Novel phenoxyalkylamine derivatives. V. Synthesis, .ALPHA.-blocking activity and quantitative structure-activity analysis of .ALPHA.-((phenoxyethylamino)propyl)-.ALPHA.-phenylacetonitrile derivatives.

KAZUYA MITANI; SHUNICHIRO SAKURAI; TOSHIHIRO SUZUKI; KOJI MORIKAWA; EIICHI KOSHINAKA; HIDEO KATO; YASUO ITO; TOSHIO FUJITA

doi:10.1248/cpb.36.4121

Novel phenoxyalkylamine derivatives. V. Synthesis, .ALPHA.-blocking activity and quantitative structure-activity analysis of .ALPHA.-((phenoxyethylamino)propyl)-.ALPHA.-phenylacetonitrile derivatives.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.36.4121 ◽

1988 ◽

Vol 36 (10) ◽

pp. 4121-4135 ◽

Cited By ~ 6

Author(s):

KAZUYA MITANI ◽

SHUNICHIRO SAKURAI ◽

TOSHIHIRO SUZUKI ◽

KOJI MORIKAWA ◽

EIICHI KOSHINAKA ◽

...

Keyword(s):

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity ◽

Alpha Blocking ◽

Blocking Activity

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ChemInform Abstract: Novel Phenoxyalkylamine Derivatives. Part 5. Synthesis, α-Blocking Activity, and Quantitative Structure-Activity Analysis of α-((Phenoxyethylamino)propyl)-α-phenylacetonitrile Derivatives (III).

ChemInform ◽

10.1002/chin.198923143 ◽

1989 ◽

Vol 20 (23) ◽

Author(s):

K. MITANI ◽

S. SAKURAI ◽

T. SUZUKI ◽

K. MORIKAWA ◽

E. KOSHINAKA ◽

...

Keyword(s):

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity ◽

Blocking Activity

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Quantitative Structure−Activity Analysis of the Algae Toxicity of Nitroaromatic Compounds

Chemical Research in Toxicology ◽

10.1021/tx9901635 ◽

2000 ◽

Vol 13 (6) ◽

pp. 441-450 ◽

Cited By ~ 57

Author(s):

Heike Schmitt ◽

Rolf Altenburger ◽

Bernd Jastorff ◽

Gerrit Schüürmann

Keyword(s):

Activity Analysis ◽

Nitroaromatic Compounds ◽

Quantitative Structure ◽

Structure Activity

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Quantitative Structure—Activity Analysis and Database-Aided Bioisosteric Structural Transformation Procedure as Methodologies of Agrochemical Design

ACS Symposium Series - Classical and Three-Dimensional QSAR in Agrochemistry ◽

10.1021/bk-1995-0606.ch002 ◽

1995 ◽

pp. 13-34 ◽

Cited By ~ 9

Author(s):

Toshio Fujita

Keyword(s):

Structural Transformation ◽

Activity Analysis ◽

Quantitative Structure ◽

Transformation Procedure ◽

Structure Activity

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Three-Dimensional Quantitative Structure—Activity Analysis of Steroidal and Dibenzoylhydrazine-Type Ecdysone Agonists

ACS Symposium Series - Classical and Three-Dimensional QSAR in Agrochemistry ◽

10.1021/bk-1995-0606.ch022 ◽

1995 ◽

pp. 288-301 ◽

Cited By ~ 21

Author(s):

Yoshiaki Nakagawa ◽

Bun-ichi Shimizu ◽

Nobuhiro Oikawa ◽

Miki Akamatsu ◽

Keiichiro Nishimura ◽

...

Keyword(s):

Three Dimensional ◽

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity

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ChemInform Abstract: A PRACTITIONER′S PERSPECTIVE OF THE ROLE OF QUANTITATIVE STRUCTURE-ACTIVITY ANALYSIS IN MEDICINAL CHEMISTRY

Chemischer Informationsdienst ◽

10.1002/chin.198131335 ◽

1981 ◽

Vol 12 (31) ◽

Author(s):

Y. C. MARTIN

Keyword(s):

Medicinal Chemistry ◽

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity

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Antifeedant effect of polygodial and drimenol derivatives againstSpodoptera frugiperdaandEpilachna paenulataand quantitative structure-activity analysis

Pest Management Science ◽

10.1002/ps.4853 ◽

2018 ◽

Vol 74 (7) ◽

pp. 1623-1629 ◽

Cited By ~ 5

Author(s):

Iván J Montenegro ◽

Soledad del Corral ◽

Georgina N Diaz Napal ◽

María C Carpinella ◽

Marco Mellado ◽

...

Keyword(s):

Activity Analysis ◽

Quantitative Structure ◽

Antifeedant Effect ◽

Structure Activity

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Quantitative Structure-Activity Analysis. Proceedings of the Second Symposium on Chemical Structure-Biological Acitivity Relationship: Quantitative Approaches, Suhl, 1976. Herausgegeben von R. Franke und P. Oehme. Abhandlungen der Akademie der Wissenschaften der DDR, Abt. Mathematik-Naturwissenschaften-Technik, Jahrgang 1978, Nr. 2 N, 452 Seiten mit zahlreichen Abb. und Tab., Akademie-Verlag, Berlin 1978. Preis: 72,—M

Nahrung/Food ◽

10.1002/food.19800240428 ◽

1980 ◽

Vol 24 (4-5) ◽

pp. 482-482

Author(s):

K. D. Schwenke

Keyword(s):

Chemical Structure ◽

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity ◽

Quantitative Approaches

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Quantitative structure–activity analysis of 5-arylidene-2,4-thiazolidinediones as aldose reductase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2005.10.069 ◽

2006 ◽

Vol 16 (3) ◽

pp. 512-520 ◽

Cited By ~ 13

Author(s):

S.V. Sambasivarao ◽

Love K. Soni ◽

Arun K. Gupta ◽

P. Hanumantharao ◽

S.G. Kaskhedikar

Keyword(s):

Aldose Reductase ◽

Activity Analysis ◽

Quantitative Structure ◽

Aldose Reductase Inhibitors ◽

Reductase Inhibitors ◽

Structure Activity

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Quantitative structure-activity analysis of larvicidal 1-(substituted benzoyl)-2-benzoyl-1-tert-butylhydrazines againstChilo suppressalis

Pesticide Science ◽

10.1002/ps.2780410210 ◽

1994 ◽

Vol 41 (2) ◽

pp. 139-147 ◽

Cited By ~ 45

Author(s):

Nobuhiro Oikawa ◽

Yoshiaki Nakagawa ◽

Keiichiro Nishimura ◽

Tamio Ueno ◽

Toshio Fujita

Keyword(s):

Activity Analysis ◽

Quantitative Structure ◽

Structure Activity

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Structure-activity relationships in prazosin-related compounds. 2. Role of the piperazine ring on .alpha.-blocking activity

Journal of Medicinal Chemistry ◽

10.1021/jm00058a005 ◽

1993 ◽

Vol 36 (6) ◽

pp. 690-698 ◽

Cited By ~ 37

Author(s):

Dario Giardina ◽

Ugo Gulini ◽

Maurizio Massi ◽

Maria G. Piloni ◽

Pierluigi Pompei ◽

...

Keyword(s):

Piperazine Ring ◽

Structure Activity Relationships ◽

Structure Activity ◽

Alpha Blocking ◽

Blocking Activity ◽

Related Compounds

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