scholarly journals Syntheses of N-Acyl Derivatives of α-Methyl-3, 4-methylenedioxyphenethylamine and their Analgesic Activity.

1963 ◽  
Vol 11 (5) ◽  
pp. 654-657 ◽  
Author(s):  
Keijiro Takagi ◽  
Yutaka Kasuya ◽  
Kyo Fujie ◽  
Minoru Watanabe ◽  
Setsuko Kayaoka
Keyword(s):  
Analgesic Activity ◽  
Derivatives Of ◽  
Acyl Derivatives

Synthesis and Analgesic Activity of 3,7-dimethylpurine-2,6-dion-1-yl Derivatives of Acetic and Butanoic Acid

2014 ◽  
Vol 11 (10) ◽  
pp. 1204-1213 ◽  
Author(s):  
Mal.gorzata Zygmunt ◽  
Pawe.l Zmudzki ◽  
Graz.yna Chl.on.-Rzepa ◽  
Jacek Sapa ◽  
Maciej Pawl.owski
Keyword(s):  
Analgesic Activity ◽  
Butanoic Acid ◽  
Derivatives Of

scholarly journals Synthesis, Antiproliferative Activity and Radical Scavenging Ability of 5-O-Acyl Derivatives of Quercetin

Molecules ◽  
2021 ◽  
Vol 26 (6) ◽  
pp. 1608
Author(s):  
Stephen Lo ◽  
Euphemia Leung ◽  
Bruno Fedrizzi ◽  
David Barker
Keyword(s):  
Antiproliferative Activity ◽  
Biological Activities ◽  
Radical Scavenging Activity ◽  
Radical Scavenging ◽  
Breast Cancer Cell Lines ◽  
Scavenging Activity ◽  
Plant Materials ◽  
Wide Range ◽  
Derivatives Of ◽  
Acyl Derivatives

Quercetin is a flavonoid that is found in many plant materials, including commonly eaten fruits and vegetables. The compound is well known for its wide range of biological activities. In this study, 5-O-acyl derivatives of quercetin were synthesised and assessed for their antiproliferative activity against the HCT116 colon cancer and MDA-MB-231 breast cancer cell lines; and their radical scavenging activity against the 2,2′-azino-bis(3-ethylbenzothiazoline-6-sulfonic acid) (ABTS) radical cation and 2,2-diphenyl-1-picrylhydrazyl (DPPH) radical species. Four derivatives were found to have improved the antiproliferative activity compared to quercetin whilst retaining radical scavenging activity.

ChemInform Abstract: O-ACYL DERIVATIVES OF 2-PYRIDINALDOXIME

1978 ◽  
Vol 9 (52) ◽  
Author(s):  
P. YA. ROMANOVSKII ◽  
A. YU. KRIKIS ◽  
G. I. CHIPENS
Keyword(s):  
Derivatives Of ◽  
Acyl Derivatives
Sign in / Sign up

Export Citation Format

Share Document