Investigation of the Histamine H3 Receptor Binding Site. Design and Synthesis of Hybrid Agonists with a Lipophilic Side Chain

2010 ◽  
Vol 53 (17) ◽  
pp. 6445-6456 ◽  
Author(s):  
Makoto Ishikawa ◽  
Takashi Watanabe ◽  
Toshiaki Kudo ◽  
Fumikazu Yokoyama ◽  
Miki Yamauchi ◽  
...  
Keyword(s):  
Binding Site ◽  
Receptor Binding ◽  
Side Chain ◽  
Receptor Binding Site ◽  
Histamine H3 Receptor ◽  
Design And Synthesis ◽  
H3 Receptor ◽  
Site Design ◽  
Histamine H3

Synthesis of S-[3-(4(5)-imidazolyl)propyl],N-[2(4-{125I}-iodophenyl)ethyl]isothiourea sulfate (125I-iodophenpropit), a new probe for histamine H3 receptor binding sites.

1992 ◽  
Vol 31 (10) ◽  
pp. 781-786 ◽  
Author(s):  
Wiro M. P. B. Menge ◽  
Henk Van Der Goot ◽  
Hendrik Timmerman ◽  
Jos. L. H. Eersels ◽  
Jacobu S. D. M. Herscheid
Keyword(s):  
Receptor Binding ◽  
Binding Sites ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Novel pyrrolidinone derivative lacks claimed histamine H3 receptor stimulation in receptor binding and functional studies

2020 ◽  
Vol 191 ◽  
pp. 112150
Author(s):  
David Reiner ◽  
Aleksandra Zivkovic ◽  
Olivier Labeeuw ◽  
Stéphane Krief ◽  
Marc Capet ◽  
...  
Keyword(s):  
Receptor Binding ◽  
Receptor Stimulation ◽  
Histamine H3 Receptor ◽  
Functional Studies ◽  
H3 Receptor ◽  
Pyrrolidinone Derivative ◽  
Histamine H3
Sign in / Sign up

Export Citation Format

Share Document