scholarly journals One-pot, three-component Fischer indolisation–N-alkylation for rapid synthesis of 1,2,3-trisubstituted indoles

2021 ◽  
Author(s):  
Christopher A. Hughes-Whiffing ◽  
Alexis Perry
Keyword(s):  
Rapid Synthesis ◽  
One Pot

One-pot Fischer indolisation indole N-alkylation enables straightforward, rapid synthesis of structurally-diverse 1,2,3-trisubstituted indoles from simple, widely-available precursors.

Facile construction of 3-indolochromenes and 3-indoloxanthenes via EDDF catalyzed one-pot three component reactions

2015 ◽  
Vol 39 (8) ◽  
pp. 6253-6260 ◽  
Author(s):  
Anuj Thakur ◽  
P. Linga Reddy ◽  
Mohit Tripathi ◽  
Diwan S. Rawat
Keyword(s):  
Ethylene Glycol ◽  
Catalytic System ◽  
Present Method ◽  
Rapid Synthesis ◽  
One Pot ◽  
By Products

EDDF–ethylene glycol, an ambiphilic catalytic system has been employed for the mild and rapid synthesis of various 3-indolochromenes and 3-indoloxanthenesviaa one-pot MCR. Besides recyclability of the catalyst, the present method circumvents the formation of any by-products.

Cascade In Situ Phosphorylation and One-Pot Glycosylation for Rapid Synthesis of Heptose-Containing Oligosaccharides

2020 ◽  
Vol 85 (24) ◽  
pp. 16060-16071
Author(s):  
Kwok-Kong Tony Mong ◽  
Kuang-Chun Cheng ◽  
I-Chen Lu ◽  
Chia-Wei Pan ◽  
Yi-Fang Wang ◽  
...  
Keyword(s):  
Rapid Synthesis ◽  
One Pot

DIPEAc promoted one-pot synthesis of dihydropyrido[2,3-d:6,5-d′]dipyrimidinetetraone and pyrimido[4,5-d]pyrimidine derivatives as potent tyrosinase inhibitors and anticancer agents: in vitro screening, molecular docking and ADMET predictions

2018 ◽  
Vol 42 (23) ◽  
pp. 18621-18632 ◽  
Author(s):  
Manisha R. Bhosle ◽  
Lalit D. Khillare ◽  
Jyotirling R. Mali ◽  
Aniket P. Sarkate ◽  
Deepak K. Lokwani ◽  
...  
Keyword(s):  
Molecular Docking ◽  
Anticancer Activity ◽  
Anticancer Agents ◽  
Oral Drug ◽  
In Vitro Screening ◽  
Pyrimidine Derivatives ◽  
Rapid Synthesis ◽  
One Pot ◽  
Tyrosinase Inhibitors

Efficient and rapid synthesis of 18 tyrosinase inhibitors with good to moderate anticancer activity and good oral drug like properties.

N-Bromosuccinimide Catalyzed One-pot and Rapid Synthesis of Acetamidobenzyl Naphthols under Mild and Solvent-free Conditions

2008 ◽  
Vol 26 (11) ◽  
pp. 2093-2097 ◽  
Author(s):  
Hamid Reza SHATERIAN ◽  
Hossein YARAHMADI ◽  
Majid GHASHANG ◽  
Moharram SAFARI MEHMANDOSTI
Keyword(s):  
Solvent Free ◽  
Rapid Synthesis ◽  
One Pot ◽  
Solvent Free Conditions
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