Synthesis and evaluation of highly selective quinazoline-2,4-dione ligands for sphingosine-1-phosphate receptor 2

RSC Medicinal Chemistry ◽

10.1039/d1md00357g ◽

2022 ◽

Author(s):

Zonghua Luo ◽

Hui Liu ◽

Yanbo Yu ◽

Robert J Gropler ◽

Robyn Klein ◽

...

Keyword(s):

Binding Assay ◽

Sphingosine 1 Phosphate

A series of twenty-nine new quinazoline-2,4-dione compounds were synthesized and their IC50 values of binding toward sphingosine 1-phosphate receptor 2 (S1PR2) were determined using a [32P]S1P binding assay. Seven compounds...

Download Full-text

Quantitative Measurement of Sphingosine 1-Phosphate by Radioreceptor-Binding Assay

Analytical Biochemistry ◽

10.1006/abio.2000.4580 ◽

2000 ◽

Vol 282 (1) ◽

pp. 115-120 ◽

Cited By ~ 80

Author(s):

Naoya Murata ◽

Koichi Sato ◽

Junko Kon ◽

Hideaki Tomura ◽

Fumikazu Okajima

Keyword(s):

Quantitative Measurement ◽

Binding Assay ◽

Sphingosine 1 Phosphate

Download Full-text

Author response for "Sphingosine 1‐phosphate/microRNA‐1249‐5p/MCP‐1 axis is involved in macrophage‐associated inflammation in fatty liver injury in mice"

10.1002/eji.201948351/v3/response1 ◽

2020 ◽

Author(s):

Xiaofang Ji ◽

Le Yang ◽

Zhi Zhang ◽

Kai Zhang ◽

Na Chang ◽

...

Keyword(s):

Liver Injury ◽

Fatty Liver ◽

Author Response ◽

Sphingosine 1 Phosphate

Download Full-text

Decision letter for "Sphingosine 1‐phosphate/microRNA‐1249‐5p/MCP‐1 axis is involved in macrophage‐associated inflammation in fatty liver injury in mice"

10.1002/eji.201948351/v3/decision1 ◽

2020 ◽

Keyword(s):

Liver Injury ◽

Fatty Liver ◽

Sphingosine 1 Phosphate

Download Full-text

Review for "Sphingosine 1‐phosphate/microRNA‐1249‐5p/MCP‐1 axis is involved in macrophage‐associated inflammation in fatty liver injury in mice"

10.1002/eji.201948351/v1/review1 ◽

2019 ◽

Author(s):

B Kleuser

Keyword(s):

Liver Injury ◽

Fatty Liver ◽

Sphingosine 1 Phosphate

Download Full-text

Author response for "Detailed and atypical HLA‐E peptide binding motifs revealed by a novel peptide exchange binding assay"

10.1002/eji.202048719/v2/response1 ◽

2020 ◽

Author(s):

Lucy C. Walters ◽

Andrew J. McMichael ◽

Geraldine M. Gillespie

Keyword(s):

Binding Assay ◽

Peptide Binding ◽

Author Response ◽

Binding Motifs ◽

Peptide Exchange

Download Full-text

Decision letter for "Detailed and atypical HLA‐E peptide binding motifs revealed by a novel peptide exchange binding assay"

10.1002/eji.202048719/v1/decision1 ◽

2020 ◽

Keyword(s):

Binding Assay ◽

Peptide Binding ◽

Binding Motifs ◽

Peptide Exchange

Download Full-text

Sphingosine 1-phosphate

AccessScience ◽

10.1036/1097-8542.900158 ◽

2015 ◽

Keyword(s):

Sphingosine 1 Phosphate

Download Full-text

Sphingosine-1-phosphate

Lipidomics Gateway ◽

10.1038/lipidmaps.2010.23 ◽

2010 ◽

Author(s):

Emma Leah

Keyword(s):

Sphingosine 1 Phosphate

Download Full-text

Sphingosine-1-phosphate induced increase in tension development of aortic valve leaflets is mediated via sphingosine-1-phosphate 2 receptor

The Thoracic and Cardiovascular Surgeon ◽

10.1055/s-0031-1297862 ◽

2012 ◽

Vol 60 (S 01) ◽

Author(s):

A Jannasch ◽

W Witt ◽

T Christ ◽

U Ravens ◽

K Matschke ◽

...

Keyword(s):

Aortic Valve ◽

Tension Development ◽

Aortic Valve Leaflets ◽

Sphingosine 1 Phosphate

Download Full-text

TBG MEASUREMENTS BY COMPETITIVE LIGAND BINDING ASSAY (CLBA)

Acta Endocrinologica ◽

10.1530/acta.0.080s015 ◽

1975 ◽

Vol 80 (1_Suppla) ◽

pp. S15

Author(s):

K. H. Rudorff ◽

H. J. Kröll ◽

J. Herrmann

Keyword(s):

Ligand Binding ◽

Binding Assay ◽

Ligand Binding Assay ◽

Competitive Ligand

Download Full-text