Aryl Hydrocarbon Receptor Activation and Cytochrome P450 1A Induction by the Mitogen-Activated Protein Kinase Inhibitor U0126 in Hepatocytes

Lise Andrieux; Sophie Langouët; Alain Fautrel; Fréderic Ezan; Joel A. Krauser; Jean F. Savouret; F. Peter Guengerich; Georges Baffet; André Guillouzo

doi:10.1124/mol.65.4.934

Aryl Hydrocarbon Receptor Activation and Cytochrome P450 1A Induction by the Mitogen-Activated Protein Kinase Inhibitor U0126 in Hepatocytes

Molecular Pharmacology ◽

10.1124/mol.65.4.934 ◽

2004 ◽

Vol 65 (4) ◽

pp. 934-943 ◽

Cited By ~ 59

Author(s):

Lise Andrieux ◽

Sophie Langouët ◽

Alain Fautrel ◽

Fréderic Ezan ◽

Joel A. Krauser ◽

...

Keyword(s):

Cytochrome P450 ◽

Protein Kinase ◽

Aryl Hydrocarbon Receptor ◽

Kinase Inhibitor ◽

Receptor Activation ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Aryl Hydrocarbon ◽

Mitogen Activated Protein ◽

Cytochrome P450 1A

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Mitogen-Activated Protein Kinase Inhibitor

10.32388/323rc0 ◽

2020 ◽

Author(s):

Keyword(s):

Protein Kinase ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Mitogen Activated Protein

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Faculty Opinions recommendation of Skepinone-L is a selective p38 mitogen-activated protein kinase inhibitor.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.13484956.14866145 ◽

2012 ◽

Author(s):

Wolfgang Peti

Keyword(s):

Protein Kinase ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Mitogen Activated Protein

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Cecal Tumorigenesis in Aryl Hydrocarbon Receptor–Deficient Mice Depends on Cecum-Specific Mitogen-Activated Protein Kinase Pathway Activation and Inflammation

American Journal Of Pathology ◽

10.1016/j.ajpath.2019.10.005 ◽

2020 ◽

Vol 190 (2) ◽

pp. 453-468 ◽

Cited By ~ 2

Author(s):

Hisanori Matoba ◽

Masaya Takamoto ◽

Chifumi Fujii ◽

Masatomo Kawakubo ◽

Eriko Kasuga ◽

...

Keyword(s):

Protein Kinase ◽

Aryl Hydrocarbon Receptor ◽

Mitogen Activated Protein Kinase ◽

Aryl Hydrocarbon ◽

Pathway Activation ◽

Mitogen Activated Protein ◽

Kinase Pathway ◽

Deficient Mice

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Effects of adding P38 mitogen-activated protein-kinase inhibitor to celsior solution in canine heart transplantation from non???heart-beating donors

Transplantation Journal ◽

10.1097/01.tp.0000101039.12835.a4 ◽

2004 ◽

Vol 77 (2) ◽

pp. 286-292 ◽

Cited By ~ 23

Author(s):

Norimasa Koike ◽

Izumi Takeyoshi ◽

Shigeru Ohki ◽

Masahiko Tokumine ◽

Koshi Matsumoto ◽

...

Keyword(s):

Protein Kinase ◽

Heart Transplantation ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Canine Heart ◽

Heart Beating ◽

Mitogen Activated Protein

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The p38 Mitogen-Activated Protein Kinase Inhibitor SB203580 Reduces Glucose Turnover by the Glucose Transporter-4 of 3T3-L1 Adipocytes in the Insulin-Stimulated State

Endocrinology ◽

10.1210/en.2004-1347 ◽

2005 ◽

Vol 146 (4) ◽

pp. 1818-1824 ◽

Cited By ~ 25

Author(s):

Merlijn Bazuine ◽

Françoise Carlotti ◽

Martijn J. W. E. Rabelink ◽

Jort Vellinga ◽

Rob C. Hoeben ◽

...

Keyword(s):

Protein Kinase ◽

Glucose Transporter ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Glucose Turnover ◽

Glucose Transporter 4 ◽

Mitogen Activated Protein

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The selective p38 mitogen-activated protein kinase inhibitor, SB203580, improves renal disease in MRL/lpr mouse model of systemic lupus

International Immunopharmacology ◽

10.1016/j.intimp.2011.04.015 ◽

2011 ◽

Vol 11 (9) ◽

pp. 1319-1326 ◽

Cited By ~ 20

Author(s):

Na Jin ◽

Qi Wang ◽

Xing Zhang ◽

Donghai Jiang ◽

Hao Cheng ◽

...

Keyword(s):

Protein Kinase ◽

Mouse Model ◽

Renal Disease ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Systemic Lupus ◽

Mitogen Activated Protein

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Pharmacokinetics of ML3403 ({4-[5-(4-Fluorophenyl)-2-methylsulfanyl-3H-imidazol-4-yl]-pyridin-2-yl}-(1-phenylethyl)-amine), a 4-Pyridinylimidazole-Type p38 Mitogen-Activated Protein Kinase Inhibitor

Drug Metabolism and Disposition ◽

10.1124/dmd.106.013409 ◽

2007 ◽

Vol 35 (6) ◽

pp. 875-883 ◽

Cited By ~ 15

Author(s):

Bernd Kammerer ◽

Holger Scheible ◽

Wolfgang Albrecht ◽

Christoph H. Gleiter ◽

Stefan Laufer

Keyword(s):

Protein Kinase ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Mitogen Activated Protein

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A novel regulatory mechanism of the mitochondrial Ca 2+ uniporter revealed by the p38 mitogen‐activated protein kinase inhibitor sb202190

The FASEB Journal ◽

10.1096/fj.02-0553fje ◽

2002 ◽

Vol 16 (14) ◽

pp. 1955-1957 ◽

Cited By ~ 64

Author(s):

Mayte Montero ◽

Carmen D. Lobatón ◽

Alfredo Moreno ◽

Javier Alvarez

Keyword(s):

Protein Kinase ◽

Regulatory Mechanism ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Mitogen Activated Protein

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p38α-Selective Mitogen-Activated Protein Kinase Inhibitor SD-282 Reduces Inflammation in a Subchronic Model of Tobacco Smoke-Induced Airway Inflammation

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.107.127092 ◽

2007 ◽

Vol 324 (3) ◽

pp. 921-929 ◽

Cited By ~ 73

Author(s):

Satyanarayana Medicherla ◽

Mary F. Fitzgerald ◽

Dianne Spicer ◽

Paul Woodman ◽

Jing Y. Ma ◽

...

Keyword(s):

Protein Kinase ◽

Airway Inflammation ◽

Tobacco Smoke ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Mitogen Activated Protein

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Proteomics-based insights into mitogen-activated protein kinase inhibitor resistance of cerebral melanoma metastases

Clinical Proteomics ◽

10.1186/s12014-018-9189-x ◽

2018 ◽

Vol 15 (1) ◽

Cited By ~ 7

Author(s):

Nina Zila ◽

Andrea Bileck ◽

Besnik Muqaku ◽

Lukas Janker ◽

Ossia M. Eichhoff ◽

...

Keyword(s):

Protein Kinase ◽

Kinase Inhibitor ◽

Protein Kinase Inhibitor ◽

Mitogen Activated Protein Kinase ◽

Melanoma Metastases ◽

Mitogen Activated Protein ◽

Inhibitor Resistance

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