N-alkoxycarbonyl amino acid N-carboxyanhydrides and N,N-dialkoxycarbonyl amino acid fluorides from N,N-diprotected amino acids

Journal of the Chemical Society Chemical Communications ◽

10.1039/c39920000812 ◽

1992 ◽

pp. 812 ◽

Cited By ~ 13

Author(s):

J. Savrda ◽

M. Wakselman

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Fmoc amino acid fluorides in peptide synthesis — Extension of the method to extremely hindered amino acids

Tetrahedron Letters ◽

10.1016/0040-4039(96)01160-4 ◽

1996 ◽

Vol 37 (31) ◽

pp. 5483-5486 ◽

Cited By ~ 33

Author(s):

Holger Wenschuh ◽

Michael Beyermann ◽

Rüdiger Winter ◽

Michael Bienert ◽

Dumitru Ionescu ◽

...

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Peptide Synthesis ◽

Amino Acid Fluorides ◽

Acid Fluorides

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ChemInform Abstract: Activation of N,N-Bis(alkoxycarbonyl) Amino Acids. Synthesis of N- Alkoxycarbonyl Amino Acid N-Carboxyanhydrides and N,N-Dialkoxycarbonyl Amino Acid Fluorides, and Their Behavior.

ChemInform ◽

10.1002/chin.199438247 ◽

2010 ◽

Vol 25 (38) ◽

pp. no-no

Author(s):

J. SAVRDA ◽

L. CHERTANOVA ◽

M. WAKSELMAN

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Amino Acid Fluorides ◽

Acid Fluorides

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ChemInform Abstract: N-Alkoxycarbonyl Amino Acid N-Carboxyanhydrides and N,N- Dialkoxycarbonyl Amino Acid Fluorides from N,N-Diprotected Amino Acids.

ChemInform ◽

10.1002/chin.199242165 ◽

2010 ◽

Vol 23 (42) ◽

pp. no-no

Author(s):

J. SAVRDA ◽

M. WAKSELMAN

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Activation of N,N-bis(alkoxycarbonyl) amino acids. Synthesis of N-alkoxycarbonyl amino acid N-carboxyanhydrides and N,N-dialkoxycarbonyl amino acid fluorides, and the behavior of these amino acid derivatives.

Tetrahedron ◽

10.1016/s0040-4020(01)80689-x ◽

1994 ◽

Vol 50 (18) ◽

pp. 5309-5322 ◽

Cited By ~ 19

Author(s):

Jaroslav Šavrda ◽

Lyubov Chertanova ◽

Michel Wakselman

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Amino Acid Derivatives ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Convenient and efficient synthesis of Boc-/Z-/Fmoc-β-amino acids employingN-protected α-amino acid fluorides

Journal of Peptide Research ◽

10.1034/j.1399-3011.2000.00683.x ◽

2000 ◽

Vol 55 (4) ◽

pp. 289-294 ◽

Cited By ~ 13

Author(s):

K. Ananda ◽

H.N. Gopi ◽

V.V. Suresh Babu

Keyword(s):

Amino Acids ◽

Amino Acid ◽

Efficient Synthesis ◽

Amino Acid Fluorides ◽

Acid Fluorides

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[(9-Fluorenylmethyl)oxy]carbonyl (FMOC) amino acid fluorides. Convienient new peptide coupling reagents applicable to the FMOC/tert-butyl strategy for solution and solid-phase syntheses.

Journal of the American Chemical Society ◽

10.1021/ja00182a041 ◽

1990 ◽

Vol 112 (26) ◽

pp. 9651-9652 ◽

Cited By ~ 152

Author(s):

Louis A. Carpino ◽

Dean Sadat-Aalaee ◽

Hann Guang Chao ◽

Robert H. DeSelms

Keyword(s):

Amino Acid ◽

Solid Phase ◽

Coupling Reagents ◽

Peptide Coupling ◽

Tert Butyl ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Synthesis of N-alkoxycarbonyl amino acid N-carboxyanhydrides (UNCAs) and N,N-dialkoxycarbonyl amino acid fluorides (U2AAFs)

Peptides 1992 ◽

10.1007/978-94-011-1470-7_84 ◽

1993 ◽

pp. 215-217

Author(s):

Michel Wakselman ◽

Jaroslav Savrda

Keyword(s):

Amino Acid ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Fmoc-amino acid fluorides: Application to multiple synthesis

Peptides 1994 ◽

10.1007/978-94-011-1468-4_75 ◽

1995 ◽

pp. 185-186 ◽

Cited By ~ 1

Author(s):

H. Wenschuh ◽

S. Rothemund ◽

M. Beyermann ◽

L. A. Carpino ◽

M. Bienert

Keyword(s):

Amino Acid ◽

Amino Acid Fluorides ◽

Acid Fluorides ◽

Multiple Synthesis

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Amino acid fluorides: Their preparation and use in peptide synthesis

Tetrahedron Letters ◽

10.1016/s0040-4039(00)79651-1 ◽

1991 ◽

Vol 32 (10) ◽

pp. 1303-1306 ◽

Cited By ~ 37

Author(s):

Jean-Nöel Bertho ◽

Albert Loffet ◽

Catherine Pinel ◽

Florence Reuther ◽

Gérard Sennyey

Keyword(s):

Amino Acid ◽

Peptide Synthesis ◽

Amino Acid Fluorides ◽

Acid Fluorides

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Amino acid fluorides: viable tools for synthesis of peptides, peptidomimetics and enantiopure heterocycles

RSC Advances ◽

10.1039/c4ra16142d ◽

2015 ◽

Vol 5 (60) ◽

pp. 48331-48362 ◽

Cited By ~ 26

Author(s):

Girish Prabhu ◽

N. Narendra ◽

Basavaprabhu Basavaprabhu ◽

V. Panduranga ◽

Vommina V. Sureshbabu

Keyword(s):

Amino Acid ◽

Biologically Active ◽

Broad Perspective ◽

Wide Range ◽

Amino Acid Fluorides ◽

Acid Fluorides

This review provides a broad perspective of the uses of amino acid fluorides in the synthesis of peptides and a wide range of other molecules including peptidomimetics, heterocycles and biologically active molecules.

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