scholarly journals Dioxotriazine derivatives as a new class of P2X3 receptor antagonists Part 2: Discovery of clinical candidate S-600918

2020 ◽  
Author(s):  
Naohiro Onodera ◽  
Hiroyuki Kai
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
New Class ◽  
Clinical Candidate

Pyrrolinone derivatives as a new class of P2X3 receptor antagonists Part 2: Discovery of orally bioavailable compounds

2019 ◽  
Vol 29 (5) ◽  
pp. 688-693 ◽  
Author(s):  
Hiroyuki Tobinaga ◽  
Takayuki Kameyama ◽  
Kentarou Asahi ◽  
Tohru Horiguchi ◽  
Miho Oohara ◽  
...  
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
New Class ◽  
Orally Bioavailable

Pyrrolinone derivatives as a new class of P2X3 receptor antagonists. Part 3: Structure-activity relationships of pyrropyrazolone derivatives

2020 ◽  
Vol 30 (24) ◽  
pp. 127636
Author(s):  
Hiroyuki Tobinaga ◽  
Takayuki Kameyama ◽  
Kentarou Asahi ◽  
Tohru Horiguchi ◽  
Miho Oohara ◽  
...  
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
New Class ◽  
Structure Activity

Dioxotriazine derivatives as a new class of P2X3 receptor antagonists: Identification of a lead and initial SAR studies

2021 ◽  
Vol 37 ◽  
pp. 127833
Author(s):  
Hiroyuki Kai ◽  
Tohru Horiguchi ◽  
Takayuki Kameyama ◽  
Kentaro Asahi ◽  
Takeshi Endoh ◽  
...  
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
New Class ◽  
Sar Studies

New P2X3 receptor antagonists. Part 1: Discovery and optimization of tricyclic compounds

2016 ◽  
Vol 26 (16) ◽  
pp. 3896-3904 ◽  
Author(s):  
Gábor Szántó ◽  
Attila Makó ◽  
Imre Bata ◽  
Bence Farkas ◽  
Sándor Kolok ◽  
...  
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
Tricyclic Compounds

scholarly journals Investigation on 2′,3′-O-Substituted ATP Derivatives and Analogs as Novel P2X3 Receptor Antagonists

2018 ◽  
Vol 10 (4) ◽  
pp. 493-498 ◽  
Author(s):  
Diego Dal Ben ◽  
Michela Buccioni ◽  
Catia Lambertucci ◽  
Gabriella Marucci ◽  
Andrea Spinaci ◽  
...  
Keyword(s):  
P2x3 Receptor ◽  
Receptor Antagonists ◽  
Atp Derivatives

4,5,6,7-Tetrahdryo-8-oxo-cycloheptimidazoles: a new class of potent non-peptide angiiotensin II receptor antagonists

1993 ◽  
Vol 3 (8) ◽  
pp. 1559-1564 ◽  
Author(s):  
Takashi Yanagisawa ◽  
Naoto Ueyama ◽  
Tomoyuki Kawai ◽  
Motoharu Sonegawa ◽  
Hiromi Baba ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
New Class
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