Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D1Antagonist (6aS,13bR)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl-5H- benzo[d]naphth[2,1-b]azepin-12-ol (Sch 39166):  1. Aziridinium Salt Based Syntheses

Richard W. Draper; Donald Hou; Radha Iyer; Gary M. Lee; Jimmy T. Liang; Janet L. Mas; Wanda Tormos; Eugene J. Vater; Frank Günter; Ingrid Mergelsberg; Dominik Scherer

doi:10.1021/op970121s

Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D1Antagonist (6aS,13bR)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl-5H- benzo[d]naphth[2,1-b]azepin-12-ol (Sch 39166): 1. Aziridinium Salt Based Syntheses

Organic Process Research & Development ◽

10.1021/op970121s ◽

1998 ◽

Vol 2 (3) ◽

pp. 175-185 ◽

Cited By ~ 15

Author(s):

Richard W. Draper ◽

Donald Hou ◽

Radha Iyer ◽

Gary M. Lee ◽

Jimmy T. Liang ◽

...

Keyword(s):

Sch 39166 ◽

Stereoselective Syntheses

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ChemInform Abstract: Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D1 Antagonist (6aS,13bR)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl-5H-benzo [d]naphth[2,1-b]azepin-12-ol (Sch 39166). Part 2. L-Homophenylalanine-Based Syntheses.

ChemInform ◽

10.1002/chin.199843183 ◽

2010 ◽

Vol 29 (43) ◽

pp. no-no

Author(s):

R. W. DRAPER ◽

D. HOU ◽

R. IYER ◽

G. M. LEE ◽

J. T. LIANG ◽

...

Keyword(s):

Sch 39166 ◽

Dopamine D1 Antagonist ◽

Stereoselective Syntheses

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Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D1Antagonist (6aS,13bR)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl- 5H-benzo[d]naphth[2,1-b]azepin-12-ol (Sch 39166): 2.l-Homophenylalanine-Based Syntheses

Organic Process Research & Development ◽

10.1021/op970122k ◽

1998 ◽

Vol 2 (3) ◽

pp. 186-193 ◽

Cited By ~ 12

Author(s):

Richard W. Draper ◽

Donald Hou ◽

Radha Iyer ◽

Gary M. Lee ◽

Jimmy T. Liang ◽

...

Keyword(s):

Sch 39166 ◽

Stereoselective Syntheses

Download Full-text

ChemInform Abstract: Novel Stereoselective Syntheses of the Fused Benzazepine Dopamine D1 Antagonist (6aS,13bR)-11-Chloro-6,6a,7,8,9,13b-hexahydro-7-methyl-5H-benzo [d]naphth[2,1-b]azepin-12-ol (Sch 39166). Part 1. Aziridinium Salt Based Syntheses.

ChemInform ◽

10.1002/chin.199842151 ◽

2010 ◽

Vol 29 (42) ◽

pp. no-no

Author(s):

R. W. DRAPER ◽

D. HOU ◽

R. IYER ◽

G. M. LEE ◽

J. T. LIANG ◽

...

Keyword(s):

Sch 39166 ◽

Dopamine D1 Antagonist ◽

Stereoselective Syntheses

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ChemInform Abstract: Stereoselective Syntheses of 4-Amino-aldoses, and Chiral Pyrrolidine Derivatives from Glycosylenamines.

ChemInform ◽

10.1002/chin.199815208 ◽

2010 ◽

Vol 29 (15) ◽

pp. no-no

Author(s):

J. FUENTES ◽

D. OLANO ◽

M. A. PRADERA

Keyword(s):

Stereoselective Syntheses

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ChemInform Abstract: STEREOSELECTIVE SYNTHESES OF ALCOHOLS. IV. CONFORMATIONAL FACTORS DETERMINING G THE STEREOCHEMISTRY OF THE ALLYL SULFOXIDE-ALLYL SULFENATE REARRANGEMENT

Chemischer Informationsdienst ◽

10.1002/chin.198025096 ◽

1980 ◽

Vol 11 (25) ◽

Author(s):

R. W. HOFFMANN ◽

R. GERLACH ◽

S. GOLDMANN

Keyword(s):

Stereoselective Syntheses

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4-alkoxycarbonyloxazoles as β-hydroxy-α-amino acid synthons: efficient stereoselective syntheses of 3-amino-2,3,6-trideoxyhexoses and a hydroxy amino acid moiety of Al-77-B

Tetrahedron ◽

10.1016/s0040-4020(01)85597-6 ◽

1990 ◽

Vol 46 (13-14) ◽

pp. 4823-4846 ◽

Cited By ~ 45

Author(s):

Yasumasa Hamada ◽

Akiyoshi Kawai ◽

Toshiaki Matsui ◽

Osamu Hara ◽

Takayuki Shioiri

Keyword(s):

Amino Acid ◽

Acid Moiety ◽

Hydroxy Amino Acid ◽

Hydroxy Amino ◽

Amino Acid Moiety ◽

Stereoselective Syntheses

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Stereoselective Syntheses of All Stereoisomers of Lariciresinol and Their Plant Growth Inhibitory Activities

Journal of Agricultural and Food Chemistry ◽

10.1021/jf203222w ◽

2011 ◽

Vol 59 (24) ◽

pp. 13089-13095 ◽

Cited By ~ 24

Author(s):

Hisashi Nishiwaki ◽

Mitsuko Kumamoto ◽

Yoshihiro Shuto ◽

Satoshi Yamauchi

Keyword(s):

Plant Growth ◽

Growth Inhibitory ◽

Inhibitory Activities ◽

Stereoselective Syntheses

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Stereoselective syntheses using carbohydrates as chiral auxiliaries

Pure and Applied Chemistry ◽

10.1351/pac199567101627 ◽

1995 ◽

Vol 67 (10) ◽

pp. 1627-1635 ◽

Cited By ~ 38

Author(s):

H. Kunz

Keyword(s):

Chiral Auxiliaries ◽

Stereoselective Syntheses

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Organoboron monosaccharides, XVIII. Stereoselective syntheses of β-D-lyxofuranosyl glycosides

Liebigs Annalen der Chemie ◽

10.1002/jlac.1990199001197 ◽

1990 ◽

Vol 1990 (11) ◽

pp. 1093-1096 ◽

Cited By ~ 3

Author(s):

Wilhelm V. Dahlhoff

Keyword(s):

Stereoselective Syntheses

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Stereoselective Syntheses of 4-Oxa Diaminopimelic Acid and Its Protected Derivatives via Aziridine Ring Opening

Organic Letters ◽

10.1021/ol701742x ◽

2007 ◽

Vol 9 (21) ◽

pp. 4211-4214 ◽

Cited By ~ 25

Author(s):

Hongqiang Liu ◽

Vijaya R. Pattabiraman ◽

John C. Vederas

Keyword(s):

Ring Opening ◽

Diaminopimelic Acid ◽

Aziridine Ring ◽

Stereoselective Syntheses

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