Structure−Activity Relationships of a New Family of Steroidal Aromatase Inhibitors. 1. Synthesis and Evaluation of a Series of Analogs Related to 19-[(Methylthio)methyl]androstenedione (RU54115)

1996 ◽  
Vol 39 (3) ◽  
pp. 757-772 ◽  
Author(s):  
Dominique Lesuisse ◽  
Jean-François Gourvest ◽  
Ouafae Benslimane ◽  
Frank Canu ◽  
Christine Delaisi ◽  
...  
Keyword(s):  
Aromatase Inhibitors ◽  
Structure Activity Relationships ◽  
New Family ◽  
Structure Activity ◽  
Steroidal Aromatase Inhibitors

New Structure–Activity Relationships of A- and D-Ring Modified Steroidal Aromatase Inhibitors: Design, Synthesis, and Biochemical Evaluation

2012 ◽  
Vol 55 (8) ◽  
pp. 3992-4002 ◽  
Author(s):  
Carla Varela ◽  
Elisiário J. Tavares da Silva ◽  
Cristina Amaral ◽  
Georgina Correia da Silva ◽  
Teresa Baptista ◽  
...  
Keyword(s):  
Aromatase Inhibitors ◽  
Design Synthesis ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Biochemical Evaluation ◽  
Steroidal Aromatase Inhibitors

Structure–activity relationships of 2-, 4-, or 6-substituted estrogens as aromatase inhibitors

2005 ◽  
Vol 96 (1) ◽  
pp. 51-58 ◽  
Author(s):  
Mitsuteru Numazawa ◽  
Momoko Ando ◽  
Yoko Watari ◽  
Takako Tominaga ◽  
Yasuko Hayata ◽  
...  
Keyword(s):  
Aromatase Inhibitors ◽  
Structure Activity Relationships ◽  
Structure Activity

scholarly journals Structure–Activity Relationships of Estrogen Derivatives as Aromatase Inhibitors. Effects of Heterocyclic Substituents

2008 ◽  
Vol 56 (9) ◽  
pp. 1304-1309 ◽  
Author(s):  
Mitsuteru Numazawa ◽  
Sachiko Komatsu ◽  
Takako Tominaga ◽  
Kouwa Yamashita
Keyword(s):  
Aromatase Inhibitors ◽  
Structure Activity Relationships ◽  
Structure Activity
Sign in / Sign up

Export Citation Format

Share Document