Ligand Residence Time at G-protein–Coupled Receptors—Why We Should Take Our Time To Study It

C. Hoffmann; M. Castro; A. Rinken; R. Leurs; S. J. Hill; H. F. Vischer

doi:10.1124/mol.115.099671

Ligand Residence Time at G-protein–Coupled Receptors—Why We Should Take Our Time To Study It

Molecular Pharmacology ◽

10.1124/mol.115.099671 ◽

2015 ◽

Vol 88 (3) ◽

pp. 552-560 ◽

Cited By ~ 49

Author(s):

C. Hoffmann ◽

M. Castro ◽

A. Rinken ◽

R. Leurs ◽

S. J. Hill ◽

...

Keyword(s):

G Protein ◽

Residence Time ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Drug-Target Residence Time-A Case for G Protein-Coupled Receptors

Medicinal Research Reviews ◽

10.1002/med.21307 ◽

2014 ◽

Vol 34 (4) ◽

pp. 856-892 ◽

Cited By ~ 115

Author(s):

Dong Guo ◽

Julia M. Hillger ◽

Adriaan P. IJzerman ◽

Laura H. Heitman

Keyword(s):

G Protein ◽

Residence Time ◽

Drug Target ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Molecular Basis of Ligand Dissociation from G Protein-Coupled Receptors and Predicting Residence Time

Methods in Molecular Biology - Computational Methods for GPCR Drug Discovery ◽

10.1007/978-1-4939-7465-8_9 ◽

2017 ◽

pp. 197-206 ◽

Cited By ~ 2

Author(s):

Dong Guo ◽

Adriaan P. IJzerman

Keyword(s):

G Protein ◽

Residence Time ◽

Molecular Basis ◽

G Protein Coupled Receptors ◽

Ligand Dissociation ◽

G Protein Coupled

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Importance of Drug-Target Residence Time at G Protein-Coupled Receptors - a Case for the Adenosine Receptors

Thermodynamics and Kinetics of Drug Binding - Methods and Principles in Medicinal Chemistry ◽

10.1002/9783527673025.ch13 ◽

2015 ◽

pp. 257-272 ◽

Cited By ~ 2

Author(s):

Dong Guo ◽

Adriaan P. IJzerman ◽

Laura H. Heitman

Keyword(s):

G Protein ◽

Residence Time ◽

Adenosine Receptors ◽

Drug Target ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Oligomerization in Health and Disease: From Enzymes to G Protein-Coupled Receptors

10.1016/s1877-1173(20)x0002-0 ◽

2020 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

Health And Disease ◽

G Protein Coupled

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G Protein-Coupled Receptors Part A

10.1016/s0091-679x(17)x0006-x ◽

2017 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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G Protein-Coupled Receptors - Signaling, Trafficking and Regulation

10.1016/s0091-679x(16)x0002-7 ◽

2016 ◽

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Enhanced Salmonella virulence instigated by bactivorous protozoa and investigation of putative protozoan G protein-coupled receptors associated with bacterial engulfment

10.31274/etd-180810-61 ◽

2014 ◽

Author(s):

Matt T. Brewer

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

Salmonella Virulence ◽

G Protein Coupled

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Faculty Opinions recommendation of Modulation of postendocytic sorting of G protein-coupled receptors.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1008239.104108 ◽

2002 ◽

Author(s):

Silvia Arber

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Faculty Opinions recommendation of Proteochemometrics modeling of the interaction of amine G-protein coupled receptors with a diverse set of ligands.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1007831.98556 ◽

2002 ◽

Author(s):

Wolfgang Guba

Keyword(s):

G Protein ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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Faculty Opinions recommendation of Measurement of the millisecond activation switch of G protein-coupled receptors in living cells.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1014169.192885 ◽

2003 ◽

Author(s):

Kees Jalink

Keyword(s):

G Protein ◽

Living Cells ◽

G Protein Coupled Receptors ◽

G Protein Coupled

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