I2/TBHP-Mediated tandem cyclization and oxidation reaction: Facile access to 2-substituted thiazoles and benzothiazoles

2019 ◽  
Vol 17 (2) ◽  
pp. 252-256 ◽  
Author(s):  
Li Liu ◽  
Chen Tan ◽  
Rong Fan ◽  
Zihan Wang ◽  
Hongguang Du ◽  
...  

The efficient synthesis of 2-substituted thiazoles and benzothiazoles has been accomplished employing readily available cysteine esters and 2-aminobenzenethiols as N and S sources.

ChemInform ◽  
2010 ◽  
Vol 26 (7) ◽  
pp. no-no
Author(s):  
R. MAREK ◽  
M. POTACEK ◽  
J. MAREK ◽  
A. DE GROOT

1994 ◽  
Vol 35 (37) ◽  
pp. 6909-6912 ◽  
Author(s):  
Radek Marek ◽  
Milan Potáček ◽  
Jaromír Marek ◽  
Alex De Groot

Tetrahedron ◽  
2006 ◽  
Vol 62 (33) ◽  
pp. 7667-7673 ◽  
Author(s):  
Anne Giraud ◽  
Olivier Provot ◽  
Jean-François Peyrat ◽  
Mouâd Alami ◽  
Jean-Daniel Brion

ChemInform ◽  
2015 ◽  
Vol 46 (8) ◽  
pp. no-no
Author(s):  
Guangcun Ge ◽  
Xiaojun Huang ◽  
Changhua Ding ◽  
Hao Li ◽  
Shili Wan ◽  
...  

2010 ◽  
Vol 16 (21) ◽  
pp. 6151-6154 ◽  
Author(s):  
Ke-Gong Ji ◽  
Hai-Tao Zhu ◽  
Fang Yang ◽  
Xing-Zhong Shu ◽  
Shu-Chun Zhao ◽  
...  

Synlett ◽  
2019 ◽  
Vol 30 (20) ◽  
pp. 2295-2299 ◽  
Author(s):  
Venu Kandula ◽  
Pradeep Kumar Thota ◽  
Poosa Mallesham ◽  
K. Raghavulu ◽  
Anindita Chatterjee ◽  
...  

An efficient synthesis of various 3-fluorochromones (3-fluoro-4H-chromene-4-ones) from enamino ketones by using Selectfluor is described. The key step in the synthesis involves tandem fluorination and cyclization to form 3-fluorochromones in good yields. The significant features of this method include simple operational procedures, a high purity of the product, and excellent regioselectivity.


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