Discovery of 1H-Indole-2-carboxamides as Novel Inhibitors of the Androgen Receptor Binding Function 3 (BF3)

2014 ◽  
Vol 57 (15) ◽  
pp. 6867-6872 ◽  
Author(s):  
Fuqiang Ban ◽  
Eric Leblanc ◽  
Huifang Li ◽  
Ravi S. N. Munuganti ◽  
Kate Frewin ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Receptor Binding ◽  
Binding Function

Inhibition of androgen receptor binding by drugs in cultured human genital skin fibroblasts

1986 ◽  
Vol 113 (1_Suppl) ◽  
pp. S152
Author(s):  
M. BREINER ◽  
G. ROMALO ◽  
H.U. SCHWEIKERT
Keyword(s):  
Androgen Receptor ◽  
Receptor Binding ◽  
Skin Fibroblasts

Participation of Critical Residues from the Extreme C-Terminal End of the Human Androgen Receptor in the Ligand Binding Function†

Biochemistry ◽  
2001 ◽  
Vol 40 (29) ◽  
pp. 8431-8437 ◽  
Author(s):  
Bouchra Tahiri ◽  
Gilles Auzou ◽  
Jean-Claude Nicolas ◽  
Charles Sultan ◽  
Brigitte Lupo
Keyword(s):  
Androgen Receptor ◽  
Ligand Binding ◽  
Binding Function ◽  
Critical Residues ◽  
Human Androgen Receptor

A preliminary MTD-PLS study for androgen receptor binding of steroid compounds

2007 ◽  
Vol 107 (8) ◽  
pp. 1707-1713
Author(s):  
Alina Bora ◽  
E. Seclaman ◽  
L. Kurunczi ◽  
Simona Funar-Timofei
Keyword(s):  
Androgen Receptor ◽  
Receptor Binding

scholarly journals Genome-wide analysis of androgen receptor binding sites in prostate cancer cells

2015 ◽  
Vol 9 (6) ◽  
pp. 2319-2324 ◽  
Author(s):  
YUE CHENG ◽  
PAN YU ◽  
XIUZHI DUAN ◽  
CHUNHUA LIU ◽  
SIQI XU ◽  
...  
Keyword(s):  
Prostate Cancer ◽  
Androgen Receptor ◽  
Cancer Cells ◽  
Receptor Binding ◽  
Binding Sites ◽  
Prostate Cancer Cells ◽  
Genome Wide Analysis ◽  
Genome Wide

In Vitro Androgen Receptor Binding Affinity and in Vivo Inhibitory Activity of 5?-Pregnane-3, 20-Dione

1988 ◽  
Vol 529 (1 Fourth Colloq) ◽  
pp. 239-241
Author(s):  
SAUDHAMINI PARTHASARATHY ◽  
ANDREA CHIN ◽  
VIRGINIA MALLOY ◽  
JONATHAN MATIAS
Keyword(s):  
Androgen Receptor ◽  
Binding Affinity ◽  
Receptor Binding ◽  
Inhibitory Activity ◽  
Receptor Binding Affinity

Abstract 3654: Targeting binding function-3 site on the androgen receptor to treat Enzalutamide-resistant prostate cancer

2015 ◽  
Author(s):  
Ravi Shashi Nayana Munuganti ◽  
Mohamed DH Hassona ◽  
Eric Leblanc ◽  
Emma T. Guns ◽  
Paul S. Rennie ◽  
...  
Keyword(s):  
Prostate Cancer ◽  
Androgen Receptor ◽  
Binding Function

Abstract 3412: Androgen receptor binding sites are highly mutated in prostate cancer

2018 ◽  
Author(s):  
Tunc Morova ◽  
Mehmet Gonen ◽  
Attila Gursoy ◽  
Ozlem Keskin ◽  
Nathan A. Lack
Keyword(s):  
Prostate Cancer ◽  
Androgen Receptor ◽  
Receptor Binding ◽  
Binding Sites
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