Selective Regulation of Gq Signaling by G Protein-Coupled Receptor Kinase 2: Direct Interaction of Kinase N Terminus with Activated Gαq

2000 ◽  
Vol 57 (4) ◽  
pp. 826-831 ◽  
Author(s):  
Michele Sallese ◽  
Stefania Mariggiò ◽  
Etrusca D'Urbano ◽  
Luisa Iacovelli ◽  
Antonio De Blasi
Keyword(s):  
G Protein ◽  
Direct Interaction ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
N Terminus ◽  
G Protein Coupled

scholarly journals Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein–Coupled Receptor Kinase 2 Inhibitors

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Vol 92 (6) ◽  
pp. 707-717 ◽  
Author(s):  
Renee Bouley ◽  
Helen V. Waldschmidt ◽  
M. Claire Cato ◽  
Alessandro Cannavo ◽  
Jianliang Song ◽  
...  
Keyword(s):  
G Protein ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
Structural Determinants ◽  
G Protein Coupled

scholarly journals Generation of Highly Selective, Potent, and Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors

2021 ◽  
Author(s):  
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Qiuyan Chen ◽  
Renee A. Bouley ◽  
Larisa V. Avramova ◽  
John J. G. Tesmer ◽  
...  
Keyword(s):  
G Protein ◽  
Receptor Kinase ◽  
G Protein Coupled Receptor ◽  
G Protein Coupled
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