scholarly journals Facile synthesis of 2-substituted benzo[b]furans and indoles by copper-catalyzed intramolecular cyclization of 2-alkynyl phenols and tosylanilines

RSC Advances ◽  
2019 ◽  
Vol 9 (31) ◽  
pp. 17975-17978 ◽  
Author(s):  
Zhouting Rong ◽  
Kexin Gao ◽  
Lei Zhou ◽  
Jianyuan Lin ◽  
Guoying Qian

A facile and inexpensive copper-catalyzed method was developed for the synthesis of 2-substituted benzo[b]furans and indoles.

2019 ◽  
Vol 17 (2) ◽  
pp. 380-387 ◽  
Author(s):  
Shuai Zou ◽  
Shu Geng ◽  
Lina Chen ◽  
Haitao Wang ◽  
Feng Huang

Visible light driven metal-free intramolecular cyclization: a facile synthesis of 3-position substituted 3,4-dihydroisoquinolin-1(2H)-one.


2013 ◽  
Vol 16 (1) ◽  
pp. 18-21 ◽  
Author(s):  
Qing Su ◽  
Pei Li ◽  
Mina He ◽  
Qiaolin Wu ◽  
Ling Ye ◽  
...  

2013 ◽  
Vol 8 (9) ◽  
pp. 1934578X1300800 ◽  
Author(s):  
Tao Zhang ◽  
Liang-Zhu Huang ◽  
You-Qiang Li ◽  
Yimg-Meng Xu ◽  
Zhen-Ting Du

A facile synthesis of (±)-heliannuol-D 1, which serves as an allelopathic chemical in nature and a potential lead compound in the search for new herbicides, has been achieved in a linear 11 steps, together with its epimer. The synthesis commenced with 4-methoxy-3-methyl-acetophenone, through the Baeyer-Villiger reaction, lithiation and addition, epoxidation and intramolecular cyclization to give (±)-heliannuol-D (1) and its epimer (1a) in 32.6% overall yield. Our synthetic approach is cost-effective; this will be helpful in applying this kind of compound for the development of a new generation of agrochemicals.


2012 ◽  
Vol 53 (39) ◽  
pp. 5248-5252 ◽  
Author(s):  
Jun Lv ◽  
Qiancai Liu ◽  
Jie Tang ◽  
Franc Perdih ◽  
Kristof Kranjc

Sign in / Sign up

Export Citation Format

Share Document