scholarly journals Stereospecific alkylation of substituted adenines by the Mitsunobu coupling reaction under microwave-assisted conditions

RSC Advances ◽  
2014 ◽  
Vol 4 (43) ◽  
pp. 22425-22433 ◽  
Author(s):  
M. E. García-Rubiño ◽  
M. C. Núñez-Carretero ◽  
D. Choquesillo-Lazarte ◽  
J. M. García-Ruiz ◽  
Yolanda Madrid ◽  
...  
Keyword(s):  
Secondary Alcohol ◽  
Coupling Reaction ◽  
Membered Ring ◽  
Mitsunobu Reaction ◽  
Microwave Assisted ◽  
Complete Inversion ◽  
Substituted Adenines

The Mitsunobu reaction under microwave-assisted conditions reveals a complete inversion of the stereogenic centre of the secondary alcohol giving an alkylated purine linked to a homochiral six-membered ring.

ChemInform Abstract: Stereospecific Alkylation of Substituted Adenines by the Mitsunobu Coupling Reaction under Microwave-Assisted Conditions.

ChemInform ◽  
2014 ◽  
Vol 46 (2) ◽  
pp. no-no
Author(s):  
M. E. Garcia-Rubino ◽  
M. C. Nunez-Carretero ◽  
D. Choquesillo-Lazarte ◽  
J. M. Garcia-Ruiz ◽  
Yolanda Madrid ◽  
...  
Keyword(s):  
Coupling Reaction ◽  
Microwave Assisted ◽  
Substituted Adenines

Diversity-Oriented Synthesis of Dibenzoazocines and Dibenzoazepines via a Microwave-Assisted Intramolecular A3-Coupling Reaction

2010 ◽  
Vol 12 (12) ◽  
pp. 2774-2777 ◽  
Author(s):  
Jitender B. Bariwal ◽  
Denis S. Ermolat’ev ◽  
Toma N. Glasnov ◽  
Kristof Van Hecke ◽  
Vaibhav P. Mehta ◽  
...  
Keyword(s):  
Coupling Reaction ◽  
Diversity Oriented Synthesis ◽  
Microwave Assisted ◽  
A3 Coupling

scholarly journals Microwave Assisted Reactions of Azaheterocycles Formedicinal Chemistry Applications

Molecules ◽  
2020 ◽  
Vol 25 (3) ◽  
pp. 716 ◽  
Author(s):  
Dorina Amariucai-Mantu ◽  
Violeta Mangalagiu ◽  
Ramona Danac ◽  
Ionel I. Mangalagiu
Keyword(s):  
Biological Activity ◽  
Medicinal Chemistry ◽  
Membered Ring ◽  
Reaction Pathways ◽  
Microwave Assisted ◽  
Main Series ◽  
Privileged Scaffolds

Microwave (MW) assisted reactions have became a powerful tool in azaheterocycles chemistry during the last decades. Five and six membered ring azaheterocycles are privileged scaffolds in modern medicinal chemistry possessing a large variety of biological activity. This review is focused on the recent relevant advances in the MW assisted reactions applied to azaheterocyclic derivatives and their medicinal chemistry applications from the last five years. The review is divided according to the main series of azaheterocycles, more precisely 5- and 6-membered ring azaheterocycles (with one, two, and more heteroatoms) and their fused analogues. In each case, the reaction pathways, the advantages of using MW, and considerations concerning biological activity of the obtained products were briefly presented.

An efficient aqueous microwave-assisted Suzuki–Miyaura cross-coupling reaction in the thiazole series

2009 ◽  
Vol 11 (11) ◽  
pp. 1736 ◽  
Author(s):  
Anita Cohen ◽  
Maxime D. Crozet ◽  
Pascal Rathelot ◽  
Patrice Vanelle
Keyword(s):  
Coupling Reaction ◽  
Cross Coupling ◽  
Microwave Assisted ◽  
Cross Coupling Reaction

Microwave-Assisted Copper-Catalyzed Cross-Coupling Reaction of Thiols with Aryl Iodides in Water

Synthesis ◽  
2014 ◽  
Vol 47 (02) ◽  
pp. 181-186 ◽  
Author(s):  
Chin-Fa Lee ◽  
Yi-An Chen ◽  
Satpal Badsara ◽  
Wan-Ting Tsai
Keyword(s):  
Coupling Reaction ◽  
Cross Coupling ◽  
Microwave Assisted ◽  
Aryl Iodides ◽  
Cross Coupling Reaction

ChemInform Abstract: Solid-Supported Rhodium(0) Nano-/Microparticles: An Efficient Ligand-Free Heterogeneous Catalyst for Microwave-Assisted Suzuki-Miyaura Cross-Coupling Reaction.

ChemInform ◽  
2013 ◽  
Vol 44 (15) ◽  
pp. no-no
Author(s):  
Nitul Ranjan Guha ◽  
Chennayala Bal Reddy ◽  
Nidhi Aggarwal ◽  
Dharminder Sharma ◽  
Arun K. Shil ◽  
...  
Keyword(s):  
Heterogeneous Catalyst ◽  
Coupling Reaction ◽  
Cross Coupling ◽  
Microwave Assisted ◽  
Cross Coupling Reaction ◽  
Ligand Free
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