Simple One-Pot Synthesis of Thieno[2,3-b]thiophene Derivatives under Solid–Liquid PTC Conditions. Useful Starting Material for the Synthesis of Biological Active Compounds

1993 ◽  
Vol 66 (7) ◽  
pp. 2011-2015 ◽  
Author(s):  
Ahmed M. M. El-Saghier
2010 ◽  
Vol 12 (10) ◽  
pp. 2430-2433 ◽  
Author(s):  
Zhongyu Duan ◽  
Sadananda Ranjit ◽  
Xiaogang Liu

2019 ◽  
Vol 15 ◽  
pp. 2840-2846
Author(s):  
Valeriya G Melekhina ◽  
Andrey N Komogortsev ◽  
Boris V Lichitsky ◽  
Vitaly S Mityanov ◽  
Artem N Fakhrutdinov ◽  
...  

The condensation of primary amines with N-(1-(4-hydroxy-6-methyl-2-oxo-2H-pyran-3-yl)-2-oxo-2-arylethyl)acetamides was explored. Thus, a previously unknown recyclization of the starting material was observed in acidic ethanol in the presence of an amine, which provided the corresponding dihydropyrrolone derivative as the major reaction product. Based on this transformation, a practical and convenient one-pot synthetic method for substituted pyrrolo[3,4-b]pyridin-5-ones could be devised.


2003 ◽  
Vol 44 (35) ◽  
pp. 6665-6667 ◽  
Author(s):  
Meena V Patel ◽  
Jeffrey J Rohde ◽  
Vijaya Gracias ◽  
Teodozyj Kolasa

Heterocycles ◽  
2008 ◽  
Vol 75 (4) ◽  
pp. 919 ◽  
Author(s):  
Kazuhiro Kobayashi ◽  
Daizo Nakamura ◽  
Shuhei Fukamachi ◽  
Hisatoshi Konishi

2013 ◽  
Vol 830 ◽  
pp. 222-225
Author(s):  
Hai Xin Ding ◽  
Si Liu ◽  
Shan Shan Gong ◽  
Qi Sun

P1,P2-Diaciclovir-5'-diphosphate has been synthesized efficiently from aciclovir 5'-H-phosphonate monoester via a one-pot reaction. This method features easily accessibleH-phosphonate starting material, short reaction time, and good isolated yield.


Heterocycles ◽  
1981 ◽  
Vol 16 (1) ◽  
pp. 151 ◽  
Author(s):  
Zen-ichi Yoshida ◽  
Shegeo Yoneda ◽  
Hideo Hirai ◽  
Etsuro Seki

2017 ◽  
Vol 41 (10) ◽  
pp. 581-585 ◽  
Author(s):  
Hao Yang ◽  
Yifan Ouyang ◽  
Yutong Sun ◽  
Zhe Wang ◽  
Xuanli Zhu ◽  
...  

An efficient one-pot synthesis of 1-(4-bromophenyl)-1 H-tetrazol-5-amine was performed using 4-bromoaniline as the starting material. A novel and widely applicable amidation procedure was then employed, whereby 1-(4-bromophenyl)-1 H-tetrazol-5-amine was acylated with different acyl chlorides in the presence of lithium bis(trimethylsilyl)amide as catalyst, for the high-yield synthesis of [1-(4-bromophenyl)-1 H-tetrazol-5-yl]amide derivatives.


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