ◽

Vol 35 (8) ◽

pp. 2481-2486 ◽

Cited By ~ 7

Author(s):

Tara Man Kadayat ◽

Mi Jin Kim ◽

Tae-Gyu Nam ◽

Pil-Hoon Park ◽

Eung-Seok Lee

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

No Production ◽

Raw 264.7 ◽

Raw 264.7 Macrophages ◽

Structure Activity ◽

Relationship Study

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Design and synthesis of novel antimicrobial peptides on the basis of α helical domain of Tenecin 1, an insect defensin protein, and structure–activity relationship study

Peptides ◽

10.1016/j.peptides.2005.08.016 ◽

2006 ◽

Vol 27 (4) ◽

pp. 640-648 ◽

Cited By ~ 24

Author(s):

Hye-sun Ahn ◽

Wonmi Cho ◽

Sun-Hee Kang ◽

Sung-Sin Ko ◽

Mi-Sun Park ◽

...

Keyword(s):

Antimicrobial Peptides ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Design And Synthesis ◽

Helical Domain ◽

Structure Activity ◽

Insect Defensin ◽

Relationship Study

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Design and Synthesis of a Piperidinone Scaffold as an Analgesic through Kappa-Opioid Receptor: Structure–Activity Relationship Study of Matrine Alkaloids

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.c15-00962 ◽

2016 ◽

Vol 64 (5) ◽

pp. 410-419 ◽

Cited By ~ 6

Author(s):

Hiroyoshi Teramoto ◽

Takayasu Yamauchi ◽

Yasushi Terado ◽

Sanae Odagiri ◽

Shigeru Sasaki ◽

...

Keyword(s):

Opioid Receptor ◽

Structure Activity Relationship ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Design And Synthesis ◽

Receptor Structure ◽

Structure Activity ◽

Relationship Study

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Structure Activity Relationship Study and Recent Advances in the Design and Synthesis about Linear Antimicrobial Peptides

Current Medicinal Chemistry - Anti-Infective Agents ◽

10.2174/1568012023354884 ◽

2002 ◽

Vol 1 (3) ◽

pp. 305-318 ◽

Cited By ~ 1

Author(s):

Keun-Hyeung Lee

Keyword(s):

Antimicrobial Peptides ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Design And Synthesis ◽

Structure Activity ◽

Recent Advances ◽

Relationship Study

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Synthesis and Structure-Activity Relationship Study of 2-Substituted- 5-(5-nitro-2-thienyl)-1,3,4-thiadiazoles as Anti-Helicobacter pylori Agents

Letters in Drug Design & Discovery ◽

10.2174/157018009789057599 ◽

2009 ◽

Vol 6 (6) ◽

pp. 468-474 ◽

Cited By ~ 1

Author(s):

Alireza Foroumadi ◽

Somayeh Sedaghat ◽

Saeed Emami ◽

Maryam Yazdanian ◽

Mohammad Moshafi ◽

...

Keyword(s):

Helicobacter Pylori ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study

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Structure-activity relationship study on the bioreduction of AZO dyes byClostridium paraputrificum

Environmental Toxicology and Chemistry ◽

10.1002/etc.5620200304 ◽

2001 ◽

Vol 20 (3) ◽

pp. 479-484

Author(s):

David Moir ◽

Sheila Masson ◽

Ih Chu

Keyword(s):

Azo Dyes ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study

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Synthesis and preliminary structure-activity relationship study of 3-methylquinazolinone derivatives as EGFR inhibitors with enhanced antiproliferative activities against tumour cells

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756366.2021.1933466 ◽

2021 ◽

Vol 36 (1) ◽

pp. 1205-1216

Author(s):

Yan Zhang ◽

Qin Wang ◽

Luolan Li ◽

Yi Le ◽

Li Liu ◽

...

Keyword(s):

Structure Activity Relationship ◽

Tumour Cells ◽

Egfr Inhibitors ◽

Activity Relationship ◽

Structure Activity ◽

Relationship Study ◽

Antiproliferative Activities

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