.alpha.-Diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases

Michael R. Angelastro; Shujaath Mehdi; Joseph P. Burkhart; Norton P. Peet; Philippe Bey

doi:10.1021/jm00163a002

.alpha.-Diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides as novel inhibitors of cysteine and serine proteinases

Journal of Medicinal Chemistry ◽

10.1021/jm00163a002 ◽

1990 ◽

Vol 33 (1) ◽

pp. 11-13 ◽

Cited By ~ 95

Author(s):

Michael R. Angelastro ◽

Shujaath Mehdi ◽

Joseph P. Burkhart ◽

Norton P. Peet ◽

Philippe Bey

Keyword(s):

Amino Acids ◽

Serine Proteinases ◽

Keto Ester ◽

Derivatives Of

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An efficient synthesis of novel .alpha.-diketone and .alpha.-keto ester derivatives of N-protected amino acids and peptides

The Journal of Organic Chemistry ◽

10.1021/jo00277a031 ◽

1989 ◽

Vol 54 (16) ◽

pp. 3913-3916 ◽

Cited By ~ 51

Author(s):

Michael R. Angelastro ◽

Norton P. Peet ◽

Philippe Bey

Keyword(s):

Amino Acids ◽

Efficient Synthesis ◽

Keto Ester ◽

Derivatives Of

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ChemInform Abstract: An Efficient Synthesis of Novel α-Diketone and α-Keto Ester Derivatives of N-Protected Amino Acids and Peptides.

ChemInform ◽

10.1002/chin.199003279 ◽

1990 ◽

Vol 21 (3) ◽

Author(s):

M. R. ANGELASTRO ◽

N. P. PEET ◽

P. BEY

Keyword(s):

Amino Acids ◽

Efficient Synthesis ◽

Keto Ester ◽

Derivatives Of

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Substances with antineoplastic activity. LIII. N-{δ-(4-pyrrolo[2,3-d]pyrimidinylthio)valeryl}amino acids and analogous derivatives of di- and triglycine

Collection of Czechoslovak Chemical Communications ◽

10.1135/cccc19731438 ◽

1973 ◽

Vol 38 (5) ◽

pp. 1438-1444 ◽

Cited By ~ 1

Author(s):

R. Kotva ◽

A. Černý ◽

M. Semonský

Keyword(s):

Amino Acids ◽

Antineoplastic Activity ◽

Derivatives Of

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AROMATIC ALDEHYDE DERIVATIVES OF PROTEINS, PEPTIDES, AND AMINO ACIDS

Journal of Biological Chemistry ◽

10.1016/s0021-9258(18)77023-3 ◽

1929 ◽

Vol 84 (2) ◽

pp. 675-682

Author(s):

H.D. Dakin

Keyword(s):

Amino Acids ◽

Aromatic Aldehyde ◽

Derivatives Of

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Derivatives of aminoquinones with N-protected amino acids

Letters in Peptide Science ◽

10.1007/bf02443542 ◽

1998 ◽

Vol 5 (4) ◽

pp. 259-262 ◽

Cited By ~ 4

Author(s):

Chrysostomos Pachatouridis ◽

Elias A. Couladouros ◽

Vassilios P. Papageorgiou ◽

Maria Liakopoulou-Kyriakides

Keyword(s):

Amino Acids ◽

Derivatives Of

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ChemInform Abstract: Derivatives of β-(Trimethylsilyl)alanine with SiCH2NH2, SiCH2OH, or SiCH2SH Functionality: Synthesis of the Silicon-Containing α-Amino Acids rac- and (R)-Me2Si(CH2R)CH2CH(NH2)COOH (R: NH2, OH, SH).

ChemInform ◽

10.1002/chin.200242213 ◽

2010 ◽

Vol 33 (42) ◽

pp. no-no

Author(s):

Reinhold Tacke ◽

Vera I. Handmann

Keyword(s):

Amino Acids ◽

Derivatives Of

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Pentacarbonyl complexes of tungsten with derivatives of amino acids

Bulletin of the Academy of Sciences of the USSR Division of Chemical Science ◽

10.1007/bf00956560 ◽

1984 ◽

Vol 33 (7) ◽

pp. 1539-1539

Author(s):

A. A. Ioganson ◽

Yu. G. Kovalev ◽

L. L. Milovanova

Keyword(s):

Amino Acids ◽

Derivatives Of

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Thin-layer and paper chromatography of dinitrophenyl derivatives of amino acids from bacterial cell wall peptidoglycans

Journal of Chromatography A ◽

10.1016/0021-9673(70)80019-x ◽

1970 ◽

Vol 47 ◽

pp. 124-126 ◽

Cited By ~ 3

Author(s):

W.D. Grant ◽

A.J. Wicken

Keyword(s):

Amino Acids ◽

Cell Wall ◽

Thin Layer ◽

Paper Chromatography ◽

Bacterial Cell ◽

Bacterial Cell Wall ◽

Derivatives Of

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Effects of N-uronoyl derivatives of neurotransmitter amino acids on rats under conditions of behavioral tests

Neurophysiology ◽

10.1007/s11062-007-0008-7 ◽

2007 ◽

Vol 39 (1) ◽

pp. 48-56

Author(s):

I. I. Korenyuk ◽

M. Yu. Ravayeva

Keyword(s):

Amino Acids ◽

Behavioral Tests ◽

Neurotransmitter Amino Acids ◽

Derivatives Of

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ChemInform Abstract: SUBSTANCES WITH ANTINEOPLASTIC ACTIVITY PART 53, N-(DELTA-(4-PYRROLO(2,3-D)PYRIMIDINYLTHIO)-VALERYL)-AMINO ACIDS AND ANALOGOUS DERIVATIVES OF DI- AND TRIGLYCINE

Chemischer Informationsdienst ◽

10.1002/chin.197334294 ◽

1973 ◽

Vol 4 (34) ◽

pp. no-no

Author(s):

R. KOTVA ◽

A. CERNY ◽

M. SEMONSKY

Keyword(s):

Amino Acids ◽

Antineoplastic Activity ◽

Derivatives Of

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