Dicarboxylic Acid Azacyclel-Prolyl-pyrrolidine Amides as Prolyl Oligopeptidase Inhibitors and Three-Dimensional Quantitative Structure−Activity Relationship of the Enzyme−Inhibitor Interactions

Elina M. Jarho; Erik A. A. Wallén; Johannes A. M. Christiaans; Markus M. Forsberg; Jarkko I. Venäläinen; Pekka T. Männistö; Jukka Gynther; Antti Poso

doi:10.1021/jm0500020

Dicarboxylic Acid Azacyclel-Prolyl-pyrrolidine Amides as Prolyl Oligopeptidase Inhibitors and Three-Dimensional Quantitative Structure−Activity Relationship of the Enzyme−Inhibitor Interactions

Journal of Medicinal Chemistry ◽

10.1021/jm0500020 ◽

2005 ◽

Vol 48 (15) ◽

pp. 4772-4782 ◽

Cited By ~ 7

Author(s):

Elina M. Jarho ◽

Erik A. A. Wallén ◽

Johannes A. M. Christiaans ◽

Markus M. Forsberg ◽

Jarkko I. Venäläinen ◽

...

Keyword(s):

Dicarboxylic Acid ◽

Enzyme Inhibitor ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Prolyl Oligopeptidase ◽

Structure Activity ◽

Relationship Of

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Cytotoxic Activity and Three-Dimensional Quantitative Structure Activity Relationship of 2-Aryl-1,8-naphthyridin-4-ones

Korean Journal of Physiology and Pharmacology ◽

10.4196/kjpp.2009.13.6.511 ◽

2009 ◽

Vol 13 (6) ◽

pp. 511 ◽

Cited By ~ 2

Author(s):

Yong Jin Kim ◽

Eun Ae Kim ◽

Mi Lyang Chung ◽

Chaeuk Im

Keyword(s):

Cytotoxic Activity ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Study on the Three-dimensional Quantitative Structure-activity Relationship of Pyridazinonyl-substituted 1,3,4-Thiadiazoles

Chinese Journal of Chemistry ◽

10.1002/cjoc.200591120 ◽

2005 ◽

Vol 23 (8) ◽

pp. 1120-1122 ◽

Cited By ~ 4

Author(s):

Zou Xia-Juan ◽

Lai Lu-Hua ◽

Jin Gui-Yu

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Three-Dimensional Quantitative Structure-Activity Relationship of ArylalkylamineN-acetyltransferase (AANAT) Inhibitors: A Comparative Molecular Field Analysis

Quantitative Structure-Activity Relationships ◽

10.1002/1521-3838(200112)20:5/6<414::aid-qsar414>3.0.co;2-v ◽

2001 ◽

Vol 20 (5-6) ◽

pp. 414-421 ◽

Cited By ~ 2

Author(s):

Philippe Chavatte ◽

Saïd Yous ◽

Nathalie Beaurain ◽

Christophe Mésangeau ◽

Gilles Ferry ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Field Analysis ◽

Molecular Field ◽

Activity Relationship ◽

Comparative Molecular Field Analysis ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Three Dimensional Quantitative Structure-Activity Relationship of 5H-Pyrido[4,3-b]indol-4-carboxamide JAK2 Inhibitors

International Journal of Molecular Sciences ◽

10.3390/ijms140612037 ◽

2013 ◽

Vol 14 (6) ◽

pp. 12037-12053 ◽

Cited By ~ 2

Author(s):

Xiaoyun Wu ◽

Shanhe Wan ◽

Jiajie Zhang

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of ◽

Jak2 Inhibitors

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Three-Dimensional Quantitative Structure−Activity Relationship of 1,4-Dihydropyridines As Antitubercular Agents

Journal of Medicinal Chemistry ◽

10.1021/jm020217z ◽

2002 ◽

Vol 45 (22) ◽

pp. 4858-4867 ◽

Cited By ~ 68

Author(s):

Prashant S. Kharkar ◽

Bhavik Desai ◽

Harsukh Gaveria ◽

Bharat Varu ◽

Rajesh Loriya ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Antitubercular Agents ◽

Structure Activity ◽

Relationship Of

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Three-Dimensional Quantitative Structure—Activity Relationship of Nucleosides Acting at the A3 Adenosine Receptor: Analysis of Binding and Relative Efficacy.

ChemInform ◽

10.1002/chin.200734215 ◽

2007 ◽

Vol 38 (34) ◽

Author(s):

Soo-Kyung Kim ◽

Kenneth A. Jacobson

Keyword(s):

Adenosine Receptor ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Relative Efficacy ◽

Quantitative Structure ◽

Structure Activity ◽

A3 Adenosine Receptor ◽

Relationship Of

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Three-Dimensional Quantitative Structure−Activity Relationship of Nucleosides Acting at the A3 Adenosine Receptor: Analysis of Binding and Relative Efficacy

Journal of Chemical Information and Modeling ◽

10.1021/ci600501z ◽

2007 ◽

Vol 47 (3) ◽

pp. 1225-1233 ◽

Cited By ~ 10

Author(s):

Soo-Kyung Kim ◽

Kenneth A. Jacobson

Keyword(s):

Adenosine Receptor ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Relative Efficacy ◽

Quantitative Structure ◽

Structure Activity ◽

A3 Adenosine Receptor ◽

Relationship Of

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Three-dimensional holographic vector of atomic interaction field for quantitative structure–activity relationship of Aza-bioisosteres of anthrapyrazoles (Aza-APs)

Journal of Molecular Graphics and Modelling ◽

10.1016/j.jmgm.2007.11.007 ◽

2008 ◽

Vol 26 (8) ◽

pp. 1252-1258 ◽

Cited By ~ 3

Author(s):

Xu Luo-nan ◽

Liang Gui-Zhao ◽

Li Zhi-liang ◽

Wang Juan ◽

Zhou Peng

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Atomic Interaction ◽

Quantitative Structure ◽

Interaction Field ◽

Structure Activity ◽

Relationship Of

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Study on Three Dimensional Quantitative Structure Activity Relationship of Benzodiazepines

Hans Journal of Medicinal Chemistry ◽

10.12677/hjmce.2016.44004 ◽

2016 ◽

Vol 04 (04) ◽

pp. 25-37 ◽

Cited By ~ 1

Author(s):

华军何

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Structure Activity ◽

Relationship Of

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Three-dimensional quantitative structure–activity relationship of 4,5,6,7-tetrahydrothienopyridines analogues as glucose-6-phosphatase inhibitors

Journal of Molecular Structure ◽

10.1016/j.molstruc.2004.12.041 ◽

2006 ◽

Vol 782 (1) ◽

pp. 49-54

Author(s):

Chong Wang ◽

Ling Yang ◽

Sheng-Li Yang

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Phosphatase Inhibitors ◽

Structure Activity ◽

Relationship Of

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