Discovery of a Non-Estrogenic Irreversible Inhibitor of 17β-Hydroxysteroid Dehydrogenase Type 1 from 3-Substituted-16β-(m-carbamoylbenzyl)-estradiol Derivatives

2013 ◽  
Vol 57 (1) ◽  
pp. 204-222 ◽  
Author(s):  
René Maltais ◽  
Diana Ayan ◽  
Alexandre Trottier ◽  
Xavier Barbeau ◽  
Patrick Lagüe ◽  
...  
Keyword(s):  
Hydroxysteroid Dehydrogenase ◽  
Irreversible Inhibitor ◽  
Estradiol Derivatives

Identification of fused 16β,17β-oxazinone-estradiol derivatives as a new family of non-estrogenic 17β-hydroxysteroid dehydrogenase type 1 inhibitors

2015 ◽  
Vol 93 ◽  
pp. 470-480 ◽  
Author(s):  
René Maltais ◽  
Alexandre Trottier ◽  
Audrey Delhomme ◽  
Xavier Barbeau ◽  
Patrick Lagüe ◽  
...  
Keyword(s):  
Hydroxysteroid Dehydrogenase ◽  
New Family ◽  
Estradiol Derivatives

The role of hepatic 11[b]-hydroxysteroid dehydrogenase type 1 in cholesterol homeostasis

2013 ◽  
pp. 1-1
Author(s):  
Kajal Manwani ◽  
Tak Y Man ◽  
Christopher J Kenyon ◽  
Ruth Andrew ◽  
Karen E Chapman ◽  
...  
Keyword(s):  
Hydroxysteroid Dehydrogenase ◽  
Cholesterol Homeostasis

Macrophage-specific 11b-hydroxysteroid dehydrogenase type 1 deficiency promotes angiogenesis but impairs resolution of K/BxN serum induced arthritis

2013 ◽  
pp. 1-1
Author(s):  
Zhenguang Zhang ◽  
Agnes Coutinho ◽  
Patrick Hadoke ◽  
Donald Salter ◽  
Jonathan Seckl ◽  
...  
Keyword(s):  
Hydroxysteroid Dehydrogenase

Suppression of 11[beta]-hydroxysteroid dehydrogenase type 1 target gene regulation by hypoxia

2016 ◽  
Author(s):  
Bushra Shammout ◽  
Adewonuola Alase ◽  
Miriam Wittmann ◽  
Paul Stewart ◽  
Ana Tiganescu
Keyword(s):  
Gene Regulation ◽  
Target Gene ◽  
Hydroxysteroid Dehydrogenase
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