scholarly journals N,N′-Disubstituted thiourea and urea derivatives: design, synthesis, docking studies and biological evaluation against nitric oxide synthase

MedChemComm ◽  
2016 ◽  
Vol 7 (4) ◽  
pp. 667-678 ◽  
Author(s):  
Mariem Chayah ◽  
M. Encarnación Camacho ◽  
M. Dora Carrión ◽  
Miguel A. Gallo ◽  
Miguel Romero ◽  
...  
Keyword(s):  
Nitric Oxide ◽  
Nitric Oxide Synthase ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Urea Derivatives ◽  
Design Synthesis ◽  
Inos Inhibitors ◽  
Oxide Synthase

N,N′-Disubstituted thioureas and ureas as nNOS and iNOS inhibitors were synthesized. Thiourea 4g was the best inhibitor without eNOS inhibition.

Synthesis, Biological Evaluation, and Docking Studies of N-Substituted Acetamidines as Selective Inhibitors of Inducible Nitric Oxide Synthase

2009 ◽  
Vol 52 (5) ◽  
pp. 1481-1485 ◽  
Author(s):  
Cristina Maccallini ◽  
Antonia Patruno ◽  
Neva Bešker ◽  
Jamila Isabella Alì ◽  
Alessandra Ammazzalorso ◽  
...  
Keyword(s):  
Nitric Oxide ◽  
Nitric Oxide Synthase ◽  
Inducible Nitric Oxide Synthase ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Selective Inhibitors ◽  
Oxide Synthase ◽  
Inducible Nitric Oxide

scholarly journals Synthesis, Bioevaluation and Docking Studies of New Imidamide Derivatives as Nitric Oxide Synthase Inhibitors

2021 ◽  
pp. 116294
Author(s):  
Fabio Arias ◽  
Francisco Franco-Montalban ◽  
Miguel Romero ◽  
M. Dora Carrión ◽  
M. Encarnación Camacho
Keyword(s):  
Nitric Oxide ◽  
Nitric Oxide Synthase ◽  
Docking Studies ◽  
Nitric Oxide Synthase Inhibitors ◽  
Oxide Synthase
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