Synthesis and Biological Evaluation of Substituted Desloratadines as Potent Arginine Vasopressin V2  Receptor Antagonists

Shuai Mu; Ying Liu; Min Gong; Deng-Ke Liu; Chang-Xiao Liu

doi:10.3390/molecules19022694

Synthesis and Biological Evaluation of Substituted Desloratadines as Potent Arginine Vasopressin V2 Receptor Antagonists

Molecules ◽

10.3390/molecules19022694 ◽

2014 ◽

Vol 19 (2) ◽

pp. 2694-2706 ◽

Cited By ~ 3

Author(s):

Shuai Mu ◽

Ying Liu ◽

Min Gong ◽

Deng-Ke Liu ◽

Chang-Xiao Liu

Keyword(s):

Arginine Vasopressin ◽

Biological Evaluation ◽

Receptor Antagonists ◽

Vasopressin V2 Receptor ◽

V2 Receptor ◽

Synthesis And Biological Evaluation

Download Full-text

Synthesis and biological evaluation of novel phenothiazine derivatives as non-peptide arginine vasopressin V2 receptor antagonists

Chinese Chemical Letters ◽

10.1016/j.cclet.2015.01.022 ◽

2015 ◽

Vol 26 (5) ◽

pp. 627-630 ◽

Cited By ~ 2

Author(s):

Shuang Zhi ◽

Shuai Mu ◽

Ying Liu ◽

Min Gong ◽

Ping-Bao Wang ◽

...

Keyword(s):

Arginine Vasopressin ◽

Biological Evaluation ◽

Phenothiazine Derivatives ◽

Receptor Antagonists ◽

Vasopressin V2 Receptor ◽

V2 Receptor ◽

Synthesis And Biological Evaluation

Download Full-text

Synthesis and Biological Evaluation of Novel Indoloazepine Derivatives as Non-Peptide Vasopressin V2 Receptor Antagonists.

ChemInform ◽

10.1002/chin.200324220 ◽

2003 ◽

Vol 34 (24) ◽

Author(s):

Jay M. Matthews ◽

et al. et al.

Keyword(s):

Biological Evaluation ◽

Receptor Antagonists ◽

Vasopressin V2 Receptor ◽

V2 Receptor ◽

Synthesis And Biological Evaluation

Download Full-text

Synthesis and biological evaluation of novel indoloazepine derivatives as non-peptide vasopressin V2 receptor antagonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(02)01059-4 ◽

2003 ◽

Vol 13 (4) ◽

pp. 753-756 ◽

Cited By ~ 23

Author(s):

Jay M Matthews ◽

Michael N Greco ◽

Leonard R Hecker ◽

William J Hoekstra ◽

Patricia Andrade-Gordon ◽

...

Keyword(s):

Biological Evaluation ◽

Receptor Antagonists ◽

Vasopressin V2 Receptor ◽

V2 Receptor ◽

Synthesis And Biological Evaluation

Download Full-text

Synthesis and Biological Evaluation of the 1-Arylpyrazole Class of σ1 Receptor Antagonists: Identification of 4-{2-[5-Methyl-1-(naphthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862)

Journal of Medicinal Chemistry ◽

10.1021/jm3007323 ◽

2012 ◽

Vol 55 (19) ◽

pp. 8211-8224 ◽

Cited By ~ 82

Author(s):

José Luis Díaz ◽

Rosa Cuberes ◽

Joana Berrocal ◽

Montserrat Contijoch ◽

Ute Christmann ◽

...

Keyword(s):

Biological Evaluation ◽

Receptor Antagonists ◽

Σ1 Receptor ◽

Synthesis And Biological Evaluation

Download Full-text

N-(2,7-Dimethyl-2-alkyl-2H-chromen-6-yl)sulfonamide derivatives as selective serotonin 5-HT6 receptor antagonists: design, synthesis, and biological evaluation

Journal of Molecular Structure ◽

10.1016/j.molstruc.2021.131417 ◽

2021 ◽

pp. 131417

Author(s):

Aizhan Abdildinova ◽

Young Chang Kim ◽

Gee-Hyung Lee ◽

Woo-Kyu Park ◽

Heeyeong Cho ◽

...

