Silver-Catalyzed Desulfurizative Annulation of 1,2-Benzisothiazoles with Ynamides to Construct Multi-Substituted Isoquinolines

2021 ◽  
Author(s):  
Rui Fu ◽  
Ran Liu ◽  
Kang Lv ◽  
Changlei Zhu ◽  
Xiaoguang Bao
Keyword(s):  
Isoquinoline Derivatives

An unprecedented silver-catalyzed desulfurizative annulation of 1,2-benzisothiazoles with ynamides is disclosed, which offers a concise protocol to access multi-substituted isoquinoline derivatives. Mechanistically, the chemo- and regio-selective N-attack of 1,2-benzisothiazoles to...

Isoquinoline derivatives as potent CRTH2 receptor antagonists: Synthesis and SAR

2012 ◽  
Vol 22 (9) ◽  
pp. 3305-3310 ◽  
Author(s):  
Rie Nishikawa-Shimono ◽  
Yoshinori Sekiguchi ◽  
Takeshi Koami ◽  
Madoka Kawamura ◽  
Daisuke Wakasugi ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Isoquinoline Derivatives

Novel bifunctional alkylating agents, 5,10-dihydropyrrolo[1,2-b]isoquinoline derivatives, synthesis and biological activity

2011 ◽  
Vol 19 (1) ◽  
pp. 275-286 ◽  
Author(s):  
Ravi Chaniyara ◽  
Naval Kapuriya ◽  
Huajin Dong ◽  
Pei-Chih Lee ◽  
Sharda Suman ◽  
...  
Keyword(s):  
Biological Activity ◽  
Alkylating Agents ◽  
Isoquinoline Derivatives

ChemInform Abstract: An Easy Access to Benzo[f]isoquinoline Derivatives Using Benzocyclobutenes Derived from Resorcinol.

ChemInform ◽  
2000 ◽  
Vol 31 (45) ◽  
pp. no-no
Author(s):  
Celine Verrat ◽  
Norbert Hoffmann ◽  
Jean Pierre Pete
Keyword(s):  
Easy Access ◽  
Isoquinoline Derivatives

scholarly journals Studies on the Syntheses of Isoquinoline Derivatives. XXIX

1954 ◽  
Vol 74 (6) ◽  
pp. 621-625
Author(s):  
Tetsuji Kametani ◽  
Kazuo Ohtsuki
Keyword(s):  
Isoquinoline Derivatives

scholarly journals Syntheses of Isoquinoline Derivatives. V

1951 ◽  
Vol 71 (11) ◽  
pp. 1257-1260 ◽  
Author(s):  
Saburo Ishiwata ◽  
Taiichi Nozaki
Keyword(s):  
Isoquinoline Derivatives
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