Synthesis of 1,3,4-trisubstituted pyrrolidines as meropenem adjuvants targeting New Delhi metallo-β-lactamase

2021 ◽  
Vol 45 (7) ◽  
pp. 3515-3534
Author(s):  
Wen Bin Jin ◽  
Chen Xu ◽  
Xiao Lin Qi ◽  
Ping Zeng ◽  
Wei Gao ◽  
...  

A promising NDM-1 inhibitor was discovered by the construction of pyrrolidine library via boric acid-catalyzed 1,3-dipolar cycloaddition and cell-based screens.

2007 ◽  
Vol 269 (1-2) ◽  
pp. 214-217 ◽  
Author(s):  
Mihir K. Chaudhuri ◽  
Sahid Hussain

1973 ◽  
Vol 38 (7) ◽  
pp. 1433-1434 ◽  
Author(s):  
Paul R. Stapp
Keyword(s):  

2012 ◽  
Vol 65 (1) ◽  
pp. 86 ◽  
Author(s):  
Sunanda B. Phadtare ◽  
R. Vijayraghavan ◽  
Ganapati S. Shankarling ◽  
Douglas R. MacFarlane

An efficient method for the synthesis of substituted 2,3-dihydro-1H-perimidine derivatives is described using bis(oxalato)boric acid (HBOB) as catalyst. The methodology provides an easily handled and recyclable catalyst for this type of reaction as an alternative platform to the conventional acid-catalyzed thermal processes. The time required to complete the reaction using HBOB was found to be shorter than conventional methods. Recycling of the catalyst has been efficiently achieved using a simple procedure.


ChemInform ◽  
2009 ◽  
Vol 40 (1) ◽  
Author(s):  
Andrei Badoiu ◽  
Gerald Bernardinelli ◽  
Jiri Mareda ◽  
E. Peter Kuendig ◽  
Florian Viton

ChemInform ◽  
2016 ◽  
Vol 47 (21) ◽  
Author(s):  
Zhenhua Zhang ◽  
Wangsheng Sun ◽  
Gongming Zhu ◽  
Junxian Yang ◽  
Ming Zhang ◽  
...  

1971 ◽  
Vol 12 (37) ◽  
pp. 3453-3454 ◽  
Author(s):  
William W. Lawrence
Keyword(s):  

2014 ◽  
Vol 7 (5) ◽  
pp. 54-58 ◽  
Author(s):  
Kabeer A. Shaikh ◽  
◽  
Sagar R. Kande ◽  
C. B. Khillare

2019 ◽  
Vol 7 (3) ◽  
pp. 1801164 ◽  
Author(s):  
Muchu Tan ◽  
Weihua Zhang ◽  
Changling Fan ◽  
Lingfang Li ◽  
Han Chen ◽  
...  

Sign in / Sign up

Export Citation Format

Share Document