Divergent Synthesis of Indole-2-carboxylic Acid Derivatives via Ligand-free Copper-catalyzed Ullmann Coupling Reaction

Heterocycles ◽  
2019 ◽  
Vol 98 (7) ◽  
pp. 904
Author(s):  
Jianjun Li ◽  
Jiadi Zhou ◽  
Yongjian Chen ◽  
Junsong Huang
2021 ◽  
Vol 125 (14) ◽  
pp. 7675-7685
Author(s):  
Tedros A. Balema ◽  
Jiayuan Miao ◽  
Natalie A. Wasio ◽  
Colin J. Murphy ◽  
Amanda M. Larson ◽  
...  

Synthesis ◽  
2012 ◽  
Vol 44 (19) ◽  
pp. 3027-3032 ◽  
Author(s):  
Yu Yuan ◽  
Ying Han ◽  
Xiaohu Wang ◽  
Xiaowei Wang ◽  
Liangzhong Lv ◽  
...  

2017 ◽  
Vol 102 ◽  
pp. 118-122 ◽  
Author(s):  
Aiqin Gao ◽  
Hongjuan Zhang ◽  
Liu Hu ◽  
Aiqin Hou ◽  
Kongliang Xie

RSC Advances ◽  
2015 ◽  
Vol 5 (81) ◽  
pp. 66104-66108 ◽  
Author(s):  
Yufen Zheng ◽  
Wenxing Zou ◽  
Laichun Luo ◽  
Jiabei Chen ◽  
Songwen Lin ◽  
...  

Coupling reaction between aryl iodides with aliphatic diols was realized with a ligand-free copper catalyst. This method was successfully applied in the process of scale-up synthesis of medicinal candidate product EMB-3.


Sign in / Sign up

Export Citation Format

Share Document