1,2,5-Thiadizole 1-oxide and 1,1-dioxide derivatives. A new class of potent histamine H2-receptor antagonists

Aldo A. Algieri; George M. Luke; Robert T. Standridge; Myron Brown; Richard A. Partyka; R. R. Crenshaw

doi:10.1021/jm00345a003

1,2,5-Thiadizole 1-oxide and 1,1-dioxide derivatives. A new class of potent histamine H2-receptor antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm00345a003 ◽

1982 ◽

Vol 25 (3) ◽

pp. 210-212 ◽

Cited By ~ 41

Author(s):

Aldo A. Algieri ◽

George M. Luke ◽

Robert T. Standridge ◽

Myron Brown ◽

Richard A. Partyka ◽

...

Keyword(s):

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

New Class

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ChemInform Abstract: 1,2,5-THIADIZOLE 1-OXIDE AND 1,1-DIOXIDE DERIVATIVES. A NEW CLASS OF POTENT HISTAMINE H2-RECEPTOR ANTAGONISTS

Chemischer Informationsdienst ◽

10.1002/chin.198233185 ◽

1982 ◽

Vol 13 (33) ◽

Author(s):

A. A. ALGIERI ◽

G. M. LUKE ◽

R. T. STANDRIDGE ◽

M. BROWN ◽

R. A. PARTYKA ◽

...

Keyword(s):

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

New Class

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Drugs from emasculated hormones: The principle of syntopic antagonism

Bioscience Reports ◽

10.1007/bf01114681 ◽

1989 ◽

Vol 9 (3) ◽

pp. 253-272 ◽

Cited By ~ 6

Author(s):

James Black

Keyword(s):

Future Research ◽

Receptor Antagonists ◽

Personal View ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

Early Stages ◽

Β Receptor

This lecture outlines the early stages in the discovery of adrenaline β-receptor antagonists and of the histamine H2-receptor antagonists. It ends with a brief personal view about future research.

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ChemInform Abstract: CRYSTAL AND MOLECULAR STRUCTURE OF HISTAMINE H2-RECEPTOR ANTAGONISTS OF THE RANITIDINE FAMILY. PART 1. 1-(5-DIMETHYLAMINOMETHYL)FURFURYLTHIOPROPAN-2-ONE THIOSEMICARBAZONE AND 1-(5-DIMETHYLAMINOMETHYL)FURFURYLTHIOPROPAN-2-ONE 1-METHYLA

Chemischer Informationsdienst ◽

10.1002/chin.198411063 ◽

1984 ◽

Vol 15 (11) ◽

Author(s):

G. CHIARI ◽

D. VITERBO

Keyword(s):

Molecular Structure ◽

Crystal And Molecular Structure ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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Effect of some new histamine H2-receptor antagonists on the guinea pig papillary muscle *1G. Bertaccini and G. Coruzzi. Institute of Pharmacology, University of Parma, Faculty of Medicine, Parma, Italy

Journal of Molecular and Cellular Cardiology ◽

10.1016/0022-2828(81)90017-1 ◽

1981 ◽

Vol 13 ◽

pp. 8

Keyword(s):

Guinea Pig ◽

Papillary Muscle ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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Inhibition of gastric alcohol dehydrogenase activity by histamine H2- receptor antagonists has no influence on the pharmacokinetics of ethanol after a moderate dose.

British Journal of Clinical Pharmacology ◽

10.1111/j.1365-2125.1994.tb04263.x ◽

1994 ◽

Vol 37 (2) ◽

pp. 208-211 ◽

Cited By ~ 10

Author(s):

A Mallat ◽

F Roudot-Thoraval ◽

JF Bergmann ◽

H Trout ◽

G Simonneau ◽

...

Keyword(s):

Alcohol Dehydrogenase ◽

Dehydrogenase Activity ◽

Moderate Dose ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

Alcohol Dehydrogenase Activity ◽

Gastric Alcohol Dehydrogenase

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(Imidazolylphenyl)formamidines. A structurally novel class of potent histamine H2 receptor antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm00369a025 ◽

1984 ◽

Vol 27 (3) ◽

pp. 380-386 ◽

Cited By ~ 42

Author(s):

Arturo Donetti ◽

Enzo Cereda ◽

Elio Bellora ◽

Alberto Gallazzi ◽

Cesare Bazzano ◽

...

Keyword(s):

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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Histamine H2 receptor antagonists and blood alcohol levels

Digestive Diseases and Sciences ◽

10.1007/bf01540445 ◽

1988 ◽

Vol 33 (6) ◽

pp. 767-768 ◽

Cited By ~ 7

Author(s):

G. Holtmann ◽

M. V. Singer

Keyword(s):

Blood Alcohol ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor ◽

Blood Alcohol Levels

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Radioprotective Effects of Histamine H2 Receptor Antagonists Famotidine and Ranitidine on Gamma-Ray Induced Chromosome Aberration and Micronuclei <i>in vitro</i> in Human Lymphocytes

American Journal of BioScience ◽

10.11648/j.ajbio.20150306.17 ◽

2015 ◽

Vol 3 (6) ◽

pp. 249

Author(s):

Narinder Kumar Sharma

Keyword(s):

Chromosome Aberration ◽

Gamma Ray ◽

Human Lymphocytes ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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LONG-TERM EFFECTS OF HISTAMINE H2-RECEPTOR ANTAGONISTS ON SERUM PARATHYROID HORMONE IN CHRONIC RENAL FAILURE

Clinical Endocrinology ◽

10.1111/j.1365-2265.1985.tb00224.x ◽

1985 ◽

Vol 23 (3) ◽

pp. 277-282 ◽

Cited By ~ 3

Author(s):

C. E. FIORE ◽

M. LUNETTA ◽

J. A. KANIS

Keyword(s):

Renal Failure ◽

Parathyroid Hormone ◽

Chronic Renal Failure ◽

Long Term Effects ◽

Serum Parathyroid Hormone ◽

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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Potential Histamine H2-Receptor Antagonists: Ranitidine Analogues Containing “Semicarbazono Equivalent” Groups

Archiv der Pharmazie ◽

10.1002/ardp.19843170604 ◽

1984 ◽

Vol 317 (6) ◽

pp. 496-501 ◽

Cited By ~ 6

Author(s):

Giovanni Sorba ◽

Roberta Fruttero ◽

Rosella Calvino ◽

Alberto Gasco ◽

Marco Orsetti

Keyword(s):

Receptor Antagonists ◽

H2 Receptor Antagonists ◽

Histamine H2 Receptor ◽

H2 Receptor

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