scholarly journals Unexpected isocyanide-based three-component bicyclization for the stereoselective synthesis of densely functionalized pyrano[3,4-c]pyrroles

2016 ◽  
Vol 52 (5) ◽  
pp. 900-903 ◽  
Author(s):  
Qian Gao ◽  
Wen-Juan Hao ◽  
Feng Liu ◽  
Shu-Jiang Tu ◽  
Shu-Liang Wang ◽  
...  
Keyword(s):  
Stereoselective Synthesis ◽  
Efficient Synthesis ◽  
Dialkyl Acetylenedicarboxylates

A novel three-component bicyclization strategy for the efficient synthesis of densely functionalized pyrano[3,4-c]pyrroles has been established from readily accessible 3-aroylacrylic acids, dialkyl acetylenedicarboxylates and isocyanides.

scholarly journals Efficient synthesis of α-alkyl-β-amino amides by transaminase-mediated dynamic kinetic resolutions

2019 ◽  
Vol 9 (15) ◽  
pp. 4083-4090 ◽  
Author(s):  
Ángela Mourelle-Insua ◽  
Daniel Méndez-Sánchez ◽  
James L. Galman ◽  
Iustina Slabu ◽  
Nicholas J. Turner ◽  
...  
Keyword(s):  
Kinetic Resolution ◽  
Stereoselective Synthesis ◽  
Efficient Synthesis ◽  
Dynamic Kinetic Resolution ◽  
Amino Amides ◽  
Kinetic Resolutions

A transaminase-catalyzed dynamic kinetic resolution is described for the stereoselective synthesis of a series of α-alkyl-β-amino amides.

Efficient Synthesis of Cyclic β-Oxophosphoranes by Microwave-Assisted Reaction of Cyclic Phosphine Oxides and Dialkyl Acetylenedicarboxylates.

ChemInform ◽  
2006 ◽  
Vol 37 (35) ◽  
Author(s):  
Gyoergy Keglevich ◽  
Eszter Dudas ◽  
Melinda Sipos ◽  
Dora Lengyel ◽  
Krisztina Ludanyi
Keyword(s):  
Phosphine Oxides ◽  
Efficient Synthesis ◽  
Dialkyl Acetylenedicarboxylates ◽  
Microwave Assisted

Stereoselective synthesis of natural product inspired carbohydrate fused pyrano[3,2-c]quinolones as antiproliferative agents

2018 ◽  
Vol 16 (12) ◽  
pp. 2049-2059 ◽  
Author(s):  
Priti Kumari ◽  
Chintam Narayana ◽  
Shraddha Dubey ◽  
Ashish Gupta ◽  
Ram Sagar
Keyword(s):  
Anticancer Activity ◽  
Natural Product ◽  
Stereoselective Synthesis ◽  
Efficient Synthesis ◽  
Antiproliferative Agents ◽  
Quinolone Derivatives

Design and efficient synthesis of new carbohydrate fused pyrano[3,2-c]quinolone derivatives and their submicromolar anticancer activity.

Sign in / Sign up

Export Citation Format

Share Document