scholarly journals Discovery of novel inhibitors of human S-adenosylmethionine decarboxylase based on in silico high-throughput screening and a non-radioactive enzymatic assay

2015 ◽  
Vol 5 (1) ◽  
Author(s):  
Chenzeng Liao ◽  
Yanlin Wang ◽  
Xiao Tan ◽  
Lidan Sun ◽  
Sen Liu
Keyword(s):  
High Throughput ◽  
In Silico ◽  
High Throughput Screening ◽  
Enzymatic Assay ◽  
Adenosylmethionine Decarboxylase

Discovery of indenopyrazoles as EGFR and VEGFR-2 tyrosine kinase inhibitors by in silico high-throughput screening

2008 ◽  
Vol 18 (1) ◽  
pp. 285-288 ◽  
Author(s):  
Taikou Usui ◽  
Hyun Seung Ban ◽  
Junpei Kawada ◽  
Takatsugu Hirokawa ◽  
Hiroyuki Nakamura
Keyword(s):  
Tyrosine Kinase ◽  
Tyrosine Kinase Inhibitors ◽  
High Throughput ◽  
In Silico ◽  
High Throughput Screening ◽  
Kinase Inhibitors

Synthesis of new hydrophilic rhodamine based enzymatic substrates compatible with droplet-based microfluidic assays

2017 ◽  
Vol 53 (39) ◽  
pp. 5437-5440 ◽  
Author(s):  
Johan Fenneteau ◽  
Dany Chauvin ◽  
Andrew D. Griffiths ◽  
Clément Nizak ◽  
Janine Cossy
Keyword(s):  
High Throughput ◽  
High Throughput Screening ◽  
Enzymatic Assay ◽  
Microfluidic Assays

The modification of rhodamine core with a hydrophilic tag yields new fluorogenic enzymatic substrates compatible with high-throughput screening using droplet-based enzymatic assay.

scholarly journals High Throughput Screening of Pharmacokinetics and Metabolism in Drug Discovery (III) —Investigation on In silico Model for Membrane Permeability and CYP1A2 Inhibition—

2005 ◽  
Vol 125 (1) ◽  
pp. 141-147 ◽  
Author(s):  
Hiroshi KOMURA ◽  
Yukie SHIGEMOTO ◽  
Iichiro KAWAHARA ◽  
Kenichi MATSUDA ◽  
Rieko ANO ◽  
...  
Keyword(s):  
Drug Discovery ◽  
Membrane Permeability ◽  
High Throughput ◽  
In Silico ◽  
High Throughput Screening

High-Throughput Screening by In silico Molecular Docking of Eryngium Foetidum (Linn.) Bioactives for Cylcooxygenase-2 Inhibition

2016 ◽  
Vol 6 (4) ◽  
pp. 232-237 ◽  
Author(s):  
Pavan Rangahanumaiah ◽  
Ravishankar Vittal Rai ◽  
Asma Saqhib ◽  
Lydia Jothi ◽  
Marula Siddha Swamy ◽  
...  
Keyword(s):  
Molecular Docking ◽  
High Throughput ◽  
In Silico ◽  
High Throughput Screening ◽  
Eryngium Foetidum ◽  
In Silico Molecular Docking

scholarly journals In Silico Prediction of SARS Protease Inhibitors by Virtual High Throughput Screening

2007 ◽  
Vol 69 (4) ◽  
pp. 269-279 ◽  
Author(s):  
Dariusz Plewczynski ◽  
Marcin Hoffmann ◽  
Marcin von Grotthuss ◽  
Krzysztof Ginalski ◽  
Leszek Rychewski
Keyword(s):  
Protease Inhibitors ◽  
High Throughput ◽  
In Silico ◽  
High Throughput Screening ◽  
In Silico Prediction
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