Photochromic peptidic NPY Y4 receptor ligands

2019 ◽  
Vol 17 (9) ◽  
pp. 2467-2478 ◽  
Author(s):  
D. Lachmann ◽  
A. Konieczny ◽  
M. Keller ◽  
B. König
Keyword(s):  
Receptor Ligands ◽  
Structural Requirements ◽  
Y4 Receptor

Photoresponsive NPY Y4R ligands, containing an azobenzene, azopyrazole, diethienylethene or a fulgimide chromophore were prepared to explore structural requirements of Y4R agonists on Y4R binding.

Oligopeptides as Neuropeptide Y Y4 Receptor Ligands: Identification of a High-Affinity Tetrapeptide Agonist and a Hexapeptide Antagonist

2020 ◽  
Vol 63 (15) ◽  
pp. 8198-8215
Author(s):  
Adam Konieczny ◽  
Diana Braun ◽  
David Wifling ◽  
Günther Bernhardt ◽  
Max Keller
Keyword(s):  
Neuropeptide Y ◽  
Receptor Ligands ◽  
High Affinity ◽  
Y4 Receptor

ChemInform Abstract: Structural Requirements for Leukotriene CysLT1 Receptor Ligands

ChemInform ◽  
2010 ◽  
Vol 28 (47) ◽  
pp. no-no
Author(s):  
M.-Q. ZHANG ◽  
M. E. ZWAAGSTRA
Keyword(s):  
Receptor Ligands ◽  
Structural Requirements

scholarly journals Understanding the structural requirements of hybrid (S)-6-((2-(4-phenylpiperazin-1-yl)ethyl)(propyl)amino)-5,6,7,8-tetrahydronaphthalen-1-ol and its analogs as D2/D3 receptor ligands: a 3D QSAR investigation

MedChemComm ◽  
2014 ◽  
Vol 5 (9) ◽  
pp. 1384-1399 ◽  
Author(s):  
Gyan Modi ◽  
Horrick Sharma ◽  
Prashant S. Kharkar ◽  
Aloke K. Dutta
Keyword(s):  
3D Qsar ◽  
Structural Factors ◽  
D3 Receptor ◽  
Receptor Ligands ◽  
Structural Requirements ◽  
Dopamine D2

The present study reports the 3D QSAR of dopamine D2/D3 ligands to gain insights into the structural factors responsible for affinity and D3 selectivity.

Clinical applications of single photon emission tomography in neuromedicine

2000 ◽  
Vol 39 (08) ◽  
pp. 218-231 ◽  
Author(s):  
F. Grünwald ◽  
T. Kuwert ◽  
K. Tatsch ◽  
O. Sabri ◽  
O. Benkert ◽  
...  
Keyword(s):  
Single Photon ◽  
Inflammatory Diseases ◽  
Photon Emission ◽  
Clinical Applications ◽  
Emission Tomography ◽  
Receptor Ligands ◽  
Single Photon Emission ◽  
The Central Nervous System ◽  
Dementing Disorders ◽  
Photon Emission Tomography

SummaryThis article gives in his second part a critical review of the clinical applications of SPECT with perfusion markers and receptor ligands in dementing disorders and psychosis. In addition this review discusses clinical applications of SPECT investigations with perfusion markers in inflammatory diseases of the central nervous system and in brain trauma.

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