Keyword(s):

Biological Evaluation ◽

Selective Serotonin ◽

Receptor Antagonists ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

Download Full-text

The treatment of vasopressin V2-receptor antagonists in cirrhosis patients with ascites: a meta-analysis of randomized controlled trials

BMC Gastroenterology ◽

10.1186/s12876-015-0297-z ◽

2015 ◽

Vol 15 (1) ◽

Cited By ~ 30

Author(s):

Long Yan ◽

Feng Xie ◽

Jiongjiong Lu ◽

Qingqiang Ni ◽

Changying Shi ◽

...

Keyword(s):

Randomized Controlled Trials ◽

Meta Analysis ◽

Controlled Trials ◽

Receptor Antagonists ◽

Randomized Controlled ◽

Vasopressin V2 Receptor ◽

V2 Receptor

Download Full-text

Nephrogenic Diabetes Insipidus Due to a New Mutation of the Arginine Vasopressin V2 Receptor Gene in a Girl Presenting with Non-Accidental Injury

Annals of Clinical Biochemistry International Journal of Laboratory Medicine ◽

10.1177/000456329903600616 ◽

1999 ◽

Vol 36 (6) ◽

pp. 779-782 ◽

Cited By ~ 9

Author(s):

C. P. C. Seem ◽

J. F. B. Dossetor ◽

M. D. Penney

Keyword(s):

Diabetes Insipidus ◽

Arginine Vasopressin ◽

Nephrogenic Diabetes Insipidus ◽

Receptor Gene ◽

Accidental Injury ◽

New Mutation ◽

Vasopressin V2 Receptor ◽

V2 Receptor ◽

Non Accidental Injury ◽

V2 Receptor Gene

Download Full-text

Synthesis and biological evaluation of 4′-[(benzimidazole-1-yl)methyl]biphenyl-2-sulfonamide derivatives as dual angiotensin II/endothelin A receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2012.06.011 ◽

2012 ◽

Vol 20 (15) ◽

pp. 4661-4667 ◽

Cited By ~ 18

Author(s):

Renren Bai ◽

Zhen Wei ◽

Jie Liu ◽

Weijia Xie ◽

Hequan Yao ◽

...

Keyword(s):

Angiotensin Ii ◽

Biological Evaluation ◽

Receptor Antagonists ◽

Endothelin A Receptor ◽

Endothelin A ◽

Synthesis And Biological Evaluation

Download Full-text

Design, synthesis, and biological evaluation of 2-(5-methyl-1H-pyrazol-1-yl) acetamide derivatives as androgen receptor antagonists

Medicinal Chemistry Research ◽

10.1007/s00044-019-02291-y ◽

2019 ◽

Vol 28 (3) ◽

pp. 380-386

Author(s):

Junze Dong ◽

Jingya Zhang ◽

Zilu Li ◽

Solomon Asnake ◽

Daoguang Zhang ◽

...

Keyword(s):

Androgen Receptor ◽

Biological Evaluation ◽

Receptor Antagonists ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Androgen Receptor Antagonists

Download Full-text

Design, synthesis, and biological evaluation of 2-(phenoxyaryl)-3-urea derivatives as novel P2Y1 receptor antagonists

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.09.014 ◽

2018 ◽

Vol 158 ◽

pp. 302-310 ◽

Cited By ~ 4

Author(s):

Jingjing Peng ◽

Lifen Zhao ◽

Lanlan Wang ◽

Hui Chen ◽

Yunguang Qiu ◽

...

Keyword(s):

Biological Evaluation ◽

P2y1 Receptor ◽

Receptor Antagonists ◽

Urea Derivatives ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

Download Full-text