Synthesis and evaluation of novel non-covalent binding quinazoline glycoside derivatives targeting the L858R and T790M variants of EGFR

RSC Advances ◽  
2016 ◽  
Vol 6 (43) ◽  
pp. 36857-36862 ◽  
Author(s):  
Renshuai Zhang ◽  
Shaopeng Chen ◽  
Xiaowei Zhang ◽  
Rilei Yu ◽  
Shengbiao Wan ◽  
...  
Keyword(s):  
Cell Line ◽  
Carcinoma Cell ◽  
Covalent Binding ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line

A series of novel quinazoline glycoside derivatives were designed, synthesized, and evaluated for their inhibition activities against EGFR-WT, EGFR/L858R/T790M, and skin epidermoid carcinoma cell line (A431).

Method for Obtaining Daedaleopsis confragosa K-1326 Extracts with Antitumor Activity

2019 ◽  
Vol 35 (1) ◽  
pp. 68-72
Author(s):  
T.V. Teplyakova ◽  
E.A. Vyazovaya ◽  
E.D. Danilenko
Keyword(s):  
Antitumor Activity ◽  
Cell Line ◽  
Carcinoma Cell ◽  
The State ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
State Assignment ◽  
Therapeutic Drugs ◽  
Prevention And Treatment ◽  
Epidermoid Carcinoma Cell Line

A method for extraction and fractionation of proteins and polysaccharides from the biomass of the basidial fungus Daedaleopsis confragosa K-1326, having antitumor activity, shown on the epidermoid carcinoma cell line A431 and the cells of melanoma В16, has been developed. This method allows for reproducible production of series of preparations and can be used to obtain preparations from other basidiomycetes. The results obtained in this work show the promising prospects for the development and use of drugs from basidiomycetes for treatment of cancer. Basidiomycetes, Daedaleopsis confragosa, antitumor activity, fractionation, extraction The work was performed under the State Assignment «Development of preventive and therapeutic drugs based on basidiomycetes for the prevention and treatment of influenza with pandemic potential».

Intracellular epidermal interleukin 1-like factors in the human epidermoid carcinoma cell line A431

1986 ◽  
Vol 100 (1) ◽  
pp. 89-96 ◽  
Author(s):  
Conrad Hauser ◽  
Jean-Michel Dayer ◽  
Fabienne Jaunin ◽  
Béatrice de Rochemonteix ◽  
Jean-Hilaire Saurat
Keyword(s):  
Cell Line ◽  
Carcinoma Cell ◽  
Interleukin 1 ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
Human Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line

Establishment and Characterization of Cisplatin-Resistant Human Epidermoid Carcinoma Cell Line, A431 Cell

Chemotherapy ◽  
1998 ◽  
Vol 44 (6) ◽  
pp. 414-420 ◽  
Author(s):  
Hiroshi Mese ◽  
Akira Sasaki ◽  
Rafael E. Alcalde ◽  
Shuko Nakayama ◽  
Tomohiro Matsumura
Keyword(s):  
Cell Line ◽  
Carcinoma Cell ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
A431 Cell ◽  
Human Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line

Modulation of EGF Receptor Activity by Changes in the GM3 Content in a Human Epidermoid Carcinoma Cell Line, A431

2000 ◽  
Vol 256 (1) ◽  
pp. 74-82 ◽  
Author(s):  
Emmanuelle J. Meuillet ◽  
Barbara Mania-Farnell ◽  
David George ◽  
Jin-Ichi Inokuchi ◽  
Eric G. Bremer
Keyword(s):  
Cell Line ◽  
Egf Receptor ◽  
Carcinoma Cell ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
Receptor Activity ◽  
Human Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line

Establishment and Characterization of Human Uterine Cervical Epidermoid Carcinoma Cell line HHUS Containing HPV 59 DNA

Human Cell ◽  
2008 ◽  
Vol 17 (3) ◽  
pp. 151-156
Author(s):  
Isamu ISHIWATA ◽  
Yuko TOKIEDA ◽  
Megumi IGUCHI ◽  
Tomoharu TAMAGAWA ◽  
Chieko ISHIWATA ◽  
...  
Keyword(s):  
Cell Line ◽  
Carcinoma Cell ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line

scholarly journals MAPK/ERK regulation of P53 in human epidermoid carcinoma cell line A431

2018 ◽  
Vol 5 (4) ◽  
pp. 23
Author(s):  
Yuqin Hao ◽  
Chunyi Kang ◽  
Xin Zhang ◽  
Shuxia Kang ◽  
Xia Liu
Keyword(s):  
Cell Line ◽  
Carcinoma Cell ◽  
Carcinoma Cell Line ◽  
Epidermoid Carcinoma ◽  
Human Epidermoid Carcinoma ◽  
Epidermoid Carcinoma Cell Line
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