scholarly journals Benzofuran Derivatives as Potent, Orally Active S1P1 Receptor Agonists: A Preclinical Lead Molecule for MS

2010 ◽  
Vol 2 (2) ◽  
pp. 97-101 ◽  
Author(s):  
Ashis K. Saha ◽  
Xiang Yu ◽  
Jian Lin ◽  
Mercedes Lobera ◽  
Anurag Sharadendu ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Orally Active

(S)- and (R)-8-(di-n-propylamino)-6,7,8,9-tetrahydro-3H-benz[e]indole-1-carbaldehyde: a new class of orally active 5-HT1A-receptor agonists

1993 ◽  
Vol 36 (15) ◽  
pp. 2059-2065 ◽  
Author(s):  
Peter Stjernloef ◽  
Maria Gullme ◽  
Thomas Elebring ◽  
Bengt Andersson ◽  
Haakan Wikstroem ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
New Class ◽  
Orally Active

Identification of 6-Hydroxypyrimidin-4(1H)-one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists

2021 ◽  
Author(s):  
Zulan Pi ◽  
James A. Johnson ◽  
Wei Meng ◽  
Monique Phillips ◽  
William A. Schumacher ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
Orally Active

Indole-propionic acid derivatives as potent, S1P3-sparing and EAE efficacious sphingosine-1-phosphate 1 (S1P1) receptor agonists

2012 ◽  
Vol 22 (8) ◽  
pp. 2794-2797 ◽  
Author(s):  
Qinghua Meng ◽  
Baowei Zhao ◽  
Qiongfeng Xu ◽  
Xuesong Xu ◽  
Guanghui Deng ◽  
...  
Keyword(s):  
Propionic Acid ◽  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Sphingosine 1 Phosphate

Preparation, Resolution, and Biological Evaluation of 5-Aryl-1,2-dihydro-5H-chromeno[3,4-f]quinolines:  Potent, Orally Active, Nonsteroidal Progesterone Receptor Agonists

1998 ◽  
Vol 41 (15) ◽  
pp. 2779-2785 ◽  
Author(s):  
James P. Edwards ◽  
Lin Zhi ◽  
Charlotte L. F. Pooley ◽  
Christopher M. Tegley ◽  
Sarah J. West ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Biological Evaluation ◽  
Receptor Agonists ◽  
Orally Active

Novel S1P1 receptor agonists – Part 5: From amino-to alkoxy-pyridines

2016 ◽  
Vol 115 ◽  
pp. 326-341 ◽  
Author(s):  
Martin H. Bolli ◽  
Cyrille Lescop ◽  
Magdalena Birker ◽  
Ruben de Kanter ◽  
Patrick Hess ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor

Novel S1P1 Receptor Agonists - Part 2: From Bicyclo[3.1.0]hexane-Fused Thiophenes to Isobutyl Substituted Thiophenes

2013 ◽  
Vol 57 (1) ◽  
pp. 78-97 ◽  
Author(s):  
Martin H. Bolli ◽  
Jörg Velker ◽  
Claus Müller ◽  
Boris Mathys ◽  
Magdalena Birker ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Fused Thiophenes

Synthesis of 4(5)-phenylimidazole-based analogues of sphingosine-1-phosphate and FTY720: Discovery of potent S1P1 receptor agonists

2005 ◽  
Vol 15 (15) ◽  
pp. 3568-3572 ◽  
Author(s):  
Jeremy J. Clemens ◽  
Michael D. Davis ◽  
Kevin R. Lynch ◽  
Timothy L. Macdonald
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Sphingosine 1 Phosphate

Pyrazole derived from (+)-3-carene; a novel potent, selective scaffold for sphingosine-1-phosphate (S1P1) receptor agonists

2010 ◽  
Vol 20 (1) ◽  
pp. 35-37 ◽  
Author(s):  
Frédéric J. Zécri ◽  
Rainer Albert ◽  
Gregory Landrum ◽  
Klaus Hinterding ◽  
Nigel G. Cooke ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Sphingosine 1 Phosphate

Enhanced Gastrointestinal Motility with Orally Active Ghrelin Receptor Agonists

2009 ◽  
Vol 329 (3) ◽  
pp. 1178-1186 ◽  
Author(s):  
Soratree Charoenthongtrakul ◽  
Derek Giuliana ◽  
Kenneth A. Longo ◽  
Elizabeth K. Govek ◽  
Anna Nolan ◽  
...  
Keyword(s):  
Gastrointestinal Motility ◽  
Ghrelin Receptor ◽  
Receptor Agonists ◽  
Orally Active
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