scholarly journals Benefits and applications of microwave-assisted synthesis of nitrogen containing heterocycles in medicinal chemistry

RSC Advances ◽  
2020 ◽  
Vol 10 (24) ◽  
pp. 14170-14197 ◽  
Author(s):  
Maged Henary ◽  
Carl Kananda ◽  
Laura Rotolo ◽  
Brian Savino ◽  
Eric A. Owens ◽  
...  
Keyword(s):  
Bioactive Compounds ◽  
Medicinal Chemistry ◽  
Research Interest ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Naturally Occurring

Nitrogen containing heterocycles are of immense research interest because they are often found as naturally occurring bioactive compounds.

scholarly journals Benzophenone: a ubiquitous scaffold in medicinal chemistry

MedChemComm ◽  
2018 ◽  
Vol 9 (11) ◽  
pp. 1803-1817 ◽  
Author(s):  
Khemchand Surana ◽  
Bharatkumar Chaudhary ◽  
Monika Diwaker ◽  
Satyasheel Sharma
Keyword(s):  
Biological Activity ◽  
Drug Discovery ◽  
Bioactive Compounds ◽  
Medicinal Chemistry ◽  
Naturally Occurring

Diaryl ketones are an important scaffold in drug discovery due to their prevalence in naturally occurring bioactive compounds. This review discusses molecules containing the benzophenone moiety that have potent biological activity.

ChemInform Abstract: Microwave-Assisted Synthesis of N-Heterocycles in Medicinal Chemistry

ChemInform ◽  
2014 ◽  
Vol 45 (3) ◽  
pp. no-no
Author(s):  
Davide Garella ◽  
Emily Borretto ◽  
Antonella Di Stilo ◽  
Katia Martina ◽  
Giancarlo Cravotto ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted

2-quinolone-based derivatives as antibacterial agents: A review

2021 ◽  
Vol 18 ◽  
Author(s):  
Oussama Moussaoui ◽  
Said Chakroune ◽  
Youssef Kandri Rodi ◽  
El Mestafa El Hadrami
Keyword(s):  
Organic Chemistry ◽  
Green Chemistry ◽  
Antibacterial Agents ◽  
Medicinal Chemistry ◽  
Antibacterial Activities ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Important Family ◽  
Reduced Toxicity ◽  
Synthetic Approaches

: The chemistry of 2-quinolones derivatives has received more attention in the field of both organic chemistry and medicinal chemistry. As several advances in the application of this important family of compounds seem too significant utility. In recent years, a variety of new, effective, and novel synthetic approaches (including green chemistry, catalyzed and microwave-assisted synthesis) have been discovered and developed for the designer of various 2-quinolone-based scaffolds, representing an area of increased interest to universities and industry, as well as, to explore their antibacterial activities and reduced toxicity than the existing ones. This review summarizes the results of the literature on the synthesis strategies of 2-quinolones derivatives and their reactivity, as well as their antibacterial evaluations against different bacteria strains.

scholarly journals Microwave-assisted synthesis of N-heterocycles in medicinal chemistry

MedChemComm ◽  
2013 ◽  
Vol 4 (10) ◽  
pp. 1323 ◽  
Author(s):  
Davide Garella ◽  
Emily Borretto ◽  
Antonella Di Stilo ◽  
Katia Martina ◽  
Giancarlo Cravotto ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted

scholarly journals Microwave-Assisted Synthesis of Bis-Heterocycles Containing the Imidazo[1,2-a]Pyridine by Groebke-Blackburn-Bienaymé Reaction

Proceedings ◽  
2019 ◽  
Vol 41 (1) ◽  
pp. 79
Author(s):  
Sandra C. Ramírez-López ◽  
Rocío Gámez-Montaño
Keyword(s):  
Medicinal Chemistry ◽  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Green Catalysis ◽  
Privileged Scaffolds

A series of six fused bis-heterocycles having imidazo[1,2-a]pyridine bound with quinoline were synthesized by microwave-assisted Groebke-Blackburn-Bienaymé reaction (GBBR) under green catalysis. The GBB products are privileged scaffolds and their synthesis is of great interest in synthetic and medicinal chemistry.

Convenient Microwave Assisted Synthesis of Naturally Occurring Methyl (E)-Cinnamates.

ChemInform ◽  
2005 ◽  
Vol 36 (42) ◽  
Author(s):  
Rajesh P. Mahajan ◽  
Shamkant L. Patil ◽  
Raghao S. Mali
Keyword(s):  
Microwave Assisted Synthesis ◽  
Microwave Assisted ◽  
Naturally Occurring
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