scholarly journals Intracellular Binding Site for a Positive Allosteric Modulator of the Dopamine D1 Receptor

2018 ◽  
Vol 94 (4) ◽  
pp. 1232-1245 ◽  
Author(s):  
Xushan Wang ◽  
Beverly A. Heinz ◽  
Yue-Wei Qian ◽  
Joan H. Carter ◽  
Robert A. Gadski ◽  
...  
Keyword(s):  
Binding Site ◽  
Dopamine D1 Receptor ◽  
D1 Receptor ◽  
Allosteric Modulator ◽  
Positive Allosteric Modulator ◽  
Intracellular Binding

Development of a Scalable Synthesis of Mevidalen (LY3154207), an Orally Available Positive Allosteric Modulator of the Human Dopamine D1 Receptor

2020 ◽  
Vol 24 (11) ◽  
pp. 2549-2564
Author(s):  
Jeffery Richardson ◽  
Kevin P. Cole ◽  
Amy C. DeBaillie ◽  
Junliang Hao ◽  
Jared Piper ◽  
...  
Keyword(s):  
Dopamine D1 Receptor ◽  
D1 Receptor ◽  
Allosteric Modulator ◽  
Positive Allosteric Modulator ◽  
Scalable Synthesis

scholarly journals Mapping a novel positive allosteric modulator binding site in the central vestibule region of human P2X7

2019 ◽  
Vol 9 (1) ◽  
Author(s):  
Stefan M. Bidula ◽  
Brett A. Cromer ◽  
Samuel Walpole ◽  
Jesus Angulo ◽  
Leanne Stokes
Keyword(s):  
Binding Site ◽  
Allosteric Modulator ◽  
Positive Allosteric Modulator

scholarly journals Characterization of a D1 Dopamine Receptor Positive Allosteric Modulator with a Novel Binding Site

2021 ◽  
Vol 35 (S1) ◽  
Author(s):  
Kathryn Luderman ◽  
R Benjamin Free ◽  
Forest Koenigsberg ◽  
Jeffrey Aubé ◽  
Kevin Frankowski ◽  
...  
Keyword(s):  
Binding Site ◽  
Dopamine Receptor ◽  
Allosteric Modulator ◽  
Positive Allosteric Modulator ◽  
D1 Dopamine Receptor
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