Catalyst-free cyclization of anthranils and cyclic amines: one-step synthesis of rutaecarpine

2019 ◽  
Vol 55 (80) ◽  
pp. 12072-12075 ◽  
Author(s):  
Jian Li ◽  
Zheng-Bing Wang ◽  
Yue Xu ◽  
Xue-Chen Lu ◽  
Shang-Rong Zhu ◽  
...  

An efficient synthesis of rutaecarpine derivatives via a catalyst-free and atom-efficiency cyclization reaction between commercially available anthranils and cyclic amines is described.

Author(s):  
Xiaoyun Ran ◽  
Qian Zhou ◽  
Jin Zhang ◽  
Shanqiang Wang ◽  
Gui Wang ◽  
...  

Started from citric acid (CA) and ethylenediamine derivatives, a solvent-free, catalyst-free and highly yield synthesis approach for bicyclic 2-pyridones was presented. Continuing to modify the core structure, a series of...


2015 ◽  
Vol 13 (35) ◽  
pp. 9186-9189 ◽  
Author(s):  
Xuebing Chen ◽  
Youzhi Wu ◽  
Jinyi Xu ◽  
Hequan Yao ◽  
Aijun Lin ◽  
...  

A Rh(iii)-catalyzed cyclization of azoles with alkynes has been developed to construct azole-fused-pyridines in good to excellent yields.


2011 ◽  
Vol 7 ◽  
pp. 1334-1341 ◽  
Author(s):  
Sanny Verma ◽  
Suman L Jain ◽  
Bir Sain

PEG-embedded potassium tribromide ([K+PEG]Br3 −) was found to be an efficient and recyclable catalyst for the synthesis of functionalized piperidines in high yields in a one step, three component coupling between aldehyde, amine and β-keto ester. At the end of the reaction the [K+PEG]Br3 − was readily regenerated from the reaction mixture by treating the residue containing [K+PEG]Br− with molecular bromine.


ChemInform ◽  
2010 ◽  
Vol 27 (7) ◽  
pp. no-no
Author(s):  
J. W. LEE ◽  
H. J. SON ◽  
J. H. LEE ◽  
Y. E. JUNG ◽  
G. J. YOON ◽  
...  

ChemInform ◽  
2009 ◽  
Vol 40 (17) ◽  
Author(s):  
Jian-Feng Zhou ◽  
Gui-Xia Gong ◽  
Li-Tao An ◽  
Yu Liu ◽  
Feng-Xia Zhu ◽  
...  

2021 ◽  
pp. 163010
Author(s):  
Jong-Hyeok Choi ◽  
Sunghun Choi ◽  
Jung Sang Cho ◽  
Hyun-Kyung Kim ◽  
Sang Mun Jeong

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