2-Phenylindoles. Effect of N-benzylation on estrogen receptor affinity, estrogenic properties, and mammary tumor inhibiting activity

Erwin Von Angerer; Josef Strohmeier

doi:10.1021/jm00384a022

2-Phenylindoles. Effect of N-benzylation on estrogen receptor affinity, estrogenic properties, and mammary tumor inhibiting activity

Journal of Medicinal Chemistry ◽

10.1021/jm00384a022 ◽

1987 ◽

Vol 30 (1) ◽

pp. 131-136 ◽

Cited By ~ 40

Author(s):

Erwin Von Angerer ◽

Josef Strohmeier

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity ◽

Estrogenic Properties

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ChemInform Abstract: 2-Phenylindoles. Effect of N-Benzylation on Estrogen Receptor Affinity, Estrogenic Properties, and Mammary Tumor Inhibiting Activity.

ChemInform ◽

10.1002/chin.198724194 ◽

1987 ◽

Vol 18 (24) ◽

Author(s):

E. VON ANGERER ◽

J. STROHMEIER

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity ◽

Estrogenic Properties

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2-Alkyl-substituted 1,1-bis(4-acetoxyphenyl)-2-phenylethenes. Estrogen receptor affinity, estrogenic and antiestrogenic properties, and mammary tumor inhibiting activity

Journal of Medicinal Chemistry ◽

10.1021/jm00158a029 ◽

1986 ◽

Vol 29 (8) ◽

pp. 1494-1498 ◽

Cited By ~ 21

Author(s):

Martin R. Schneider

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity

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ChemInform Abstract: 2-Alkyl Substituted 1,1-Bis(4-acetoxyphenyl)-2-phenylethenes. Estrogen Receptor Affinity, Estrogenic and Antiestrogenic Properties, and Mammary Tumor Inhibiting Activity.

ChemInform ◽

10.1002/chin.198703156 ◽

1987 ◽

Vol 18 (3) ◽

Author(s):

M. R. SCHNEIDER

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity

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ChemInform Abstract: 2-PHENYLINDOLES. RELATIONSHIP BETWEEN STRUCTURE, ESTROGEN RECEPTOR AFFINITY, AND MAMMARY TUMOR INHIBITING ACTIVITY IN THE RAT

Chemischer Informationsdienst ◽

10.1002/chin.198512186 ◽

1985 ◽

Vol 16 (12) ◽

Author(s):

E. VON ANGERER ◽

J. PREKAJAC ◽

J. STROHMEIER

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity

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2-Phenylindoles. Relationship between structure, estrogen receptor affinity, and mammary tumor inhibiting activity in the rat

Journal of Medicinal Chemistry ◽

10.1021/jm00377a011 ◽

1984 ◽

Vol 27 (11) ◽

pp. 1439-1447 ◽

Cited By ~ 89

Author(s):

Erwin Von Angerer ◽

Jelica Prekajac ◽

Josef Strohmeier

Keyword(s):

Estrogen Receptor ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Affinity ◽

Estrogen Receptor Affinity

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Ring-substituted 1,1,2,2-tetraalkylated 1,2-bis(hydroxyphenyl)ethanes. 4. Synthesis, estrogen receptor binding affinity, and evaluation of antiestrogenic and mammary tumor inhibiting activity of symmetrically disubstituted 1,1,2,2-tetramethyl-1,2-bis(hydroxyphenyl)ethanes

Journal of Medicinal Chemistry ◽

10.1021/jm00147a031 ◽

1985 ◽

Vol 28 (9) ◽

pp. 1295-1301 ◽

Cited By ~ 16

Author(s):

Rolf W. Hartmann ◽

Walter Schwarz ◽

Alexander Heindl ◽

Helmut Schoenenberger

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Binding Affinity ◽

Estrogen Receptor Binding

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2-Hydroxyestradiol-17α and 4-hydroxyestradiol-17α, catechol estrogfn analogs with reduced estrogen receptor affinity

Steroids ◽

10.1016/0039-128x(80)90063-x ◽

1980 ◽

Vol 36 (1) ◽

pp. 13-20 ◽

Cited By ~ 26

Author(s):

George R. Merriam ◽

Neil J. MacLusky ◽

Leslie A. Johnson ◽

Frederick Naftolin

Keyword(s):

Estrogen Receptor ◽

Receptor Affinity ◽

Estrogen Receptor Affinity

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Estrogen receptor affinity and effects on MCF-7 cell growth of triarylethylene carboxylic acids related to tamoxifen

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/0960-0760(92)90452-o ◽

1992 ◽

Vol 42 (6) ◽

pp. 613-616 ◽

Cited By ~ 5

Author(s):

Susanne Wilson ◽

Peter C. Ruenitz ◽

Jan A. Ruzicka

Keyword(s):

Estrogen Receptor ◽

Cell Growth ◽

Carboxylic Acids ◽

Receptor Affinity ◽

Estrogen Receptor Affinity ◽

Mcf 7

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ChemInform Abstract: RING-SUBSTITUTED 1,1,2,2-TETRAALKYLATED 1,2-BIS(HYDROXYPHENYL)ETHANES. 4. SYNTHESIS, ESTROGEN RECEPTOR BINDING AFFINITY, AND EVALUATION OF ANTIESTROGENIC AND MAMMARY TUMOR INHIBITING ACTIVITY OF SYMMETRICALLY DISUBSTITUTED 1,1,2,2-TET

Chemischer Informationsdienst ◽

10.1002/chin.198552194 ◽

1985 ◽

Vol 16 (52) ◽

Author(s):

R. W. HARTMANN ◽

W. SCHWARZ ◽

A. HEINDL ◽

H. SCHOENENBERGER

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Binding Affinity ◽

Estrogen Receptor Binding

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ChemInform Abstract: RING-SUBSTITUTED 1,2-DIALKYLATED 1,2-BIS(HYDROXYPHENYL)ETHANES. 3. SYNTHESIS, , ESTROGEN RECEPTOR BINDING AFFINITY, AND EVALUATION OF ANTIESTROGENIC AND MAMMARY TUMOR INHIBITING ACTIVITY OF 2,2′-DISUBSTITUTED BUTESTROLS AND 6,6′-DISUB

Chemischer Informationsdienst ◽

10.1002/chin.198448165 ◽

1984 ◽

Vol 15 (48) ◽

Author(s):

R. W. HARTMANN ◽

A. HEINDL ◽

W. SCHWARZ ◽

H. SCHOENENBERGER

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Receptor Binding Affinity ◽

Estrogen Receptor Binding

Download Full-text