scholarly journals Study of Cationic and Nonionic Mixed Micelles with NaBr and 3,5-Cl2C6H3CO2Na by Use of Probe Nucleophilic Reaction of Piperidine with Ionized Phenyl Salicylate

2018 ◽  
Vol 67 (1) ◽  
pp. 55-66
Author(s):  
Ibrahim Isah Fagge ◽  
Khalisanni Khalid ◽  
Muhammad Azri Mohd Noh ◽  
Nor Saadah Muhammad Yusof ◽  
Sharifuddin Md Zain ◽  
...  
Keyword(s):  
Mixed Micelles ◽  
Nucleophilic Reaction ◽  
Phenyl Salicylate

Mixed Micelles as Nano Polymer Therapeutics of Docetaxel: Increased In vitro Cytotoxicity and Decreased In vivo Toxicity

2018 ◽  
Vol 15 (4) ◽  
pp. 564-575 ◽  
Author(s):  
Arehalli S. Manjappa ◽  
Popat S. Kumbhar ◽  
Prajakta S. Khopade ◽  
Ajit B. Patil ◽  
John I. Disouza
Keyword(s):  
Mixed Micelles ◽  
In Vitro Cytotoxicity ◽  
Polymer Therapeutics ◽  
In Vivo Toxicity

Preparation and characterization of the ion-fixed mixed micelles with superior stability

2015 ◽  
Vol 489 (1-2) ◽  
pp. 268-276 ◽  
Author(s):  
Yang Li ◽  
Yang Fu ◽  
Hongyu Guo ◽  
Lixue Zhang ◽  
Lingling Huang ◽  
...  
Keyword(s):  
Mixed Micelles

scholarly journals Brain targeting efficiency of intranasal clozapine-loaded mixed micelles following radio labeling with Technetium-99m

Drug Delivery ◽  
2021 ◽  
Vol 28 (1) ◽  
pp. 1524-1538
Author(s):  
Sinar Sayed ◽  
Fatma M. Elsharkawy ◽  
Maha M. Amin ◽  
Hesham A. Shamsel-Din ◽  
Ahmed B. Ibrahim
Keyword(s):  
Mixed Micelles ◽  
Brain Targeting ◽  
Technetium 99M ◽  
Targeting Efficiency ◽  
Radio Labeling

scholarly journals Recombinant acyl-CoA:cholesterol acyltransferase-1 (ACAT-1) purified to essential homogeneity utilizes cholesterol in mixed micelles or in vesicles in a highly cooperative manner.

1999 ◽  
Vol 274 (7) ◽  
pp. 4480
Author(s):  
Catherine C.Y. Chang ◽  
Chi-Yu Gregory Lee ◽  
Ellen T. Chang ◽  
Jonathan C. Cruz ◽  
Marc C. Levesque ◽  
...  
Keyword(s):  
Mixed Micelles

Water soluble biguanide salts and their 1,3,5-triazine derivatives as inhibitors of acetylcholinesterase and α-glucosidase

2020 ◽  
Vol 235 (10) ◽  
pp. 465-475
Author(s):  
Ozge Gungor ◽  
Seda Nur Kertmen Kurtar ◽  
Muhammet Kose
Keyword(s):  
Spectroscopic Method ◽  
Substitute Aniline ◽  
Water Soluble ◽  
X Ray Diffraction ◽  
Nucleophilic Reaction ◽  
X Ray ◽  
Triazine Derivatives ◽  
Acidic Conditions ◽  
Approved Drugs ◽  
Solid State Structures

AbstractSeven biguanide derivatives were prepared by the nucleophilic reaction between dicyandiamide and p-substitute aniline derivatives or memantine or adamantine under acidic conditions. The cyclization of the biguanide compounds were also conducted via acetone to give 1,3,5-triazine derivatives. The structures of the synthesized compounds were characterized by analytical methods. The solid state structures of [HL5]Cl, [H2L7]Cl2, [HL1a]Cl and [HL5a]Cl were investigated by X-ray diffraction study. The acetylcholinesterase and α-glucosidase inhibitor properties of the compounds were then evaluated by the spectroscopic method. The compounds were found to show considerable acetylcholinesterase and α-glucosidase inhibitory activities compared to the approved drugs. The cyclization of biguanide derivatives with acetone did not affect inhibition of acetylcholinesterase, yet increased the α-glucosidase inhibition.

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