5-Hydroxyindole-2-carboxylic Acid Amides: Novel Histamine-3 Receptor Inverse Agonists for the Treatment of Obesity

2009 ◽  
Vol 52 (13) ◽  
pp. 3855-3868 ◽  
Author(s):  
Pascale David Pierson ◽  
Alec Fettes ◽  
Christian Freichel ◽  
Silvia Gatti-McArthur ◽  
Cornelia Hertel ◽  
...  
Keyword(s):  
Carboxylic Acid ◽  
Inverse Agonists ◽  
Carboxylic Acid Amides ◽  
Treatment Of Obesity

1-Sulfonyl-4-acylpiperazines as Selective Cannabinoid-1 Receptor (CB1R) Inverse Agonists for the Treatment of Obesity

2009 ◽  
Vol 52 (8) ◽  
pp. 2550-2558 ◽  
Author(s):  
Petr Vachal ◽  
Joan M. Fletcher ◽  
Tung M. Fong ◽  
Cathy C. R.-R. Huang ◽  
Julie Lao ◽  
...  
Keyword(s):  
Inverse Agonists ◽  
Cannabinoid 1 Receptor ◽  
Treatment Of Obesity

scholarly journals Local Anesthetics I. N-Alkyl Pyrrolidine and N-Alkyl Piperidine Carboxylic Acid Amides.

1957 ◽  
Vol 11 ◽  
pp. 1183-1190 ◽  
Author(s):  
Bo af Ekenstam ◽  
Börje Egnér ◽  
Gösta Pettersson
Keyword(s):  
Carboxylic Acid ◽  
Local Anesthetics ◽  
Carboxylic Acid Amides

Reactions of N-Allyl- and N,N-Diallyltrifluoromethanesulfonamides with Carboxylic Acid Amides under Oxidizing Conditions

2018 ◽  
Vol 54 (6) ◽  
pp. 855-860 ◽  
Author(s):  
V. V. Astakhova ◽  
M. Yu. Moskalik ◽  
A. S. Ganin ◽  
B. A. Shainyan
Keyword(s):  
Carboxylic Acid ◽  
Carboxylic Acid Amides

ChemInform Abstract: 1,5-DIPHENYLFORMAZAN-3-CARBOXYLIC ACID AMIDES

1984 ◽  
Vol 15 (28) ◽  
Author(s):  
T. S. KOLODINA ◽  
G. V. AVRAMENKO ◽  
B. I. STEPANOV
Keyword(s):  
Carboxylic Acid ◽  
Carboxylic Acid Amides

New Carboxylic Acid Amides of the Pyrrole Series: Synthetic Routes and Biological Aspects

2008 ◽  
Vol 63 (4) ◽  
pp. 351-362 ◽  
Author(s):  
Harald Walter
Keyword(s):  
Carboxylic Acid ◽  
Activity Level ◽  
Complex Ii ◽  
Carboxylic Acid Amides ◽  
Biological Aspects ◽  
Synthetic Routes ◽  
Special Complex ◽  
Sar Analysis

AbstractComplex II inhibitors play an important role in agrochemical fungicide research and have been known for more than 40 years. With the introduction of ortho-substituted heterocyclic amides, a breakthrough in activity level and spectrum within this class was achieved. In the meantime all major agrochemical companies have entered this field. In this paper, a special complex II subclass, the pyrrole carboxamides, will be introduced in more detail and the synthesis of selected compounds as well as a short biological SAR analysis of the pyrrole subclass will be discussed.

ChemInform Abstract: One-Pot Synthesis of (2E)- and (2E,4E)-Unsaturated Carboxylic Acid Amides via Organotellurium Reagents.

ChemInform ◽  
2010 ◽  
Vol 22 (44) ◽  
pp. no-no
Author(s):  
W.-J. XIAO ◽  
L.-L. SHI ◽  
Z.-Q. CHEN ◽  
Y.-Z. HUANG ◽  
S. A. LANG
Keyword(s):  
Carboxylic Acid ◽  
One Pot ◽  
Unsaturated Carboxylic Acid ◽  
One Pot Synthesis ◽  
Carboxylic Acid Amides
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