Syntheses and in vitro evaluation of 4-(2-aminoethyl)-2(3H)-indolones and related compounds as peripheral prejunctional dopamine receptor agonists

Robert M. DeMarinis; Ralph F. Hall; Robert G. Franz; Charles Webster; William F. Huffman; Mark S. Schwartz; Carl Kaiser; Stephen T. Ross; Gregory Gallagher

doi:10.1021/jm00156a010

Syntheses and in vitro evaluation of 4-(2-aminoethyl)-2(3H)-indolones and related compounds as peripheral prejunctional dopamine receptor agonists

Journal of Medicinal Chemistry ◽

10.1021/jm00156a010 ◽

1986 ◽

Vol 29 (6) ◽

pp. 939-947 ◽

Cited By ~ 22

Author(s):

Robert M. DeMarinis ◽

Ralph F. Hall ◽

Robert G. Franz ◽

Charles Webster ◽

William F. Huffman ◽

...

Keyword(s):

Dopamine Receptor ◽

In Vitro Evaluation ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Related Compounds

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ChemInform Abstract: Syntheses and in vitro Evaluation of 4-(2-Aminoethyl)-2(3H)-indolones and Related Compounds as Peripheral Prejunctional Dopamine Receptor Agonists.

Chemischer Informationsdienst ◽

10.1002/chin.198643149 ◽

1986 ◽

Vol 17 (43) ◽

Author(s):

R. M. DEMARINIS ◽

G. JUN. GALLAGHER ◽

R. F. HALL ◽

R. G. FRANZ ◽

C. WEBSTER ◽

...

Keyword(s):

Dopamine Receptor ◽

In Vitro Evaluation ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Related Compounds

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The role of dopamine pathway on human sperm: in vitro effect of dopamine receptor agonists and antagonists on sperm motility, kinetics and viability

Endocrine Abstracts ◽

10.1530/endoabs.41.ep712 ◽

2016 ◽

Author(s):

Angelis Cristina de ◽

Federica Cariati ◽

Giacomo Galdiero ◽

Giorgio Coppola ◽

Mariano Galdiero ◽

...

Keyword(s):

Dopamine Receptor ◽

Sperm Motility ◽

Human Sperm ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Vitro Effect ◽

Receptor Agonists And Antagonists

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3-PPP antagonizes the in vitro effects of D-1 and D-2 dopamine receptor agonists in rat neostriatum

European Journal of Pharmacology ◽

10.1016/0014-2999(83)90486-7 ◽

1983 ◽

Vol 91 (2-3) ◽

pp. 317-320 ◽

Cited By ~ 9

Author(s):

Johan F. Plantjé ◽

Arie H. Mulder ◽

Johannes C. Stoof

Keyword(s):

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

In Vitro Effects

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Effect of dopamine receptor agonists and antagonists on release of dopamine in the rabbit caudate nucleus in vitro

Naunyn-Schmiedeberg s Archives of Pharmacology ◽

10.1007/bf00497003 ◽

1978 ◽

Vol 305 (1) ◽

pp. 27-36 ◽

Cited By ~ 211

Author(s):

K. Starke ◽

W. Reimann ◽

A. Zumstein ◽

G. Hertting

Keyword(s):

Caudate Nucleus ◽

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Rabbit Caudate Nucleus ◽

Receptor Agonists And Antagonists

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Characterization of dopamine autoreceptor and [3H]spiperone binding sites in vitro with classical and novel dopamine receptor agonists

European Journal of Pharmacology ◽

10.1016/0014-2999(83)90387-4 ◽

1983 ◽

Vol 88 (1) ◽

pp. 11-26 ◽

Cited By ~ 109

Author(s):

John Lehmann ◽

Michael Briley ◽

Salamon Z. Langer

Keyword(s):

Dopamine Receptor ◽

Binding Sites ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Dopamine Autoreceptor

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ChemInform Abstract: A Molecular Mechanics Approach to the Understanding of Presynaptic Selectivity for Centrally Acting Dopamine Receptor Agonists of the Phenylpiperidine Series.

ChemInform ◽

10.1002/chin.198711340 ◽

1987 ◽

Vol 18 (11) ◽

Author(s):

T. LILJEFORS ◽

H. WIKSTROEM

Keyword(s):

Molecular Mechanics ◽

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists

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Dopamine receptor agonists alter gap prestimulus modulation

Psychopharmacology ◽

10.1007/s002130050444 ◽

1997 ◽

Vol 134 (3) ◽

pp. 213-220 ◽

Cited By ~ 4

Author(s):

D. S. Leitner ◽

Eileen M. Girten

Keyword(s):

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists

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On-off effects of dopamine receptor agonists in the hemi-parkinsonian rat

European Journal of Pharmacology ◽

10.1016/0014-2999(93)90006-4 ◽

1993 ◽

Vol 242 (1) ◽

pp. 31-36 ◽

Cited By ~ 12

Author(s):

Peter B. Silverman

Keyword(s):

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists

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Vascular Dopamine and Dopamine Receptor Agonists

Dopamine Receptor Agonists ◽

10.1007/978-1-4757-0310-8_8 ◽

1984 ◽

pp. 195-208 ◽

Cited By ~ 2

Author(s):

Barry A. Berkowitz ◽

Robert Erickson ◽

Bodgan Zabko-Potavpovich ◽

Eliot H. Ohlstein

Keyword(s):

Dopamine Receptor ◽

Dopamine Receptor Agonists ◽

Receptor Agonists

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Discriminative stimulus effects of direct‐ and indirect‐ acting dopamine receptor agonists in free‐feeding and food‐restricted mice.

The FASEB Journal ◽

10.1096/fasebj.27.1_supplement.1098.16 ◽

2013 ◽

Vol 27 (S1) ◽

Author(s):

Gregory T Collins ◽

Jonathan A Jackson ◽

Cedric Henson ◽

Wouter Koek ◽

Charles P France

Keyword(s):

Dopamine Receptor ◽

Discriminative Stimulus ◽

Dopamine Receptor Agonists ◽

Receptor Agonists ◽

Discriminative Stimulus Effects ◽

Stimulus Effects ◽

Free Feeding

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