Synthesis, Biological Activity, and Conformational Analysis of Fourseco-d-15,19-bisnor-1α,25-Dihydroxyvitamin D Analogues, Diastereomeric at C17 and C20

Xiaoming Zhou; Gui-Dong Zhu; Dirk Van Haver; Maurits Vandewalle; Pierre J. De Clercq; Annemieke Verstuyf; Roger Bouillon

doi:10.1021/jm980736v

Synthesis, Biological Activity, and Conformational Analysis of Fourseco-d-15,19-bisnor-1α,25-Dihydroxyvitamin D Analogues, Diastereomeric at C17 and C20

Journal of Medicinal Chemistry ◽

10.1021/jm980736v ◽

1999 ◽

Vol 42 (18) ◽

pp. 3539-3556 ◽

Cited By ~ 26

Author(s):

Xiaoming Zhou ◽

Gui-Dong Zhu ◽

Dirk Van Haver ◽

Maurits Vandewalle ◽

Pierre J. De Clercq ◽

...

Keyword(s):

Biological Activity ◽

Conformational Analysis ◽

Dihydroxyvitamin D

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Synthesis, biological activity, and conformational analysis of CD-ring modified trans-decalin 1α,25-dihydroxyvitamin D analogsElectronic supplementary information (ESI) available: Further experimental details. See http://www.rsc.org/suppdata/ob/b2/b209147j/

Organic & Biomolecular Chemistry ◽

10.1039/b209147j ◽

2002 ◽

Vol 1 (2) ◽

pp. 257-267 ◽

Cited By ~ 31

Author(s):

Yong-Jun Chen ◽

Ling-Jie Gao ◽

Ibrahim Murad ◽

Annemieke Verstuyf ◽

Lieve Verlinden ◽

...

Keyword(s):

Biological Activity ◽

Conformational Analysis ◽

Supplementary Information ◽

Dihydroxyvitamin D

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Biological activity and conformational analysis of C20 and C14 epimers of CD-ring modified trans-decalin 1α,25-dihydroxyvitamin D analogs

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/j.jsbmb.2004.03.052 ◽

2004 ◽

Vol 89-90 ◽

pp. 61-66 ◽

Cited By ~ 5

Author(s):

Pierre J. De Clercq ◽

Ibrahim Murad ◽

Ling-Jie Gao ◽

Yong-Jun Chen ◽

Dirk Van Haver ◽

...

Keyword(s):

Biological Activity ◽

Conformational Analysis ◽

Dihydroxyvitamin D

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Synthetic Strategy and Biological Activity of A-ring Stereoisomers of 1,25- Dihydroxyvitamin D3 and C2-Modified Analogues

Current Topics in Medicinal Chemistry ◽

10.2174/1568026615666141208102907 ◽

2014 ◽

Vol 14 (21) ◽

pp. 2446-2453 ◽

Cited By ~ 2

Author(s):

Toshie Fujishima ◽

Tsutomu Suenaga ◽

Takato Nozaki

Keyword(s):

Biological Activity ◽

Dihydroxyvitamin D ◽

1,25 Dihydroxyvitamin D ◽

Synthetic Strategy

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Synthesis, Conformational Analysis, and Biological Activity of a Rigid Carbocyclic Analogue of 2′-Deoxy Aristeromycin Built on a Bicyclo[3.1.0]hexane Template

Nucleosides and Nucleotides ◽

10.1080/07328319608002382 ◽

1996 ◽

Vol 15 (1-3) ◽

pp. 235-250 ◽

Cited By ~ 43

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Maqbool A. Siddiqui ◽

Harry Ford ◽

Clifford George ◽

Victor E. Marquez

Keyword(s):

Biological Activity ◽

Conformational Analysis

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Quaternary Indolizidine and Indolizidone Iminosugars as Potential Immunostimulating and Glycosidase Inhibitory Agents: Synthesis, Conformational Analysis, Biological Activity, and Molecular Docking Study

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.5b00951 ◽

2015 ◽

Vol 58 (19) ◽

pp. 7820-7832 ◽

Cited By ~ 19

Author(s):

Nitin J. Pawar ◽

Vijay Singh Parihar ◽

Ayesha Khan ◽

Rakesh Joshi ◽

Dilip D. Dhavale

Keyword(s):

Biological Activity ◽

Molecular Docking ◽

Conformational Analysis ◽

Docking Study ◽

Molecular Docking Study ◽

Inhibitory Agents

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ChemInform Abstract: Biological Activity of Transformed Steroids. Part 21. Synthesis, Conformational Analysis and Biological Activity of D7′-Pentarane-16α,7α-cycloheptanoprogesterone.

Chemischer Informationsdienst ◽

10.1002/chin.198628322 ◽

1986 ◽

Vol 17 (28) ◽

Author(s):

A. V. KAMERNITSKII ◽

I. S. LEVINA ◽

L. E. KULIKOVA ◽

I. L. SHAMOVSKII ◽

V. V. KORKHOV ◽

...

Keyword(s):

Biological Activity ◽

Conformational Analysis

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Biological Activity of Fluorine-Substituted 1,25-Dihydroxyvitamin D3 in Rats, in Chicken and in Japanese Quails

Annals of Nutrition and Metabolism ◽

10.1159/000177171 ◽

1986 ◽

Vol 30 (1) ◽

pp. 9-14 ◽

Cited By ~ 4

Author(s):

W.A. Rambeck ◽

H. Weiser ◽

H. Zucker

Keyword(s):

Biological Activity ◽

Dihydroxyvitamin D ◽

1,25 Dihydroxyvitamin D ◽

Japanese Quails

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Synthesis, Biological Activity, and Conformational Analysis of Peptidomimetic Analogues of theSaccharomyces cerevisiaeα-Factor Tridecapeptide†

Biochemistry ◽

10.1021/bi980787u ◽

1998 ◽

Vol 37 (36) ◽

pp. 12465-12476 ◽

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Y. Larry Zhang ◽

Hanumantha Rao Marepalli ◽

Hui-fen Lu ◽

Jeffrey M. Becker ◽

Fred Naider

Keyword(s):

Biological Activity ◽

Conformational Analysis

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Synthesis, biological activity, conformational analysis by NMR and molecular modeling of N-formyl-L-Met-L-Pro-L-Phe-OMe, a praline analogue of the chemotactic peptide N-formyl-L-Met-L-Leu-L-Phe-OH

International journal of peptide & protein research ◽

10.1111/j.1399-3011.1993.tb00482.x ◽

2009 ◽

Vol 41 (6) ◽

pp. 595-605 ◽

Cited By ~ 13

Author(s):

H. DUGAS ◽

M. LAROCHE ◽

M. PTAK ◽

H. LABBÉ

Keyword(s):

Biological Activity ◽

Molecular Modeling ◽

Conformational Analysis ◽

Chemotactic Peptide

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New synthesis and conformational analysis of lipid A: biological activity and supramolecular assembly

Journal of Endotoxin Research ◽

10.1177/09680519990050012001 ◽

1999 ◽

Vol 5 (1-2) ◽

pp. 46-51 ◽

Cited By ~ 17

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Koichi Fukase ◽

Masato Oikawa ◽

Yasuo Suda ◽

Wen-Chi Liu ◽

Yoshiyuki Fukase ◽

...

Keyword(s):

Biological Activity ◽

Conformational Analysis ◽

Lipid A ◽

Supramolecular Assembly ◽

New Synthesis

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