δ-Amino β-Keto Esters, a Designed Polyfunctionalized Chiral Building Block for Alkaloid Synthesis. Asymmetric Synthesis of (R)-(+)-2-Phenylpiperidine and (−)-SS20846A

Franklin A. Davis; Bin Chao; Tianan Fang; Joanna M. Szewczyk

doi:10.1021/ol005580j

δ-Amino β-Keto Esters, a Designed Polyfunctionalized Chiral Building Block for Alkaloid Synthesis. Asymmetric Synthesis of (R)-(+)-2-Phenylpiperidine and (−)-SS20846A

Organic Letters ◽

10.1021/ol005580j ◽

2000 ◽

Vol 2 (8) ◽

pp. 1041-1043 ◽

Cited By ~ 51

Author(s):

Franklin A. Davis ◽

Bin Chao ◽

Tianan Fang ◽

Joanna M. Szewczyk

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Keto Esters ◽

Alkaloid Synthesis ◽

Chiral Building Block

Download Full-text

ChemInform Abstract: δ-Amino β-Keto Esters, a Designed Polyfunctionalized Chiral Building Block for Alkaloid Synthesis. Asymmetric Synthesis of (R)-(+)-2-Phenylpiperidine and (-)-SS20846A.

ChemInform ◽

10.1002/chin.200031150 ◽

2010 ◽

Vol 31 (31) ◽

pp. no-no

Author(s):

Franklin A. Davis ◽

Bin Chao ◽

Tianan Fang ◽

Joanna M. Szewczyk

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Keto Esters ◽

Alkaloid Synthesis ◽

Chiral Building Block

Download Full-text

Asymmetric Synthesis of a Chiral Building Block for Cyclopentanoids: A Novel Enantioselective Synthesis of Preclavulone A.

ChemInform ◽

10.1002/chin.200710224 ◽

2007 ◽

Vol 38 (10) ◽

Author(s):

Giuseppe Zanoni ◽

Alessio Porta ◽

Enrico Brunoldi ◽

Giovanni Vidari

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Enantioselective Synthesis ◽

Chiral Building Block

Download Full-text

ChemInform Abstract: Bicyclo(3.3.1)nonanes as Synthetic Intermediates. Part 21. Enantiodivergent Synthesis of the cis,cis 2,6-Disubstituted Piperidin- 3-ol Chiral Building Block for Alkaloid Synthesis.

ChemInform ◽

10.1002/chin.199745247 ◽

2010 ◽

Vol 28 (45) ◽

pp. no-no

Author(s):

T. MOMOSE ◽

N. TOYOOKA ◽

M. JIN

Keyword(s):

Building Block ◽

Alkaloid Synthesis ◽

Chiral Building Block ◽

Synthetic Intermediates

Download Full-text

Bicyclo[3.3.1]nonanes as synthetic intermediates. Part 21.1 Enantiodivergent synthesis of the cis,cis 2,6-disubstituted piperidin-3-ol chiral building block for alkaloid synthesis

Journal of the Chemical Society Perkin Transactions 1 ◽

10.1039/a608490g ◽

1997 ◽

pp. 2005-2014 ◽

Cited By ~ 15

Author(s):

Takefumi Momose ◽

Naoki Toyooka ◽

Makoto Jin

Keyword(s):

Building Block ◽

Alkaloid Synthesis ◽

Chiral Building Block ◽

Synthetic Intermediates

Download Full-text

ChemInform Abstract: Asymmetric Synthesis of the Indolizidine Alkaloids 207A, 209B, and 235B′: 6-Substituted 2,3-Didehydropiperidine-2-carboxylate as a Versatile Chiral Building Block.

ChemInform ◽

10.1002/chin.199432217 ◽

2010 ◽

Vol 25 (32) ◽

pp. no-no

Author(s):

T. MOMOSE ◽

N. TOYOOKA

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Indolizidine Alkaloids ◽

Chiral Building Block

Download Full-text

98% Enantioselectivity in the asymmetric synthesis of a useful chiral building block by heterogeneous method: Enantioselective hydrogenation of ethyl-benzoylformate over cinchona modified Pt/Al2O3 catalysts in the acetic acid

Catalysis Communications ◽

10.1016/s1566-7367(02)00058-4 ◽

2002 ◽

Vol 3 (3) ◽

pp. 125-127 ◽

Cited By ~ 47

Author(s):

Mária Sutyinszki ◽

Kornél Szöri ◽

Károly Felföldi ◽

Mihály Bartók

Keyword(s):

Acetic Acid ◽

Asymmetric Synthesis ◽

Building Block ◽

Enantioselective Hydrogenation ◽

Chiral Building Block ◽

Ethyl Benzoylformate

Download Full-text

Asymmetric synthesis of (−)- and (+)-kainic acid using a planar chiral amide as a chiral building block

Tetrahedron Letters ◽

10.1016/j.tetlet.2008.08.058 ◽

2008 ◽

Vol 49 (44) ◽

pp. 6327-6329 ◽

Cited By ~ 35

Author(s):

Katsuhiko Tomooka ◽

Toshiyuki Akiyama ◽

Phewluangdee Man ◽

Masaki Suzuki

Keyword(s):

Asymmetric Synthesis ◽

Kainic Acid ◽

Building Block ◽

Chiral Building Block

Download Full-text

ChemInform Abstract: Asymmetric Cleavage of 9-Azabicyclo(3.3.1)nona-3-one into cis-2,6- Disubstituted Piperidine. A Facile Approach to a Chiral Building Block for Alkaloid Synthesis.

ChemInform ◽

10.1002/chin.199135166 ◽

2010 ◽

Vol 22 (35) ◽

pp. no-no

Author(s):

T. MOMOSE ◽

N. TOYOOKA ◽

Y. HIRAI

Keyword(s):

Building Block ◽

Alkaloid Synthesis ◽

Chiral Building Block

Download Full-text

Asymmetric Synthesis of a Chiral Building Block for Cyclopentanoids: A Novel Enantioselective Synthesis of Preclavulone A

The Journal of Organic Chemistry ◽

10.1021/jo061321h ◽

2006 ◽

Vol 71 (22) ◽

pp. 8459-8466 ◽

Cited By ~ 14

Author(s):

Giuseppe Zanoni ◽

Alessio Porta ◽

Enrico Brunoldi ◽

Giovanni Vidari

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Enantioselective Synthesis ◽

Chiral Building Block

Download Full-text

An Asymmetric Synthesis of a Quaternary Chiral Building Block from Ethylmalonic Acid: A Preparation of Key Synthetic Intermediates of Hunteria- and Aspidosperma-type Indole Alkaloids

Heterocycles ◽

10.3987/com-90-5418 ◽

1990 ◽

Vol 31 (6) ◽

pp. 1017 ◽

Cited By ~ 10

Author(s):

Keiichiro Fukumoto ◽

Masataka Ihara ◽

Ken Yasui ◽

Nobuaki Takayanagi

Keyword(s):

Asymmetric Synthesis ◽

Building Block ◽

Indole Alkaloids ◽

Ethylmalonic Acid ◽

Chiral Building Block ◽

Synthetic Intermediates

Download Full-text