Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2at the Mouse Melanocortin Receptors. 4. Modifications at the Trp Position

Jerry Ryan Holder; Zhimin Xiang; Rayna M. Bauzo; Carrie Haskell-Luevano

doi:10.1021/jm020296e

Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2at the Mouse Melanocortin Receptors. 4. Modifications at the Trp Position

Journal of Medicinal Chemistry ◽

10.1021/jm020296e ◽

2002 ◽

Vol 45 (26) ◽

pp. 5736-5744 ◽

Cited By ~ 37

Author(s):

Jerry Ryan Holder ◽

Zhimin Xiang ◽

Rayna M. Bauzo ◽

Carrie Haskell-Luevano

Keyword(s):

Melanocortin Receptors ◽

Structure Activity Relationships ◽

Structure Activity

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Structure–Activity Relationships of Peptides Incorporating a Bioactive Reverse-Turn Heterocycle at the Melanocortin Receptors: Identification of a 5800-fold Mouse Melanocortin-3 Receptor (mMC3R) Selective Antagonist/Partial Agonist versus the Mouse Melanocortin-4 Receptor (mMC4R)

Journal of Medicinal Chemistry ◽

10.1021/jm301253y ◽

2013 ◽

Vol 56 (7) ◽

pp. 2747-2763 ◽

Cited By ~ 6

Author(s):

Anamika Singh ◽

Marvin Dirain ◽

Rachel Witek ◽

James R. Rocca ◽

Arthur S. Edison ◽

...

Keyword(s):

Partial Agonist ◽

Melanocortin Receptors ◽

Selective Antagonist ◽

Structure Activity Relationships ◽

Structure Activity ◽

Melanocortin 4 Receptor ◽

Reverse Turn

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The Molecular Pharmacology of Alpha-Melanocyte Stimulating Hormone: Structure-Activity Relationships for Melanotropins at Melanocortin Receptors

Melanocortin Receptors, The ◽

10.1385/1-59259-031-4:239 ◽

2003 ◽

pp. 239-261 ◽

Cited By ~ 2

Author(s):

Victor J. Hruby ◽

Guoxia Han

Keyword(s):

Melanocortin Receptors ◽

Molecular Pharmacology ◽

Structure Activity Relationships ◽

Melanocyte Stimulating Hormone ◽

Structure Activity ◽

Stimulating Hormone

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Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH2at the Mouse Melanocortin Receptors: Part 2 Modifications at the Phe Position

Journal of Medicinal Chemistry ◽

10.1021/jm010524p ◽

2002 ◽

Vol 45 (14) ◽

pp. 3073-3081 ◽

Cited By ~ 52

Author(s):

Jerry Ryan Holder ◽

Rayna M. Bauzo ◽

Zhimin Xiang ◽

Carrie Haskell-Luevano

Keyword(s):

Melanocortin Receptors ◽

Structure Activity Relationships ◽

Structure Activity

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Comparative Functional Alanine Positional Scanning of the α-Melanocyte Stimulating Hormone and NDP-Melanocyte Stimulating Hormone Demonstrates Differential Structure–Activity Relationships at the Mouse Melanocortin Receptors

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.6b00098 ◽

2016 ◽

Vol 7 (7) ◽

pp. 984-994 ◽

Cited By ~ 3

Author(s):

Aleksandar Todorovic ◽

Mark D. Ericson ◽

Ryan D. Palusak ◽

Nicholas B. Sorensen ◽

Michael S. Wood ◽

...

Keyword(s):

Melanocortin Receptors ◽

Structure Activity Relationships ◽

Melanocyte Stimulating Hormone ◽

Differential Structure ◽

Structure Activity ◽

Positional Scanning ◽

Stimulating Hormone

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Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH2at the Mouse Melanocortin Receptors. 1. Modifications at the His Position

Journal of Medicinal Chemistry ◽

10.1021/jm0104872 ◽

2002 ◽

Vol 45 (13) ◽

pp. 2801-2810 ◽

Cited By ~ 43

Author(s):

Jerry Ryan Holder ◽

Rayna M. Bauzo ◽

Zhimin Xiang ◽

Carrie Haskell-Luevano

Keyword(s):

Melanocortin Receptors ◽

Structure Activity Relationships ◽

Structure Activity

Download Full-text