scholarly journals Design, synthesis of 4-aminoquinoline-derived thiazolidines and their antimalarial activity and heme polymerization inhibition studies

2012 ◽  
Vol 28 (3) ◽  
pp. 619-626 ◽  
Author(s):  
V. Raja Solomon ◽  
W. Haq ◽  
Kumkum Srivastava ◽  
Sunil K. Puri ◽  
S.B. Katti
Keyword(s):  
Antimalarial Activity ◽  
Design Synthesis ◽  
Inhibition Studies

Design, Synthesis and Antimalarial Activity of Some New Aminoalcoholpyrrolo[1,2-a]quinoxaline Derivatives

2016 ◽  
Vol 13 (9) ◽  
pp. 932-942 ◽  
Author(s):  
Jean Guillon ◽  
Stéphane Moreau ◽  
Luisa Ronga ◽  
Louise Basmacyian ◽  
Anita Cohen ◽  
...  
Keyword(s):  
Antimalarial Activity ◽  
Design Synthesis ◽  
Quinoxaline Derivatives

scholarly journals Synthetic spirocyclic endoperoxides: new antimalarial scaffolds

MedChemComm ◽  
2015 ◽  
Vol 6 (2) ◽  
pp. 357-362 ◽  
Author(s):  
Margherita Brindisi ◽  
Sandra Gemma ◽  
Sanil Kunjir ◽  
Luisa Di Cerbo ◽  
Simone Brogi ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Antimalarial Activity ◽  
Design Synthesis ◽  
Docking Calculation

Design, synthesis and molecular docking calculation studies led to the identification of novel spirocyclic peroxides with in vitro and in vivo antimalarial activity.

ChemInform Abstract: Design, Synthesis, and Urease Inhibition Studies of a Series of 4-Amino-5-aryl-3H-1,2,4-triazole-3-thiones.

ChemInform ◽  
2010 ◽  
Vol 41 (38) ◽  
pp. no-no
Author(s):  
Mahmood-ul-Hassan Khan ◽  
Shahid Hameed ◽  
Khawaja A. Yasin ◽  
Tashfeen Akhtar ◽  
Khalid M. Khan
Keyword(s):  
Urease Inhibition ◽  
Design Synthesis ◽  
Inhibition Studies

scholarly journals Design, Synthesis and Antimalarial Activity of Novel, Quinoline-Based, Zinc Metallo-Aminopeptidase Inhibitors.

ChemInform ◽  
2003 ◽  
Vol 34 (50) ◽  
Author(s):  
Marian Flipo ◽  
Isabelle Florent ◽  
Philippe Grellier ◽  
Christian Sergheraert ◽  
Rebecca Deprez-Poulain
Keyword(s):  
Antimalarial Activity ◽  
Design Synthesis ◽  
Aminopeptidase Inhibitors

Design, synthesis and in vitro antimalarial activity of spiroperoxides

Tetrahedron ◽  
2006 ◽  
Vol 62 (33) ◽  
pp. 7699-7711 ◽  
Author(s):  
Hong-Xia Jin ◽  
Qi Zhang ◽  
Hye-Sook Kim ◽  
Yusuke Wataya ◽  
He-Hua Liu ◽  
...  
Keyword(s):  
Antimalarial Activity ◽  
Design Synthesis

Design, synthesis and glycosidase inhibition studies of novel triazole fused iminocyclitol-δ-lactams

2019 ◽  
Vol 17 (5) ◽  
pp. 1130-1140 ◽  
Author(s):  
Venkatesan Santhanam ◽  
Pradeep Pant ◽  
B. Jayaram ◽  
Namakkal G. Ramesh
Keyword(s):  
Design Synthesis ◽  
Key Steps ◽  
Inhibition Studies ◽  
Glycosidase Inhibition

Synthesis of novel triazole fused iminocyclitol-δ-lactams, from tri-O-benzyl-d-glucal, involving intermolecular [3 + 2]cycloaddition and intramolecular lactamisation reactions as key steps is described.

ChemInform Abstract: The Design, Synthesis and Biological Evaluation of Stable Ozonides with Antimalarial Activity.

ChemInform ◽  
2010 ◽  
Vol 27 (36) ◽  
pp. no-no
Author(s):  
L.-C. DE ALMEIDA BARBOSA ◽  
D. CUTLER ◽  
J. MANN ◽  
M. J. CRABBE ◽  
G. C. KIRBY ◽  
...  
Keyword(s):  
Antimalarial Activity ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

The design, synthesis and biological evaluation of stable ozonides with antimalarial activity

1996 ◽  
pp. 1101 ◽  
Author(s):  
Luiz-Claudio de Almeida Barbosa ◽  
David Cutler ◽  
John Mann ◽  
M. James Crabbe ◽  
Geoffrey C. Kirby ◽  
...  
Keyword(s):  
Antimalarial Activity ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, synthesis, inhibition studies, and molecular modeling of pepstatin analogues addressing different secreted aspartic proteinases of Candida albicans

2013 ◽  
Vol 85 (7) ◽  
pp. 881-887 ◽  
Author(s):  
Cosimo D. Cadicamo ◽  
Jérémie Mortier ◽  
Gerhard Wolber ◽  
Marie Hell ◽  
Ina E. Heinrich ◽  
...  
Keyword(s):  
Candida Albicans ◽  
Molecular Modeling ◽  
Aspartic Proteinases ◽  
Design Synthesis ◽  
Synthesis Inhibition ◽  
Inhibition Studies
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