Conformationally restricted analogs of histamine H1 receptor antagonists, trans- and cis-1-benzyl-3-dimethylamino-6-phenylpiperidine

Ahmed E. Ahmed; Patrick E. Hanna; Vernon R. Grund

doi:10.1021/jm00223a020

Conformationally restricted analogs of histamine H1 receptor antagonists, trans- and cis-1-benzyl-3-dimethylamino-6-phenylpiperidine

Journal of Medicinal Chemistry ◽

10.1021/jm00223a020 ◽

1976 ◽

Vol 19 (1) ◽

pp. 117-122 ◽

Cited By ~ 5

Author(s):

Ahmed E. Ahmed ◽

Patrick E. Hanna ◽

Vernon R. Grund

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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Conformationally restricted analogs of histamine H1 receptor antagonists. 2-Phenyl- and 2-benzyl-1,2,3,4-tetrahydro-4-dimethylaminoisoquinoline

Journal of Medicinal Chemistry ◽

10.1021/jm00255a027 ◽

1974 ◽

Vol 17 (9) ◽

pp. 1020-1023 ◽

Cited By ~ 11

Author(s):

Patrick E. Hanna ◽

Vernon R. Grund ◽

M. W. Anders

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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Conformationally restricted analogs of histamine H1 receptor antagonists. trans- and cis-1,5-Diphenyl-3-dimethylaminopyrrolidine

Journal of Medicinal Chemistry ◽

10.1021/jm00267a001 ◽

1973 ◽

Vol 16 (9) ◽

pp. 963-968 ◽

Cited By ~ 12

Author(s):

Patrick E. Hanna ◽

Ahmed E. Ahmed

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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ChemInform Abstract: CONFORMATIONALLY RESTRICTED ANALOGS OF HISTAMINE H1 RECEPTOR ANTAGONISTS, TRANS- AND CIS-1-BENZYL-3-DIMETHYLAMINO-6-PHENYLPIPERIDINE

Chemischer Informationsdienst ◽

10.1002/chin.197617235 ◽

1976 ◽

Vol 7 (17) ◽

pp. no-no

Author(s):

A. E. AHMED ◽

P. E. HANNA ◽

V. R. GRUND

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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ChemInform Abstract: CONFORMATIONALLY RESTRICTED ANALOGS OF HISTAME H1 RECEPTOR ANTAGONISTS, 2-PHENYL- AND 2-BENZYL-1,2,3,4-TETRAHYDRO-4-DIMETHYLAMINOISOQUINOLINE

Chemischer Informationsdienst ◽

10.1002/chin.197501282 ◽

1975 ◽

Vol 6 (1) ◽

pp. no-no

Author(s):

P. E. HANNA ◽

V. R. GRUND ◽

M. W. ANDERS

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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ChemInform Abstract: CONFORMATIONALLY RESTRICTED ANALOGS OF HISTAMIN H1 RECEPTOR ANTAGONISTS, TRANS- AND CIS-1,5-DIPHENYL-3-DIMETHYLAMINOPYRROLIDINE

Chemischer Informationsdienst ◽

10.1002/chin.197351248 ◽

1973 ◽

Vol 4 (51) ◽

pp. no-no

Author(s):

P. E. HANNA ◽

A. E. AHMED

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Conformationally Restricted ◽

Conformationally Restricted Analogs

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Histamine H1-Receptor Antagonists, Promethazine and Homochlorcyclizine, Increase the Steady-State Plasma Concentrations of Haloperidol and Reduced Haloperidol

Therapeutic Drug Monitoring ◽

10.1097/00007691-200304000-00008 ◽

2003 ◽

Vol 25 (2) ◽

pp. 192-196 ◽

Cited By ~ 11

Author(s):

Akihito Suzuki ◽

Norio Yasui-Furukori ◽

Kazuo Mihara ◽

Tsuyoshi Kondo ◽

Hanako Furukori ◽

...

Keyword(s):

Steady State ◽

Plasma Concentrations ◽

H1 Receptor ◽

Receptor Antagonists ◽

Reduced Haloperidol ◽

Histamine H1 Receptor ◽

State Plasma

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Design of Phthalazinone Amide Histamine H1 Receptor Antagonists for Use in Rhinitis

ACS Medicinal Chemistry Letters ◽

10.1021/acsmedchemlett.7b00112 ◽

2017 ◽

Vol 8 (5) ◽

pp. 577-581 ◽

Cited By ~ 8

Author(s):

Panayiotis A. Procopiou ◽

Alison J. Ford ◽

Paul M. Gore ◽

Brian E. Looker ◽

Simon T. Hodgson ◽

...

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor

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Molecular Determinants Responsible for Sedative and Non-sedative Properties of Histamine H1–Receptor Antagonists

Journal of Pharmacological Sciences ◽

10.1254/jphs.13169fp ◽

2014 ◽

Vol 124 (2) ◽

pp. 160-168 ◽

Cited By ~ 5

Author(s):

Yoshihiro Uesawa ◽

Shigeru Hishinuma ◽

Masaru Shoji

Keyword(s):

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Molecular Determinants

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ChemInform Abstract: Indole Amide Derivatives: Synthesis, Structure-Activity Relationships, and Molecular Modeling Studies of a New Series of Histamine H1-Receptor Antagonists.

ChemInform ◽

10.1002/chin.199929124 ◽

2010 ◽

Vol 30 (29) ◽

pp. no-no

Author(s):

Sandra Battaglia ◽

Enrico Boldrini ◽

Federico Da Settimo ◽

Giulio Dondio ◽

Concettina La Motta ◽

...

Keyword(s):

Molecular Modeling ◽

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Structure Activity Relationships ◽

Structure Activity ◽

Modeling Studies ◽

Amide Derivatives ◽

Molecular Modeling Studies

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Anti-Inflammatory Actions of Histamine H1 Receptor Antagonists Unrelated to H1 Receptor Blockade

Clinical Immunotherapeutics ◽

10.1007/bf03259340 ◽

1996 ◽

Vol 5 (6) ◽

pp. 449-464 ◽

Cited By ~ 3

Author(s):

Claus Kroegel ◽

Verena Herzog ◽

Birgit Knöchel ◽

Peter Julius ◽

Dirk Wagnetz ◽

...

Keyword(s):

Receptor Blockade ◽

H1 Receptor ◽

Receptor Antagonists ◽

Histamine H1 Receptor ◽

Anti Inflammatory

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