Contribution of Binding Enthalpy and Entropy to Affinity of Antagonist and Agonist Binding at Human and Guinea Pig Histamine H1-Receptor

2009 ◽  
Vol 76 (1) ◽  
pp. 25-37 ◽  
Author(s):  
Hans-Joachim Wittmann ◽  
Roland Seifert ◽  
Andrea Strasser
Keyword(s):  
Guinea Pig ◽  
Agonist Binding ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Enthalpy And Entropy ◽  
Binding Enthalpy

scholarly journals Histamine H1 -receptor-mediated modulation of the delayed rectifier K+ current in guinea-pig atrial cells: opposite effects on IKs and IKr

1999 ◽  
Vol 128 (7) ◽  
pp. 1545-1553 ◽  
Author(s):  
Yasunori Matsumoto ◽  
Takehiko Ogura ◽  
Hiroko Uemura ◽  
Toshihiro Saito ◽  
Yoshiaki Masuda ◽  
...  
Keyword(s):  
Guinea Pig ◽  
Delayed Rectifier ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Atrial Cells ◽  
K Current

Linking agonist binding to histamine H1 receptor activation

2005 ◽  
Vol 1 (2) ◽  
pp. 98-103 ◽  
Author(s):  
Aldo Jongejan ◽  
Martijn Bruysters ◽  
Juan A Ballesteros ◽  
Eric Haaksma ◽  
Remko A Bakker ◽  
...  
Keyword(s):  
Receptor Activation ◽  
Agonist Binding ◽  
H1 Receptor ◽  
Histamine H1 Receptor

scholarly journals Molecular cloning of guinea-pig histamine H1 receptor gene.

1993 ◽  
Vol 61 ◽  
pp. 261
Author(s):  
Yoshiyuki Horio ◽  
Yasutake Mori ◽  
Katsumi Fujimoto ◽  
Seiji Ito ◽  
Hiroyuki Fukui
Keyword(s):  
Guinea Pig ◽  
Molecular Cloning ◽  
Receptor Gene ◽  
H1 Receptor ◽  
Histamine H1 Receptor

scholarly journals Histamine H1 -receptor-mediated increase in the Ca2+ transient without a change in the Ca2+ current in electrically stimulated guinea-pig atrial myocytes

1998 ◽  
Vol 124 (8) ◽  
pp. 1744-1750 ◽  
Author(s):  
Kimihiro Yoshimoto ◽  
Yuichi Hattori ◽  
Hideki Houzen ◽  
Morio Kanno ◽  
Keishu Yasuda
Keyword(s):  
Guinea Pig ◽  
Atrial Myocytes ◽  
H1 Receptor ◽  
Histamine H1 Receptor

Multiple Differences in Agonist and Antagonist Pharmacology between Human and Guinea Pig Histamine H1-Receptor

2003 ◽  
Vol 305 (3) ◽  
pp. 1104-1115 ◽  
Author(s):  
Roland Seifert ◽  
Katharina Wenzel-Seifert ◽  
Tilmann Bürckstümmer ◽  
Heinz H. Pertz ◽  
Walter Schunack ◽  
...  
Keyword(s):  
Guinea Pig ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Agonist And Antagonist

Histamine H1-receptor-mediated cyclic GMP production in guinea-pig lung tissue is an l-arginine-dependent process

1991 ◽  
Vol 42 (2) ◽  
pp. 271-277 ◽  
Author(s):  
Rob Leurs ◽  
Marion M. Brozius ◽  
Wilco Jansen ◽  
Aalt Bast ◽  
Hendrik Timmerman
Keyword(s):  
Guinea Pig ◽  
Lung Tissue ◽  
Cyclic Gmp ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Dependent Process ◽  
Gmp Production
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