Water-Soluble Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines as Human A3 Adenosine Receptor Antagonists

2012 ◽  
Vol 55 (11) ◽  
pp. 5380-5390 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Giulia Saponaro ◽  
Romeo Romagnoli ◽  
Mojgan Aghazadeh Tabrizi ◽  
Stefania Baraldi ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Water Soluble ◽  
Receptor Antagonists ◽  
A3 Adenosine Receptor

Imidazo[2,1-i]purin-5-ones and Related Tricyclic Water-Soluble Purine Derivatives:  Potent A2A- and A3-Adenosine Receptor Antagonists†

2002 ◽  
Vol 45 (16) ◽  
pp. 3440-3450 ◽  
Author(s):  
Christa E. Müller ◽  
Mark Thorand ◽  
Ramatullah Qurishi ◽  
Martina Diekmann ◽  
Kenneth A. Jacobson ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Water Soluble ◽  
Purine Derivatives ◽  
Receptor Antagonists ◽  
A3 Adenosine Receptor

Affinity prediction on A3 adenosine receptor antagonists: The chemometric approach

2011 ◽  
Vol 19 (22) ◽  
pp. 6853-6859 ◽  
Author(s):  
Feng Luan ◽  
André Melo ◽  
Fernanda Borges ◽  
M. Natália D.S. Cordeiro
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
Affinity Prediction ◽  
A3 Adenosine Receptor ◽  
Chemometric Approach

One-Pot Reaction To Obtain N,N′-Disubstituted Guanidines of Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine Scaffold as Human A3 Adenosine Receptor Antagonists

2015 ◽  
Vol 58 (13) ◽  
pp. 5355-5360 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Stefania Baraldi ◽  
Giulia Saponaro ◽  
Mojgan Aghazadeh Tabrizi ◽  
Romeo Romagnoli ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Receptor Antagonists ◽  
One Pot ◽  
A3 Adenosine Receptor

A2A-selective adenosine receptor antagonists: Development of water-soluble prodrugs and a new tritiated radioligand

1998 ◽  
Vol 45 (3-4) ◽  
pp. 190-197 ◽  
Author(s):  
Christa E. M�ller ◽  
Roland Sauer ◽  
Yuris Maurinsh ◽  
Rosa Huertas ◽  
Friederike F�lle ◽  
...  
Keyword(s):  
Adenosine Receptor ◽  
Water Soluble ◽  
Receptor Antagonists
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